Molecular Complexity as a Driver for Chemical Process Innovation in the Pharmaceutical Industry von Caille, Seb, Cui, Sheng, Faul, Margaret M, Mennen, Steven M, Tedrow, Jason S, Walker, Shawn D

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The Evolution of High-Throughput Experimentation in Pharmaceutical Development and Perspectives on the Future von Mennen, Steven M, Alhambra, Carolina, Allen, C. Liana, Barberis, Mario, Berritt, Simon, Brandt, Thomas A, Campbell, Andrew D, Castañón, Jesús, Cherney, Alan H, Christensen, Melodie, Damon, David B, Eugenio de Diego, J, García-Cerrada, Susana, García-Losada, Pablo, Haro, Rubén, Janey, Jacob, Leitch, David C, Li, Ling, Liu, Fangfang, Lobben, Paul C, MacMillan, David W. C, Magano, Javier, McInturff, Emma, Monfette, Sebastien, Post, Ronald J, Schultz, Danielle, Sitter, Barbara J, Stevens, Jason M, Strambeanu, Iulia I, Twilton, Jack, Wang, Ke, Zajac, Matthew A

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Enantioselective Total Synthesis of (+)-Gliocladine C: Convergent Construction of Cyclotryptamine-Fused Polyoxopiperazines and a General Approach for Preparing Epidithiodioxopipera... von DeLorbe, John E, Jabri, Salman Y, Mennen, Steven M, Overman, Larry E, Zhang, Fang-Li

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Asymmetric Catalysis Mediated by Synthetic Peptides von Davie, Elizabeth A. Colby, Mennen, Steven M, Xu, Yingju, Miller, Scott J

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General Approach for Preparing Epidithiodioxopiperazines from Trioxopiperazine Precursors: Enantioselective Total Syntheses of (+)- and (−)-Gliocladine C, (+)-Leptosin D, (+)-T988C... von DeLorbe, John E, Horne, David, Jove, Richard, Mennen, Steven M, Nam, Sangkil, Zhang, Fang-Li, Overman, Larry E

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Synthesis of the Hydrazinyl Pyridine Intermediate: Phase-Appropriate Delivery von Wilsily, Ashraf, Mennen, Steven M, Cosbie, Andrew, Milne, Jacqueline E

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Xantphos as a Branch-Selective Ligand for the Acyclic sec-Alkyl Negishi Cross-Coupling of Heteroaryl Halides von Cherney, Alan H, Hedley, Simon J, Mennen, Steven M, Tedrow, Jason S

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Process Development and Protein Engineering Enhanced Nitroreductase-Catalyzed Reduction of 2‑Methyl-5-nitro-pyridine von Bornadel, Amin, Bisagni, Serena, Pushpanath, Ahir, Slabu, Iustina, LePaih, Jacques, Cherney, Alan H, Mennen, Steven M, Hedley, Simon J, Tedrow, Jason, Dominguez, Beatriz

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Synthesis of 4‑Substituted Phthalazin-1(2H)‑ones from 2‑Acylbenzoic Acids: Controlling Hydrazine in a Pharmaceutical Intermediate through PAT-Guided Process Development von Mennen, Steven M, Mak-Jurkauskas, Melody L, Bio, Matthew M, Hollis, L. Steven, Nadeau, Kelly A, Clausen, Andrew M, Hansen, Karl B

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Thiazolylalanine-Derived Catalysts for Enantioselective Intermolecular Aldehyde−Imine Cross-Couplings von Mennen, Steven M, Gipson, John D, Kim, Yoona R, Miller, Scott J

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Development of a Factory Process for Omecamtiv Mecarbil, a Novel Cardiac Myosin Activator von Caille, Seb, Allgeier, Alan M, Bernard, Charles, Correll, Tiffany L, Cosbie, Andrew, Crockett, Richard D, Cui, Sheng, Faul, Margaret M, Hansen, Karl B, Huggins, Seth, Langille, Neil, Mennen, Steven M, Morgan, Bradley P, Morrison, Henry, Muci, Alexander, Nagapudi, Karthik, Quasdorf, Kyle, Ranganathan, Krishnakumar, Roosen, Philipp, Shi, Xianqing, Thiel, Oliver R, Wang, Fang, Tvetan, Justin T, Woo, Jacqueline C. S, Wu, Steven, Walker, Shawn D

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Development of a Bio-Inspired Acyl-Anion Equivalent Macrocyclization and Synthesis of a trans-Resorcylide Precursor von Mennen, Steven M, Miller, Scott J

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A peptide-catalyzed asymmetric Stetter reaction von Mennen, Steven M, Blank, Jarred T, Tran-Dubé, Michelle B, Imbriglio, Jason E, Miller, Scott J

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Synthesis of aziridinomitosenes through base-catalyzed conjugate addition von Tsuboike, Kazunari, Guerin, David J., Mennen, Steven M., Miller, Scott J.

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Synergistic nitroreductase/vanadium catalysis enables chemoselective nitro reductions to anilines in the absence of hydrogen gas von Bisagni, Serena, Bornadel, Amin, Cherney, Alan H., Hedley, Simon J., LePaih, Jacques, Mennen, Steven M., Pushpanath, Ahir, Slabu, Iustina, Tedrow, Jason, Dominguez, Beatriz

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POLYMORPHIC FORMS OF (S)-12-FLUORO-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE von Kelly, Colin, Mennen, Steven M

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POLYMORPHIC FORMS OF (S)-12-FLUORO-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE von KELLY, Colin, MENNEN, Steven M

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ChemInform Abstract: Synthesis of 4-Substituted Phthalazin-1(2H)-ones from 2-Acylbenzoic Acids: Controlling Hydrazine in a Pharmaceutical Intermediate Through PAT-Guided Process De... von Mennen, Steven M., Mak-Jurkauskas, Melody L., Bio, Matthew M., Hollis, L. Steven, Nadeau, Kelly A., Clausen, Andrew M., Hansen, Karl B.

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MACROCYCLIC AZOLOPYRIDINES von Mennen, Steven M, Mayo, Robert Alex

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POLYMORPHIC FORMS OF (S)-12-FLUORO-4-(1-METHYL-1H-PYRAZOL-5-YL)-7A,8,13,14-TETRAHYDRO-7H-[1,2,4]TRIAZOLO[4',3':1,6]PYRIDO[3,2-B]BENZOFURO[4,3-FG][1,4]OXAZONINE von KELLY, Colin, MENNEN, Steven M

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