Enantioselective Synthesis of Janus Kinase Inhibitor INCB018424 via an Organocatalytic Aza-Michael Reaction von Lin, Qiyan, Meloni, David, Pan, Yongchun, Xia, Michael, Rodgers, James, Shepard, Stacey, Li, Mei, Galya, Laurine, Metcalf, Brian, Yue, Tai-Yuen, Liu, Pingli, Zhou, Jiacheng

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Quaternary Chiral Center via Diastereoselective Enolate Amination Enables the Synthesis of an Anti-inflammatory Agent von Magnus, Nicholas A, Campagna, Silvio, Confalone, Pat N, Savage, Scott, Meloni, David J, Waltermire, Robert E, Wethman, Robert G, Yates, Mathew

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Discovery of INCB3284, a Potent, Selective, and Orally Bioavailable hCCR2 Antagonist von Xue, Chu-Biao, Feng, Hao, Cao, Ganfeng, Huang, Taisheng, Glenn, Joseph, Anand, Rajan, Meloni, David, Zhang, Ke, Kong, Lingquan, Wang, Anlai, Zhang, Yingxin, Zheng, Changsheng, Xia, Michael, Chen, Lihua, Tanaka, Hiroyuki, Han, Qi, Robinson, D. J, Modi, Dilip, Storace, Lou, Shao, Lixin, Sharief, Vaqar, Li, Mei, Galya, Laurine G, Covington, Maryanne, Scherle, Peggy, Diamond, Sharon, Emm, Tom, Yeleswaram, Swamy, Contel, Nancy, Vaddi, Kris, Newton, Robert, Hollis, Greg, Friedman, Steven, Metcalf, Brian

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Efficient Synthesis of Losartan, A Nonpeptide Angiotensin II Receptor Antagonist von Larsen, Robert D, King, Anthony O, Chen, Cheng Y, Corley, Edward G, Foster, Bruce S, Roberts, F. Edward, Yang, Chunhua, Lieberman, David R, Reamer, Robert A, Tschaen, David M, Verhoeven, Thomas R, Reider, Paul J, Lo, Young S, Rossano, Lucius T, Brookes, A. Sidney, Meloni, David, Moore, James R, Arnett, John F

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Ethynylphenyl carbonates and carbamates as dual-action acetylcholinesterase inhibitors and anti-inflammatory agents von Saxena, Jaya, Meloni, David, Huang, Mou-Tuan, Heck, Diane E., Laskin, Jeffrey D., Heindel, Ned D., Young, Sherri C.

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Atmospheric lepton fluxes at ultrahigh energies von Illana, José Ignacio, Masip, Manuel, Meloni, Davide

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Discovery of INCB3344, a potent, selective and orally bioavailable antagonist of human and murine CCR2 von Xue, Chu-Biao, Wang, Anlai, Meloni, David, Zhang, Ke, Kong, Ling, Feng, Hao, Glenn, Joseph, Huang, Taisheng, Zhang, Yingxin, Cao, Ganfeng, Anand, Rajan, Zheng, Changsheng, Xia, Michael, Han, Qi, Robinson, D.J., Storace, Lou, Shao, Lixin, Li, Mei, Brodmerkel, Carrie M., Covington, Maryanne, Scherle, Peggy, Diamond, Sharon, Yeleswaram, Swamy, Vaddi, Kris, Newton, Robert, Hollis, Greg, Friedman, Steven, Metcalf, Brian

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Discovery of INCB8761/PF-4136309, a Potent, Selective, and Orally Bioavailable CCR2 Antagonist von Xue, Chu-Biao, Wang, Anlai, Han, Qi, Zhang, Yingxin, Cao, Ganfeng, Feng, Hao, Huang, Taisheng, Zheng, Changsheng, Xia, Michael, Zhang, Ke, Kong, Lingquan, Glenn, Joseph, Anand, Rajan, Meloni, David, Robinson, D. J, Shao, Lixin, Storace, Lou, Li, Mei, Hughes, Robert O, Devraj, Rajesh, Morton, Philip A, Rogier, D. Joseph, Covington, Maryanne, Scherle, Peggy, Diamond, Sharon, Emm, Tom, Yeleswaram, Swamy, Contel, Nancy, Vaddi, Kris, Newton, Robert, Hollis, Greg, Metcalf, Brian

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(Aminoalkoxy)chromones. Selective .sigma. receptor ligands von Erickson, Ronald H, Natalie, Kenneth J, Bock, William, Lu, Zhijian, Farzin, Farzaneh, Sherrill, Ronald G, Meloni, David J, Patch, Raymond J, Rzesotarski, Waclaw J

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Discovery of INCB9471, a Potent, Selective, and Orally Bioavailable CCR5 Antagonist with Potent Anti-HIV-1 Activity von Xue, Chu-Biao, Chen, Lihua, Cao, Ganfeng, Zhang, Ke, Wang, Anlai, Meloni, David, Glenn, Joseph, Anand, Rajan, Xia, Michael, Kong, Ling, Huang, Taisheng, Feng, Hao, Zheng, Changsheng, Li, Mei, Galya, Laurine, Zhou, Jiacheng, Shin, Niu, Baribaud, Fredric, Solomon, Kim, Scherle, Peggy, Zhao, Bitao, Diamond, Sharon, Emm, Tom, Keller, Douglas, Contel, Nancy, Yeleswaram, Swamy, Vaddi, Kris, Hollis, Gregory, Newton, Robert, Friedman, Steven, Metcalf, Brian

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PROCESS AND INTERMEDIATES FOR PREPARING A JAK INHIBITOR von Meloni, David, Chen, Shili, Su, Naijing, Jia, Zhongjiang, Pan, Yongchun, Liu, Pingli, Zhou, Jiacheng, Xia, Michael

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Process and intermediates for preparing a JAK inhibitor von Meloni, David, Chen, Shili, Su, Naijing, Jia, Zhongjiang, Pan, Yongchun, Liu, Pingli, Zhou, Jiacheng, Xia, Michael

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PROCESS AND INTERMEDIATES FOR PREPARING A JAK1 INHIBITOR von Chen, Shili, Su, Naijing, Pan, Yongchun, Liu, Pingli, Meloni, David J, Zhou, Jiacheng, Xia, Michael

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Process and intermediates for preparing a JAK1 inhibitor von Chen, Shili, Su, Naijing, Pan, Yongchun, Liu, Pingli, Meloni, David J, Zhou, Jiacheng, Xia, Michael

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SOLID FORMS OF A JAK INHIBITOR AND PROCESS OF PREPARING THE SAME von MELONI, David, LIU, Weiguo, JIA, Zhongjiang, PAN, Yongchun, LIU, Pingli, ZHOU, Jiacheng, HOUSTON, Travis

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SOLID FORMS OF JAK INHIBITOR AND PROCESS OF PREPARING THE SAME von Meloni, David, Houston, Travis, Liu, Weiguo, Jia, Zhongjiang, Pan, Yongchun, Liu, Pingli, Zhou, Jiacheng

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Salts of a PD-1/PD-L1 inhibitor von Jia, Zhongjiang, Pan, Yongchun, Liu, Pingli, Meloni, David J, Wu, Yongzhong, Li, Qun, Zhou, Jiacheng

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PROCESS AND INTERMEDIATES FOR PREPARING A JAK INHIBITOR von Parks, James M, Chen, Shili, Su, Naijing, Liu, Weiguo, Pan, Yongchun, Liu, Pingli, Meloni, David J, Zhou, Jiacheng, Xia, Michael

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PROCESS AND INTERMEDIATES FOR PREPARING BARICITINIB von SU, Naijing, MELONI, David, CHEN, Shili, XIA, Michael, JIA, Zhongjiang, PAN, Yongchun, ZHOU, Jiacheng, LIU, Pingli

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Process and intermediates for preparing a JAK inhibitor von Parks, James M, Chen, Shili, Su, Naijing, Liu, Weiguo, Pan, Yongchun, Liu, Pingli, Meloni, David J, Zhou, Jiacheng, Xia, Michael

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