Temperature-dependences of the kinetics of reactions of papain and actinidin with a series of reactivity probes differing in key molecular recognition features von Gul, Sheraz, Mellor, Geoffrey W, Thomas, Emrys W, Brocklehurst, Keith

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Rational design of 4-amino-5,6-diaryl-furo[2,3- d]pyrimidines as potent glycogen synthase kinase-3 inhibitors von Miyazaki, Yasushi, Maeda, Yutaka, Sato, Hideyuki, Nakano, Masato, Mellor, Geoffrey W.

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Discovery of 6-Aryl-7-alkoxyisoquinoline Inhibitors of IκB Kinase-β (IKK-β) von Christopher, John A, Bamborough, Paul, Alder, Catherine, Campbell, Amanda, Cutler, Geoffrey J, Down, Kenneth, Hamadi, Ahmed M, Jolly, Adrian M, Kerns, Jeffrey K, Lucas, Fiona S, Mellor, Geoffrey W, Miller, David D, Morse, Mary A, Pancholi, Kiritkant D, Rumsey, William, Solanke, Yemisi E, Williamson, Rick

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The discovery of 2-amino-3,5-diarylbenzamide inhibitors of IKK-α and IKK-β kinases von Christopher, John A., Avitabile, Barbara G., Bamborough, Paul, Champigny, Aurelie C., Cutler, Geoffrey J., Dyos, Susan L., Grace, Ken G., Kerns, Jeffrey K., Kitson, Jeremy D., Mellor, Geoffrey W., Morey, James V., Morse, Mary A., O’Malley, Carolyn F., Patel, Champa B., Probst, Nicholas, Rumsey, William, Smith, Clive A., Wilson, Michael J.

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3,5-Disubstituted-indole-7-carboxamides: The discovery of a novel series of potent, selective inhibitors of IKK-β von Miller, David D., Bamborough, Paul, Christopher, John A., Baldwin, Ian R., Champigny, Aurelie C., Cutler, Geoffrey J., Kerns, Jeffrey K., Longstaff, Timothy, Mellor, Geoffrey W., Morey, James V., Morse, Mary A., Nie, Hong, Rumsey, William L., Taggart, John J.

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5-(1 H-Benzimidazol-1-yl)-3-alkoxy-2-thiophenecarbonitriles as potent, selective, inhibitors of IKK-ε kinase von Bamborough, Paul, Christopher, John A., Cutler, Geoffrey J., Dickson, Marion C., Mellor, Geoffrey W., Morey, James V., Patel, Champa B., Shewchuk, Lisa M.

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Development of a CD28/CD86 (B7-2) Binding Assay for High Throughput Screening by Homogeneous Time-Resolved Fluorescence von Mellor, Geoffrey W., Burden, M. Neil, Preaudat, Marc, Joseph, Yvonne, Cooksley, Susan B., Ellis, Jonathan H., Banks, Martyn N.

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3,5-Disubstituted-indole-7-carboxamides: The discovery of a novel series of potent, selective inhibitors of IIK-β von MILLER, David D, BAMBOROUGH, Paul, MORSE, Mary A, HONG NIE, RUMSEY, William L, TAGGART, John J, CHRISTOPHER, John A, BALDWIN, Ian R, CHAMPIGNY, Aurelie C, CUTLER, Geoffrey J, KERNS, Jeffrey K, LONGSTAFF, Timothy, MELLOR, Geoffrey W, MOREY, James V

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Searching for Chemokine Receptor Binding Antagonists by High Throughput Screening von Mellor, Geoffrey W., Fogarty, Simon J., O’Brien, M. Shane, Congreve, Miles, Banks, Martyn N., Mills, Kirsten M., Jefferies, Barbara, Houston, John G.

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Discovery of 6-Aryl-7-alkoxyisoquinoline Inhibitors of IKB Kinase-β (IKK-β) von CHRISTOPHER, John A, BAMBOROUGH, Paul, MELLOR, Geoffrey W, MILLER, David D, MORSE, Mary A, PANCHOLI, Kiritkant D, RUMSEY, William, SOLANKE, Yemisi E, WILLIAMSON, Rick, ALDER, Catherine, CAMPBELL, Amanda, CUTLER, Geoffrey J, DOWN, Kenneth, HAMADI, Ahmed M, JOLLY, Adrian M, KERNS, Jeffrey K, LUCAS, Fiona S

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Development and Validation of a Fluoroimmunoassay for Urinary Normetanephrine von Gallacher, Gerard, Mellor, Geoffrey W, Landon, John, Sjostrom, Lena

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Discovery of 6-aryl-7-alkoxyisoquinoline inhibitors of IkappaB kinase-beta (IKK-beta) von Christopher, John A, Bamborough, Paul, Alder, Catherine, Campbell, Amanda, Cutler, Geoffrey J, Down, Kenneth, Hamadi, Ahmed M, Jolly, Adrian M, Kerns, Jeffrey K, Lucas, Fiona S, Mellor, Geoffrey W, Miller, David D, Morse, Mary A, Pancholi, Kiritkant D, Rumsey, William, Solanke, Yemisi E, Williamson, Rick

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Characterization of the Electrostatic Perturbation of a Catalytic Site (Cys)-S –/(His)-Im +H Ion-pair in One Type of Serine Proteinase Architecture by Kinetic and Computational Stu... von Plou, Francisco J., Kowlessur, Devanand, Malthouse, Paul G.J., Mellor, Geoffrey W., Hartshorn, Michael J., Pinitglang, Surapong, Patel, Hasu, Topham, Christopher M., Thomas, Emrys W., Verma, Chandra, Brocklehurst, Keith

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Catalytic antibody activity elicited by active immunisation : evidence for natural variation involving preferential stabilization of the transition state von GALLACHER, G, JACKON, C. S, SEARCEY, M, GOEL, R, MELLOR, G. W, SMITH, C. Z, BROCKLEHURST, K

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Comparison of three different activation methods for coupling antibodies to magnetisable cellulose particles von Al-Abdulla, Ibrahim H., Mellor, Geoffrey W., Childerstone, Michael S., Sidki, Ahmad M., Smith, David S.

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5-(1H-Benzimidazol-1-yl)-3-alkoxy-2-thiophenecarbonitriles as Potent, Selective, Inhibitors of IKK-ε Kinase von Bamborough, Paul, Christopher, John A., Cutler, Geoffrey J., Dickson, Marion C., Mellor, Geoffrey W., Morey, James V., Patel, Champa B., Shewchuk, Lisa M.

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Catalytic antibody activity elicited by active immunisation von GALLACHER, Gerard, JACKSON, Caroline S., SEARCEY, Mark, GOEL, Rajiv, MELLOR, Geoffrey W., SMITH, Carmen Z., BROCKLEHURST, Keith

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Derivatives of hydroxymethoxy mandelic acid (HMMA), homovanillic acid (HVA), antibodies and labelled substances prepared therefrom, and immunoassays using these von HO, YEE-PING, GALLACHER, GERARD, MELLOR, GEOFFREY W

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Derivatives of hydroxymethoxy mandelic acid (HMMA), homovanillic acid (HVA), antibodies and labelled substances prepared therefrom, and immunoassays using these von HO, YEE-PING, GALLACHER, GERARD, MELLOR, GEOFFREY W

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The classification of feeding and eating disorders in the ICD-11: results of a field study comparing proposed ICD-11 guidelines with existing ICD-10 guidelines von Claudino, Angélica M, Pike, Kathleen M, Hay, Phillipa, Keeley, Jared W, Evans, Spencer C, Rebello, Tahilia J, Bryant-Waugh, Rachel, Dai, Yunfei, Zhao, Min, Matsumoto, Chihiro, Herscovici, Cecile Rausch, Mellor-Marsá, Blanca, Stona, Anne-Claire, Kogan, Cary S, Andrews, Howard F, Monteleone, Palmiero, Pilon, David Joseph, Thiels, Cornelia, Sharan, Pratap, Al-Adawi, Samir, Reed, Geoffrey M

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