Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design von Meanwell, Nicholas A

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Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design von Meanwell, Nicholas A

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Improving Drug Design: An Update on Recent Applications of Efficiency Metrics, Strategies for Replacing Problematic Elements, and Compounds in Nontraditional Drug Space von Meanwell, Nicholas A

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Bioisosteres of the Phenyl Ring: Recent Strategic Applications in Lead Optimization and Drug Design von Subbaiah, Murugaiah A. M, Meanwell, Nicholas A

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The expanding role of prodrugs in contemporary drug design and development von Rautio, Jarkko, Meanwell, Nicholas A., Di, Li, Hageman, Michael J.

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Metabolic and Pharmaceutical Aspects of Fluorinated Compounds von Johnson, Benjamin M, Shu, Yue-Zhong, Zhuo, Xiaoliang, Meanwell, Nicholas A

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The pyridazine heterocycle in molecular recognition and drug discovery von Meanwell, Nicholas A.

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Applications of Fluorine in Medicinal Chemistry von Gillis, Eric P, Eastman, Kyle J, Hill, Matthew D, Donnelly, David J, Meanwell, Nicholas A

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A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design von Beno, Brett R, Yeung, Kap-Sun, Bartberger, Michael D, Pennington, Lewis D, Meanwell, Nicholas A

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Applications of fluorine-containing amino acids for drug design von Mei, Haibo, Han, Jianlin, Klika, Karel D., Izawa, Kunisuke, Sato, Tatsunori, Meanwell, Nicholas A., Soloshonok, Vadim A.

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Tailor‐Made Amino Acids and Fluorinated Motifs as Prominent Traits in Modern Pharmaceuticals von Mei, Haibo, Han, Jianlin, White, Sarah, Graham, Daniel J., Izawa, Kunisuke, Sato, Tatsunori, Fustero, Santos, Meanwell, Nicholas A., Soloshonok, Vadim A.

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Applications of Bioisosteres in the Design of Biologically Active Compounds von Meanwell, Nicholas A

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Synthesis of Cyclobutane-Fused Tetracyclic Scaffolds via Visible-Light Photocatalysis for Building Molecular Complexity von Oderinde, Martins S, Mao, Edna, Ramirez, Antonio, Pawluczyk, Joseph, Jorge, Christine, Cornelius, Lyndon A. M, Kempson, James, Vetrichelvan, Muthalagu, Pitchai, Manivel, Gupta, Anuradha, Gupta, Arun Kumar, Meanwell, Nicholas A, Mathur, Arvind, Dhar, T. G. Murali

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Photocatalytic Dearomative Intermolecular [2 + 2] Cycloaddition of Heterocycles for Building Molecular Complexity von Oderinde, Martins S, Ramirez, Antonio, Dhar, T G Murali, Cornelius, Lyndon A M, Jorge, Christine, Aulakh, Darpandeep, Sandhu, Bhupinder, Pawluczyk, Joseph, Sarjeant, Amy A, Meanwell, Nicholas A, Mathur, Arvind, Kempson, James

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The crystal structure of NS5A domain 1 from genotype 1a reveals new clues to the mechanism of action for dimeric HCV inhibitors von Lambert, Sebastian M., Langley, David R., Garnett, James A., Angell, Richard, Hedgethorne, Katy, Meanwell, Nicholas A., Matthews, Steve J.

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Preclinical Profile and Characterization of the Hepatitis C Virus NS3 Protease Inhibitor Asunaprevir (BMS-650032) von MCPHEE, Fiona, SHEAFFER, Amy K, CHAOQUN CHEN, LEE, Min S, MOSURE, Kathy, SUN, Li-Qiang, SINZ, Michael, MEANWELL, Nicholas A, COLONNO, Richard J, KNIPE, Jay, SCOLA, Paul, FRIBORG, Jacques, HERNANDEZ, Dennis, FALK, Paul, GUANGZHI ZHAI, LEVINE, Steven, CHANIEWSKI, Susan, FEI YU, BARRY, Diana

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Allosteric Modulators of Drug Targets

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Applications of Isosteres of Piperazine in the Design of Biologically Active Compounds: Part 1 von Meanwell, Nicholas A., Loiseleur, Olivier

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Applications of Isosteres of Piperazine in the Design of Biologically Active Compounds: Part 2 von Meanwell, Nicholas A., Loiseleur, Olivier

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Homology models of the HIV-1 attachment inhibitor BMS-626529 bound to gp120 suggest a unique mechanism of action von Langley, David R., Roy Kimura, S., Sivaprakasam, Prasanna, Zhou, Nannan, Dicker, Ira, McAuliffe, Brian, Wang, Tao, Kadow, John F., Meanwell, Nicholas A., Krystal, Mark

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