Development of a Concise Multikilogram Synthesis of LPA‑1 Antagonist BMS-986020 via a Tandem Borylation–Suzuki Procedure von Smith, Michael J, Lawler, Michael J, Kopp, Nathaniel, Mcleod, Douglas D, Davulcu, Akin H, Lin, Dong, Katipally, Kishta, Sfouggatakis, Chris

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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 3. Mechanistic Studies Enable a Scale-Independent Friedel–Crafts Acylation von Beutner, Gregory L, Albrecht, Jacob, Fan, Junying, Fanfair, Dayne, Lawler, Michael J, Bultman, Michael, Chen, Ke, Ivy, Sabrina, Schild, Richard L, Tripp, Jonathan C, Murugesan, Saravanababu, Dambalas, Konstantinos, McLeod, Douglas D, Sweeney, Jason T, Eastgate, Martin D, Conlon, David A

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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 6. Friedel–Crafts Acylation/Hydrolysis and Amidation von Zheng, Bin, Silverman, Steven M, Steinhardt, Sarah E, Kolotuchin, Sergei, Iyer, Vidya, Fan, Junying, Skliar, Dimitri, McLeod, Douglas D, Bultman, Michael, Tripp, Jonathan C, Murugesan, Saravanababu, La Cruz, Thomas E, Sweeney, Jason T, Eastgate, Martin D, Conlon, David A

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Preparation of the HIV Attachment Inhibitor BMS-663068. Part 9. Active Pharmaceutical Ingredient Process Development and Powder Properties von La Cruz, Thomas E, Saurer, Eric M, Engstrom, Joshua, Bultman, Michael S, Forest, Robert, Akpinar, Fulya, Ferreira, Glenn, Ho, Jeanne W, Huang, Masano, Soltani, Michelle, Murugesan, Saravanababu, Fanfair, Dayne, Ramirez, Antonio, Rosso, Victor W, Erdemir, Deniz, Rosenbaum, Tamar, Haslam, Michelle, Grier, Stephen, Peddicord, Michael, Pathirana, Charles, Marshall, Jonathan, Ding, Wei, Huang, Yande, Ayers, Sloan, Braem, Alan, Schild, Richard L, Ivy, Sabrina E, Payack, Joseph, McLeod, Douglas D, Nikitczuk, Whitney, Doubleday, Wendel, Shah, Sapna, Conlon, David A

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Process Research and Development for a Tetrazole-Based Growth Hormone Secretagogue (GHS) Pharmaceutical Development Candidate von Davulcu, Akin H, McLeod, Douglas D, Li, Jun, Katipally, Kishta, Littke, Adam, Doubleday, Wendel, Xu, Zhongmin, McConlogue, Cary W, Lai, Chiajen J, Gleeson, Margaret, Schwinden, Mark, Parsons, Rodney L

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Stereoselective Process for a CCR3 Antagonist von Yue, Tai-Yuen, McLeod, Douglas D, Albertson, Kevin B, Beck, Steven R, Deerberg, Joerg, Fortunak, Joseph M, Nugent, William A, Radesca, Lilian A, Tang, Liya, Xiang, Cathie Dong

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Kilogram Synthesis of a LFA-1/ICAM Inhibitor von DelMonte, Albert J, Waltermire, Robert E, Fan, Yu, McLeod, Douglas D, Gao, Zhinong, Gesenberg, Kirsten D, Girard, Kevin P, Rosingana, Miguel, Wang, Xuebao, Kuehne-Willmore, Jennifer, Braem, Alan D, Castoro, John A

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Stereoselective Synthesis of the Nonproteinogenic Amino Acid (2S,3R)-3-Amino-2-hydroxydecanoic Acid from (4S,5S)-4-Formyl-5-vinyl-2-oxazolidinone von Wee, Andrew G. H, McLeod, Douglas D

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Stereoselective Synthesis of the Nonproteinogenic Amino Acid (2S,3R)-3-Amino-2-hydroxydecanoic Acid from (4S,5S)-4-Formyl-5-vinyl-2-oxazolidinone von Wee, Andrew G. H, McLeod, Douglas D

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Steric and Electronic Influences on the Diastereoselectivity of the Rh2(OAc)4-Catalyzed C−H Insertion in Chiral Ester Diazoanilides:  Synthesis of Chiral, Nonracemic 4-Substituted... von Wee, Andrew G. H, Liu, Baosheng, McLeod, Douglas D

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Steric and Electronic Influences on the Diastereoselectivity of the Rh 2 (OAc) 4 -Catalyzed C−H Insertion in Chiral Ester Diazoanilides:  Synthesis of Chiral, Nonracemic 4-Substitu... von Wee, Andrew G. H., Liu, Baosheng, McLeod, Douglas D.

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Asymmetric catalytic hydrogenation process for preparation of chiral cyclic -aminoesters von Deerberg, Joerg, McLeod, Douglas D, Yue, Tai-Yuen

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Asymmetric catalytic hydrogenation process for preparation of chiral cyclic beta-aminoesters von MCLEOD DOUGLAS D, YUE TAI-YUEN, DEERBERG JOERG

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Asymmetric catalytic hydrogenation process for preparation of chiral cyclic beta-aminoesters von MCLEOD DOUGLAS D, YUE TAI-YUEN, DEERBERG JOERG

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ChemInform Abstract: Synthesis of (2R,3S)-3-Hydroxy-2-hydroxymethylpyrrolidine from (4S,5S)-3-Benzyl-4-formyl-5-vinyl-2-oxazolidinone von Wee, Andrew G. H., McLeod, Douglas D., Rankin, Trent J.

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CRYSTALLINE FORMS AND PROCESS FOR PREPARING SPIRO-HYDANTOIN COMPOUNDS von WEI CHENKOU, MCLEOD DOUGLAS D, DHAR T.G. MURALI, MALLEY MARY F, FAN YU, DELMONTE ALBERT J, WALTERMIRE ROBERT E, GOUGOUTAS JACK Z

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Crystalline forms and process for preparing spiro-hydantoin compounds von DelMonte, Albert J, Dhar, T. G. Murali, Fan, Yu, Gougoutas, Jack Z, Malley, Mary F, McLeod, Douglas D, Waltermire, Robert E, Wei, Chenkou

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Crystalline forms and process for preparing spiro-hydantoin compounds von WEI CHENKOU, DHAR T. G. MURALI, MCLEOD DOUGLAS D, MALLEY MARY F, FAN YU, DELMONTE ALBERT J, WALTERMIRE ROBERT E, GOUGOUTAS JACK Z

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Pyridyl-substituted spiro-hydantoin crystalline forms and process von CHEN BANGI, MCLEOD DOUGLAS D, ZHANG HUIPING, DHAR T.G. M, GLEESON MARGARET, DELMONTE ALBERT J, GALELLA MICHAEL, GOUGOUTAS JACK Z

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CRYSTALLINE FORMS OF6-[(5S,9R)-9-(4-CYANOPHENYL)-3-(3,5-DICHLOROPHENYL)-1-METHYL-2,4-DIOXO-1,3,7-TRIAZASPIRO[4.4]NON-7-YL]NICOTINIC ACID AS INHIBITORS OF CD18 INTEGRINS, ICAMS AND/... von ZHANG, HUIPING, MCLEOD, DOUGLAS D, GALELLA, MICHAEL, GOUGOUTAS, JACK Z, CHEN, BANG CHI, DELMONTE, ALBERT J, GLEESON, MARGARET, DHAR, T. G. MURALI

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