Development of Targeted Alpha Particle Therapy for Solid Tumors von Tafreshi, Narges K, Doligalski, Michael L, Tichacek, Christopher J, Pandya, Darpan N, Budzevich, Mikalai M, El-Haddad, Ghassan, Khushalani, Nikhil I, Moros, Eduardo G, McLaughlin, Mark L, Wadas, Thaddeus J, Morse, David L

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Discovery of a novel proteasome inhibitor selective for cancer cells over non-transformed cells von Kazi, Aslamuzzaman, Lawrence, Harshani, Guida, Wayne C., McLaughlin, Mark L., Springett, Gregory M., Berndt, Norbert, Yip, Richard M., Sebti, Said M.

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Intramolecular Quenching of Tryptophan Fluorescence by the Peptide Bond in Cyclic Hexapeptides von Adams, Paul D, Chen, Yu, Ma, Kan, Zagorski, Michael G, Sönnichsen, Frank D, McLaughlin, Mark L, Barkley, Mary D

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Melanocortin 1 Receptor-Targeted α-Particle Therapy for Metastatic Uveal Melanoma von Tafreshi, Narges K, Tichacek, Christopher J, Pandya, Darpan N, Doligalski, Michael L, Budzevich, Mikalai M, Kil, HyunJoo, Bhatt, Nikunj B, Kock, Nancy D, Messina, Jane L, Ruiz, Epifanio E, Delva, Nella C, Weaver, Adam, Gibbons, William R, Boulware, David C, Khushalani, Nikhil I, El-Haddad, Ghassan, Triozzi, Pierre L, Moros, Eduardo G, McLaughlin, Mark L, Wadas, Thaddeus J, Morse, David L

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Biodistribution and Multicompartment Pharmacokinetic Analysis of a Targeted α Particle Therapy von Tichacek, Christopher J, Tafreshi, Narges K, Kil, HyunJoo, Engelman, Robert W, Doligalski, Michael L, Budzevich, Mikalai M, Gage, Kenneth L, McLaughlin, Mark L, Wadas, Thaddeus J, Silva, Ariosto, Moros, Eduardo, Morse, David L

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Intraoperative Guidance of Pancreatic Cancer Resection Using a Toll-like Receptor 2-Targeted Fluorescence Molecular Imaging Agent von Huynh, Amanda S, Cohen, Allison S, Doligalski, Michael, Casagni, Todd J, Moberg, Valerie E, Huang, Xuan, Morse, Jennifer, Abrahams, Dominique, Lloyd, Mark C, Centeno, Barbara A, Baldwin, Margaret K, McLaughlin, Mark L, Vagner, Josef, Morse, David L

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Structure and properties of DOTA-chelated radiopharmaceuticals within the Ac decay pathway von Khabibullin, Artem R, Karolak, Aleksandra, Budzevich, Mikalai M, McLaughlin, Mark L, Morse, David L, Woods, Lilia M

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Abstract 517: An MC1R targeted 225Ac radiopharmaceutical agent for treatment of uveal melanoma von Tafreshi, Narges K., Doligalski, Michael L., Pandya, Darpan N., Joo Kil, Hyun, Budzevich, Mikalai, Wadas, Thaddeus J., McLaughlin, Mark L., Morse, David

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Lipophilicity Determines Routes of Uptake and Clearance, and Toxicity of an Alpha-Particle-Emitting Peptide Receptor Radiotherapy von Tafreshi, Narges K, Kil, HyunJoo, Pandya, Darpan N, Tichacek, Christopher J, Doligalski, Michael L, Budzevich, Mikalai M, Delva, Nella C, Langsen, Michael L, Vallas, John A, Boulware, David C, Engelman, Robert W, Gage, Kenneth L, Moros, Eduardo G, Wadas, Thaddeus J, McLaughlin, Mark L, Morse, David L

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MTI-101 (cyclized HYD1) binds a CD44 containing complex and induces necrotic cell death in multiple myeloma von Gebhard, Anthony W, Jain, Priyesh, Nair, Rajesh R, Emmons, Michael F, Argilagos, Raul F, Koomen, John M, McLaughlin, Mark L, Hazlehurst, Lori A

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Acquisition of resistance toward HYD1 correlates with a reduction in cleaved α4 integrin expression and a compromised CAM-DR phenotype von Emmons, Michael F, Gebhard, Anthony W, Nair, Rajesh R, Baz, Rachid, McLaughlin, Mark L, Cress, Anne E, Hazlehurst, Lori A

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Structure and properties of DOTA-chelated radiopharmaceuticals within the 225Ac decay pathway von Khabibullin, Artem R, Karolak, Aleksandra, Budzevich, Mikalai M, McLaughlin, Mark L, Morse, David L, Woods, Lilia M

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Facile Iterative Synthesis of 2,5-Terpyrimidinylenes as Nonpeptidic α-Helical Mimics von Anderson, Laura, Zhou, Mingzhou, Sharma, Vasudha, McLaughlin, Jillian M, Santiago, Daniel N, Fronczek, Frank R, Guida, Wayne C, McLaughlin, Mark L

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Structure and properties of DOTA-chelated radiopharmaceuticals within the 225 Ac decay pathway von Khabibullin, Artem R, Karolak, Aleksandra, Budzevich, Mikalai M, McLaughlin, Mark L, Morse, David L, Woods, Lilia M

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Bioactivity improvement via display of the hydrophobic core of HYD1 in a cyclic β‐hairpin‐like scaffold, MTI‐101 von Jain, Priyesh, Badger, David B., Liang, Yi, Gebhard, Anthony W., Santiago, Daniel, Murray, Philip, Kaulagari, Sridhar R., Gauthier, Ted J., Nair, Rajesh, Kumar, MohanRaja, Guida, Wayne C., Hazlehurst, Lori A., McLaughlin, Mark L.

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Molecular docking/dynamics studies of Aurora A kinase inhibitors von Talele, Tanaji T., McLaughlin, Mark L.

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De Novo Antimicrobial Peptides with Low Mammalian Cell Toxicity von Javadpour, Maryam M, Juban, Martha M, Lo, Wai-Chun J, Bishop, Steven M, Alberty, J. Brannon, Cowell, Scott M, Becker, Calvin L, McLaughlin, Mark L

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Identification of a disruptor of the MDM2-p53 protein–protein interaction facilitated by high-throughput in silico docking von Lawrence, Harshani R., Li, Zhenyu, Richard Yip, M.L., Sung, Shen-Shu, Lawrence, Nicholas J., McLaughlin, Mark L., McManus, Gregory J., Zaworotko, Michael J., Sebti, Saïd M., Chen, Jiandong, Guida, Wayne C.

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Photophysical Studies of the Trans to Cis Isomerization of the Push−Pull Molecule: 1-(Pyridin-4-yl)-2-(N-methylpyrrol-2-yl)ethene (mepepy) von Mokdad, Audrey, Belof, Jonathan L, Yi, Sung Wook, Shuler, Stephen E, McLaughlin, Mark L, Space, Brian, Larsen, Randy W

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Synthesis of Extended Linear Aromatics Using Tandem Diels-Alder Aromatization Reactions von Morris, J. Larry, Becker, Calvin L, Fronczek, Frank R, Daly, William H, McLaughlin, Mark L

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