Samarium(II) iodide-induced reductive cyclization of unactivated olefinic ketones. Sequential radical cyclization/intermolecular nucleophilic addition and substitution reactions von Molander, Gary A, McKie, Jeffrey A

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Stereochemical Investigations of Samarium(II) Iodide-Promoted 5-Exo and 6-Exo Ketyl-Olefin Radical Cyclization Reactions von Molander, Gary A, McKie, Jeffrey A

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Synthesis of Substituted Cyclooctanols by a Samarium(II) Iodide Promoted 8-Endo Radical Cyclization Process von Molander, Gary A, McKie, Jeffrey A

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Intramolecular nucleophilic acyl substitution reactions of halo-substituted esters and lactones. New applications of organosamarium reagents von Molander, Gary A, McKie, Jeffrey A

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Lead identification of a potent benzopyranone selective estrogen receptor modulator von McKie, Jeffrey A., Bhagwat, Shripad S., Brady, Helen, Doubleday, Mary, Gayo, Leah, Hickman, Mathew, Jalluri, Ravi K., Khammungkhune, Sak, Kois, Adam, Mortensen, Deborah, Richard, Normand, Sapienza, John, Shevlin, Graziella, Stein, Bernd, Sutherland, May

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Effects of SP500263, a novel, potent antiestrogen, on breast cancer cells and in xenograft models von BRADY, Helen, DESAI, Sonal, STEIN, Bernd, GAYO-FUNG, Leah M, KHAMMUNGKHUNE, Sak, MCKIE, Jeffrey A, O'LEARY, Eoin, PASCASIO, Laura, SUTHERLAND, May Kung, ANDERSON, David W, BHAGWAT, Shripad S

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Total Synthesis of (+)-Duocarmycin A, epi-(+)-Duocarmycin A and Their Unnatural Enantiomers:  Assessment of Chemical and Biological Properties von Boger, Dale L, McKie, Jeffrey A, Nishi, Takahide, Ogiku, Tsuyoshi

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A facile synthesis of bicyclo[m.n.1]alkan-1-ols. Evidence for organosamarium intermediates in the samarium(II) iodide promoted intramolecular Barbier-type reaction von Molander, Gary A, McKie, Jeffrey A

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Enantioselective Total Synthesis of (+)-Duocarmycin A, epi-(+)-Duocarmycin A, and Their Unnatural Enantiomers von Boger, Dale L, McKie, Jeffrey A, Nishi, Takahide, Ogiku, Tsuyoshi

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An Efficient Synthesis of 1,2,9,9a-Tetrahydrocyclopropa[c]benz[e]indol-4-one CBI: An Enhanced and Simplified Analog of the CC-1065 and Duocarmycin Alkylation Subunits von Boger, Dale L, McKie, Jeffrey A

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Synthesis and Properties of Substituted CBI Analogs of CC-1065 and the Duocarmycins Incorporating the 7-Methoxy-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one (MCBI) Alkylation... von Boger, Dale L, McKie, Jeffrey A, Cai, Hui, Cacciari, Barbara, Baraldi, P. G

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A comparative study of the solvolysis reactivity, regioselectivity, and stereochemistry of the duocarmycin a and sa alkylation subunits von Boger, Dale L., Goldberg, Joel, McKie, Jeffrey A.

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Samarium(II) iodide induced sequential intramolecular nucleophilic acyl substitution and stereospecific intramolecular Meerwein-Ponndorf-Verley reduction/Oppenauer oxidation von Molander, Gary A, McKie, Jeffrey A

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A Hammett correlation for CC-1065 and duocarmycin analogs: Magnitude of substituent electronic effects on functional reactivity von Boger, Dale L., McKie, Jeffrey A., Han, Nianhe, Tarby, Christine M., Riggs, Haiqiong W., Kitos, Paul A.

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Remarkable enantioselective 1,4-addition reactions of chiral allylphosphonyl anions (ambident nucleophiles) with cyclic enones (ambident electrophiles) von Hua, Duy H, King, Roch Chan Yu, McKie, Jeffrey A, Myer, Les

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Asymmetric Synthesis of the CBI Alkylation Subunit of the CC-1065 and Duocarmycin Analogs von Boger, Dale L., McKie, Jeffrey A., Boyce, Christopher W.

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4-((4-(2-pyrrolidinylethoxy)phenyl)methyl)-3-(4-(trifluoromethyl)phenyl)-7-hydroxychromen-2one, pharmaceutically acceptable salts thereof and methods of use therewith von BHAGWAT SHRIPAD S, MCKIE JEFFREY A

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BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH von MARTIN MISSBACH, JOHANNE RENAUD, JEFFREY A. MCKIE, SHRIPAD S. BHAGWAT

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Lead Identification (IIa) of a Potent Benzopyranone Selective Estrogen Receptor Modulator von McKie, Jeffrey A., ., et al

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Benzopyranone compounds, compositions thereof, and methods of treatment therewith von MARTIN MISSBACH, JOHANNE RENAUD, JEFFREY A. MCKIE, SHRIPAD S. BHAGWAT

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