Synthesis of Macrocyclic, Potential Protease Inhibitors Using a Generic Scaffold von Dumez, Estelle, Snaith, John S, Jackson, Richard F. W, McElroy, Andrew B, Overington, John, Wythes, Martin J, Withka, Jane M, McLellan, Thomas J

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Discovery of Potent & Selective Inhibitors of Activated Thrombin-Activatable Fibrinolysis Inhibitor for the Treatment of Thrombosis von Bunnage, Mark E, Blagg, Julian, Steele, John, Owen, Dafydd R, Allerton, Charlotte, McElroy, Andrew B, Miller, Duncan, Ringer, Tracy, Butcher, Ken, Beaumont, Kevin, Evans, Karen, Gray, Andrew J, Holland, Stephen J, Feeder, Neil, Moore, Robert S, Brown, David G

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Regulation of tumour necrosis factor-α processing by a metalloproteinase inhibitor von McGeehan, Gerard M, Becherer, J. David, Bast, Robert C, Boyer, Cinda M, Champion, Brian, Connolly, Kevin M, Conway, James G, Furdon, Paul, Karp, Stephen, Kidao, Sudha, McElroy, Andrew B, Nichols, James, Pryzwansky, Katherine M, Schoenen, Frank, Sekut, Les, Truesdale, Anne, Verghese, Margrith, Warner, Janet, Ways, Judy P

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Structure of the Catalytic Domain of Fibroblast Collagenase Complexed with an Inhibitor von Lovejoy, Brett, Cleasby, Anne, Hassell, Anne M., Longley, Kelly, Luthe, Michael A., Weigl, Debra, McGeehan, Gerard, McElroy, Andrew B., Drewry, David, Lambert, Millard H., Jordan, Steven R.

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Conformationally constrained tachykinin analogs: potent and highly selective neurokinin NK-2 receptor agonists von Deal, Martyn J, Hagan, Russell M, Ireland, Simon J, Jordan, Christopher C, McElroy, Andrew B, Porter, Barry, Ross, Barry C, Stephens-Smith, Michaela, Ward, Peter

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Design of Selective Thrombin Inhibitors Based on the (R)-Phe-Pro-Arg Sequence von Danilewicz, John C, Abel, Stuart M, Brown, Alan D, Fish, Paul V, Hawkeswood, Edward, Holland, Stephen J, James, Keith, McElroy, Andrew B, Overington, John, Powling, Michael J, Rance, David J

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New .kappa.-receptor agonists based upon a 2-[(alkylamino)methyl]piperidine nucleus von Scopes, David I. C, Hayes, Norman F, Bays, David E, Belton, David, Brain, John, Brown, Dearg S, Judd, Duncan B, McElroy, Andrew B, Meerholz, Clive A

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Matrix Metalloproteinase Inhibitors Containing a [(Carboxyalkyl)amino]zinc Ligand: Modification of the P1 and P2' Residues von Brown, Frank K, Brown, Peter J, Bickett, D. Mark, Chambers, C. Lynn, Davies, H. Geoff, Deaton, David N, Drewry, David, Foley, Michael, McElroy, Andrew B

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Highly potent and selective heptapeptide antagonists of the neurokinin NK-2 receptor von McElroy, Andrew B, Clegg, Stephen P, Deal, Martyn J, Ewan, George B, Hagan, Russell M, Ireland, Simon J, Jordan, Christopher C, Porter, Barry, Ross, Barry C

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Patent Update: Neurokinin Receptor Antagonists von McElroy, Andrew B

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New Spiropiperidines as Potent and Selective Non-Peptide Tachykinin NK2 Receptor Antagonists von Smith, Paul W, Cooper, Anthony W. J, Bell, Richard, Beresford, Isabel J. M, Gore, Paul M, McElroy, Andrew B, Pritchard, John M, Saez, Victoria, Taylor, Neil R

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Control over absolute (R,S), relative (syn,anti) and geometrical (E,Z) stereochemistry in the synthesis of allylically substituted alkenes from diphenylphosphinoyl epoxy alcohols von Clayden, Jonathan, McElroy, Andrew B., Warren, Stuart

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Matrix metalloproteinase inhibitors containing a [(carboxyalkyl)amino] zinc ligand: Modification of the P1 and P2' residues. [Erratum to document cited in CA120:238898] von Brown, Frank K, Brown, Peter J, Bickett, D. Mark, Chambers, C. Lynn, Davies, H. Geoff, Deaton, David N, Drewry, David, Foley, Michael, McElroy, Andrew B

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Synthesis, antinociceptive activity and opioid receptor profiles of substituted trans-3-(decahydro- and octahydro-4a-isoquinolinyl)phenols von Judd, Duncan B, Brown, Dearg S, Lloyd, Jane E, McElroy, Andrew B, Scopes, David I. C, Birch, Phillip J, Hayes, Ann G, Sheehan, Michael J

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Diastereoselective epoxidation of allylic phosphine oxides von Clayden, Jonathan, Collington, Eric W., Egert, Ernst, McElroy, Andrew B., Warren, Stuart

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The synthesis of (Z)-penta-2,4-dien-1-ol and substituted (E)-pentadienols by the stereochemically controlled Horner–Wittig reaction von Brown, Paul S., Greeves, Nicholas, McElroy, Andrew B., Warren, Stuart

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Stereochemical control (E/Z and syn/anti) by the diphenylphosphinoyl group in the synthesis of allylic alcohols by allylic rearrangement and by 1,4-diastereoselective reduction of... von CLAYDEN, J, COLLINGTON, E. W, ELLIOTT, J, MARTIN, S. J, MCELROY, A. B, WARREN, S, WATERSON, D

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A regiospecific route to conjugated enones via α-phenylthio ketones von DURMAN, J, ELLIOTT, J, MCELROY, A. B, WARREN, S

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Matrix metalloproteinase inhibitors containing a (carboxyalkyl)amino zinc ligand : modification of the P1 and P2' residues von BROWN, F. K, BROWN, P. J, MCGEEHAN, G. M, MYERS, P. L, NORTON, D, SALOVICH, J. M, SCHOENEN, F. J, WARD, P, BICKETT, D. M, CHAMBERS, C. L, DAVIES, H. G, DEATON, D. N, DREWRY, D, FOLEY, M, MCELROY, A. B, GREGSON, M

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Synthesis, antinociceptive activity, and opioid receptor profiles of 10-substituted-6-oxamorphinans von MCELROY, A. B, BAYS, D. E, SCOPES, D. I. C, HAYES, A. G, SHEEHAN, M. J

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