Discovery of a Potent and Selective Covalent p300/CBP Inhibitor von Mastracchio, Anthony, Lai, Chunqiu, Digiammarino, Enrico, Ready, Damien B, Lasko, Loren M, Bromberg, Kenneth D, McClellan, William J, Montgomery, Debra, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Patterson, Melanie J, Sun, Chaohong C, Rosenberg, Saul, Lai, Albert, Michaelides, Michael R

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Discovery of potent and selective thienopyrimidine inhibitors of Aurora kinases von McClellan, William J., Dai, Yujia, Abad-Zapatero, Cele, Albert, Daniel H., Bouska, Jennifer J., Glaser, Keith B., Magoc, Terry J., Marcotte, Patrick A., Osterling, Donald J., Stewart, Kent D., Davidsen, Steven K., Michaelides, Michael R.

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Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors von Wang, Le, Pratt, John K, Soltwedel, Todd, Sheppard, George S, Fidanze, Steven D, Liu, Dachun, Hasvold, Lisa A, Mantei, Robert A, Holms, James H, McClellan, William J, Wendt, Michael D, Wada, Carol, Frey, Robin, Hansen, T. Matthew, Hubbard, Robert, Park, Chang H, Li, Leiming, Magoc, Terrance J, Albert, Daniel H, Lin, Xiaoyu, Warder, Scott E, Kovar, Peter, Huang, Xiaoli, Wilcox, Denise, Wang, Rongqi, Rajaraman, Ganesh, Petros, Andrew M, Hutchins, Charles W, Panchal, Sanjay C, Sun, Chaohong, Elmore, Steven W, Shen, Yu, Kati, Warren M, McDaniel, Keith F

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Reduction of nanoparticle exposure to welding aerosols by modification of the ventilation system in a workplace von Lee, Myong-Hwa, McClellan, William J., Candela, Joe, Andrews, Dan, Biswas, Pratim

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Discovery and Structure−Activity Relationship of Antagonists of B-Cell Lymphoma 2 Family Proteins with Chemopotentiation Activity in Vitro and in Vivo von Wendt, Michael D, Shen, Wang, Kunzer, Aaron, McClellan, William J, Bruncko, Milan, Oost, Thorsten K, Ding, Hong, Joseph, Mary K, Zhang, Haichao, Nimmer, Paul M, Ng, Shi-Chung, Shoemaker, Alexander R, Petros, Andrew M, Oleksijew, Anatol, Marsh, Kennan, Bauch, Joy, Oltersdorf, Tilman, Belli, Barbara A, Martineau, Darlene, Fesik, Stephen W, Rosenberg, Saul H, Elmore, Steven W

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Studies Leading to Potent, Dual Inhibitors of Bcl-2 and Bcl-xL von Bruncko, Milan, Oost, Thorsten K, Belli, Barbara A, Ding, Hong, Joseph, Mary K, Kunzer, Aaron, Martineau, Darlene, McClellan, William J, Mitten, Michael, Ng, Shi-Chung, Nimmer, Paul M, Oltersdorf, Tilman, Park, Cheol-Min, Petros, Andrew M, Shoemaker, Alexander R, Song, Xiaohong, Wang, Xilu, Wendt, Michael D, Zhang, Haichao, Fesik, Stephen W, Rosenberg, Saul H, Elmore, Steven W

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Naphthamidine urokinase plasminogen activator inhibitors with improved pharmacokinetic properties von Bruncko, Milan, McClellan, William J., Wendt, Michael D., Sauer, Daryl R., Geyer, Andrew, Dalton, Christopher R., Kaminski, Michele A., Weitzberg, Moshe, Gong, Jane, Dellaria, Joseph F., Mantei, Robert, Zhao, Xumiao, Nienaber, Vicki L., Stewart, Kent, Klinghofer, Vered, Bouska, Jennifer, Rockway, Todd W., Giranda, Vincent L.

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Interaction with the S1β-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors von Wendt, Michael D., Geyer, Andrew, McClellan, William J., Rockway, Todd W., Weitzberg, Moshe, Zhao, Xumiao, Mantei, Robert, Stewart, Kent, Nienaber, Vicki, Klinghofer, Vered, Giranda, Vincent L.

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Interaction with the S1β-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors von WENDT, Michael D, GEYER, Andrew, GIRANDA, Vincent L, MCCLELLAN, William J, ROCKWAY, Todd W, WEITZBERG, Moshe, XUMIAO ZHAO, MANTEI, Robert, STEWART, Kent, NIENABER, Vicki, KLINGHOFER, Vered

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Reduction of nanoparticle exposure to welding aerosols by modification of the ventilation system in a workplace von Lee, Myong-Hwa, McClellan, William J., Candela, Joe, Andrews, Dan, Biswas, Pratim

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BROMODOMAIN INHIBITORS von Fidanze, Steven D, Kati, Warren M, Sheppard, George S, Wada, Carol K, Wang, Le, McDaniel, Keith F, Holms, James H, Mantei, Robert A, Pratt, John K, McClellan, William J, Liu, Dachun, Dai, Yujia, Hasvold, Lisa

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Conformationally defined adrenergic agents. 1. Design and synthesis of novel .alpha.2-selective adrenergic agents: electrostatic repulsion based conformational prototypes von DeBernardis, John F, Kerkman, Daniel J, Winn, Martin, Bush, Eugene N, Arendsen, David L, McClellan, William J, Kyncl, John J, Basha, Fatima Z

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BROMODOMAIN INHIBITORS von WADA, CAROL K, MCDANIEL, KEITH F, HASVOLD, LISA, LIU, DACHUN, MANTEI, ROBERT A, SHEPPARD, GEORGE S, HOLMS, JAMES H, MCCLELLAN, WILLIAM J, WANG, LE, PRATT, JOHN K, KATI, WARREN M, DAI, YUJIA, FIDANZE, STEVEN D

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BROMODOMAIN INHIBITORS von Fidanze, Steven D, Kati, Warren M, Sheppard, George S, Wada, Carol K, Wang, Le, McDaniel, Keith F, Holms, James H, Mantei, Robert A, Pratt, John K, McClellan, William J, Liu, Dachun, Dai, Yujia, Hasvold, Lisa

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A simple, high-yielding method for the methylenation of catechols von Zelle, Robert E., McClellan, William J.

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COMPOUNDS USEFUL FOR INHIBITING CHK1 von DE JONGE, Marc, Rene, MCCLELLAN, William, J

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PROCESS FOR THE PREPARATION OF A SULFONAMIDE DERIVATIVE von HEXAMER, Laura, TAO, Zhi-fu, WANG, Le, SOUERS, Andrew, J, WENDT, Michael, D, DING, Hong, PETROS, Andrew, M, DOHERTY, George, A, MANTEI, Robert, A, WANG, Gary, T, ELMORE, Steven, W, PARK, Cheol-min, BRUNCKO, Milan, MCCLELLAN, William, J, PARK, Chang, H, WANG, Xilu, KUNZER, Aaron, R, HASVOLD, Lisa, SONG, Xiaohong, SULLIVAN, Gerard, M

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APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES von TAO, ZHI-FU, DOHERTY, GEORGE A, SULLIVAN, GERARD M, LESSENE, GUILLAUME LAURENT, PARK, CHANG H, WANG, XILU, SONG, XIAOHONG, ELMORE, STEVEN W, HASVOLD, LISA, MANTEI, ROBERT A, PETROS, ANDREW M, DING, HONG, MCCLELLAN, WILLIAM J, PARK, CHEOL-MIN, WANG, LE, KUNZER, AARON R, WENDT, MICHAEL D, BRUNCKO, MILAN, DAI, YUJIA, HEXAMER, LAURA, CZABOTAR, PETER EDWARD, SOUERS, ANDREW J, COLMAN, PETER MALCOM, WANG, GARY T

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Bromodomain inhibitors von DAI, Yujia, WANG, Le, SHEPPARD, George S, MANTEI, Robert A, McDANIEL, Keith F, PRATT, John K, HOLMS, James H, LIU, Dachun, HASVOLD, Liza, McCLELLAN, William J, FIDANZE, Steven D, KATI, Warren M, WADA, Carol K

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Bromodomain inhibitors von McClellan, William J, Frey, Robin R, Wada, Carol K, Wang, Le, Hansen, Todd M, McDaniel, Keith F, Liu, Dachun, Pratt, John K

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