Characterization of vabicaserin (SCA-136), a selective 5-hydroxytryptamine 2C receptor agonist von Dunlop, John, Watts, Stephanie W, Barrett, James E, Coupet, Joseph, Harrison, Boyd, Mazandarani, Hossein, Nawoschik, Stanley, Pangalos, Menelas N, Ramamoorthy, Siva, Schechter, Lee, Smith, Deborah, Stack, Gary, Zhang, Jean, Zhang, Guoming, Rosenzweig-Lipson, Sharon

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Antiobesity-like effects of the 5-HT2C receptor agonist WAY-161503 von Rosenzweig-Lipson, Sharon, Zhang, Jean, Mazandarani, Hossein, Harrison, Boyd L, Sabb, Annmarie, Sabalski, Joan, Stack, Gary, Welmaker, Greg, Barrett, James E, Dunlop, John

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Structure–activity study of novel tricyclic benzazepine arginine vasopressin antagonists von Sum, Fuk-Wah, Dusza, John, Santos, Efren Delos, Grosu, George, Reich, Marvin, Du, Xumei, Albright, J.Donald, Chan, Peter, Coupet, Joseph, Ru, Xun, Mazandarani, Hossein, Saunders, Trina

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Discovery of 5-Arylsulfonamido-3- (pyrrolidin-2-ylmethyl)-1H-indole Derivatives as Potent, Selective 5-HT6 Receptor Agonists and Antagonists von Cole, Derek C, Lennox, William J, Lombardi, Sabrina, Ellingboe, John W, Bernotas, Ronald C, Tawa, Gregory J, Mazandarani, Hossein, Smith, Deborah L, Zhang, Guoming, Coupet, Joseph, Schechter, Lee E

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5-Fluoro-2-methyl- N -[4-(5 H -pyrrolo[2,1- c ]- [1,4]benzodiazepin-10(11 H )-ylcarbonyl)-3- chlorophenyl]benzamide (VPA-985):  An Orally Active Arginine Vasopressin Antagonist wit... von Albright, J. Donald, Reich, Marvin F., Delos Santos, Efren G., Dusza, John P., Sum, Fuk-Wah, Venkatesan, Aranapakam M., Coupet, Joseph, Chan, Peter S., Ru, Xun, Mazandarani, Hossein, Bailey, Trina

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N1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives are potent and selective 5-HT6 receptor antagonists von COLE, Derek C, ELLINGBOE, John W, LENNOX, William J, MAZANDARANI, Hossein, SMITH, Deborah L, STOCK, Joseph R, GUOMING ZHANG, PING ZHOU, SCHECHTER, Lee E

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Conformationally constrained N1-arylsulfonyltryptamine derivatives as 5-HT6 receptor antagonists von COLE, Derek C, LENNOX, William J, STOCK, Joseph R, ELLINGBOE, John W, MAZANDARANI, Hossein, SMITH, Deborah L, GUOMING ZHANG, TAWA, Gregory J, SCHECHTER, Lee E

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5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]- [1,4]benzodiazepin-10(11H)-ylcarbonyl)-3- chlorophenyl]benzamide (VPA-985):  An Orally Active Arginine Vasopressin Antagonist with Select... von Albright, J. Donald, Reich, Marvin F, Delos Santos, Efren G, Dusza, John P, Sum, Fuk-Wah, Venkatesan, Aranapakam M, Coupet, Joseph, Chan, Peter S, Ru, Xun, Mazandarani, Hossein, Bailey, Trina

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New Generation Dopaminergic Agents. Part 8: Heterocyclic Bioisosteres that Exploit the 7-OH-2-(aminomethyl)chroman D2 Template von Mewshaw, Richard E., Zhao, Rulin, Shi, Xiaojie, Marquis, Karen, Brennan, Julie A., Mazandarani, Hossein, Coupet, Joseph, Andree, Terrance H.

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Antiobesity-like effects of the 5-HT 2C receptor agonist WAY-161503 von Rosenzweig-Lipson, Sharon, Zhang, Jean, Mazandarani, Hossein, Harrison, Boyd L., Sabb, Annmarie, Sabalski, Joan, Stack, Gary, Welmaker, Greg, Barrett, James E., Dunlop, John

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Antiobesity-like effects of the 5-HT2C receptor agonist WAY-161503 von ROSENZWEIG-LIPSON, Sharon, ZHANG, Jean, MAZANDARANI, Hossein, HARRISON, Boyd L, SABB, Annmarie, SABALSKI, Joan, STACK, Gary, WELMAKER, Greg, BARRETT, James E, DUNLOP, John

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N1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives are potent and selective 5-HT6 receptor antagonists von Cole, Derek C, Ellingboe, John W, Lennox, William J, Mazandarani, Hossein, Smith, Deborah L, Stock, Joseph R, Zhang, Guoming, Zhou, Ping, Schechter, Lee E

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N 1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1 H-indole derivatives are potent and selective 5-HT 6 receptor antagonists von Cole, Derek C., Ellingboe, John W., Lennox, William J., Mazandarani, Hossein, Smith, Deborah L., Stock, Joseph R., Zhang, Guoming, Zhou, Ping, Schechter, Lee E.

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Conformationally constrained N 1-arylsulfonyltryptamine derivatives as 5-HT 6 receptor antagonists von Cole, Derek C., Lennox, William J., Stock, Joseph R., Ellingboe, John W., Mazandarani, Hossein, Smith, Deborah L., Zhang, Guoming, Tawa, Gregory J., Schechter, Lee E.

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Discovery of 5-Arylsulfonamido-3- (pyrrolidin-2-ylmethyl)-1 H -indole Derivatives as Potent, Selective 5-HT 6 Receptor Agonists and Antagonists von Cole, Derek C., Lennox, William J., Lombardi, Sabrina, Ellingboe, John W., Bernotas, Ronald C., Tawa, Gregory J., Mazandarani, Hossein, Smith, Deborah L., Zhang, Guoming, Coupet, Joseph, Schechter, Lee E.

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Synthesis and 5-hydroxytryptamine (5-HT) activity of 2,3,4,4a-tetrahydro-1H-pyrazino[1,2-a]quinoxalin-5-(6H)ones and 2,3,4,4a, 5,6-hexahydro-1H-pyrazino[1,2-a]quinoxalines von WELMAKER, G. S, NELSON, J. A, ROSENZWEIG-LIPSON, S, SUKOFF, S, YINGXIN ZHANG, SABALSKI, J. E, SABB, A. L, POTOSKI, J. R, GRAZIANO, D, KAGAN, M, COUPET, J, DUNLOP, J, MAZANDARANI, H

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New Generation Dopaminergic Agents. Part 8: Heterocyclic Bioisosteres that Exploit the 7-OH-2-(aminomethyl)chroman D 2 Template von Mewshaw, Richard E., Zhao, Rulin, Shi, Xiaojie, Marquis, Karen, Brennan, Julie A., Mazandarani, Hossein, Coupet, Joseph, Andree, Terrance H.

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New Generation Dopaminergic Agents. 1. Discovery of a Novel Scaffold Which Embraces the D2 Agonist Pharmacophore. Structure−Activity Relationships of a Series of 2-(Aminomethyl)chr... von Mewshaw, Richard E, Kavanagh, Joseph, Stack, Gary, Marquis, Karen L, Shi, Xiaojie, Kagan, Michael Z, Webb, Michael B, Katz, Alan H, Park, Anna, Kang, Young H, Abou-Gharbia, Magid, Scerni, Rosemary, Wasik, Theodore, Cortes-Burgos, Luz, Spangler, Taylor, Brennan, Julie A, Piesla, Michael, Mazandarani, Hossein, Cockett, Mark I, Ochalski, Rafal, Coupet, Joseph, Andree, Terrance H

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New generation dopaminergic agents. Part 8: heterocyclic bioisosteres that exploit the 7-OH-2-(aminomethyl)chroman D(2) template von Mewshaw, Richard E, Zhao, Rulin, Shi, Xiaojie, Marquis, Karen, Brennan, Julie A, Mazandarani, Hossein, Coupet, Joseph, Andree, Terrance H

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New generation dopaminergic agents. Part8 : Heterocyclic bioisosteres that exploit the 7-OH-2-(aminomethyl)chroman D2 template von MEWSHAW, Richard E, RULIN ZHAO, XIAOJIE SHI, MARQUIS, Karen, BRENNAN, Julie A, MAZANDARANI, Hossein, COUPET, Joseph, ANDREE, Terrance H

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