An androgen receptor N-terminal domain antagonist for treating prostate cancer von Myung, Jae-Kyung, Banuelos, Carmen A, Fernandez, Javier Garcia, Mawji, Nasrin R, Wang, Jun, Tien, Amy H, Yang, Yu Chi, Tavakoli, Iran, Haile, Simon, Watt, Kate, McEwan, Iain J, Plymate, Stephen, Andersen, Raymond J, Sadar, Marianne D

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Regression of Castrate-Recurrent Prostate Cancer by a Small-Molecule Inhibitor of the Amino-Terminus Domain of the Androgen Receptor von Andersen, Raymond J., Mawji, Nasrin R., Wang, Jun, Wang, Gang, Haile, Simon, Myung, Jae-Kyung, Watt, Kate, Tam, Teresa, Yang, Yu Chi, Bañuelos, Carmen A., Williams, David E., McEwan, Iain J., Wang, Yuzhou, Sadar, Marianne D.

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Cotargeting Androgen Receptor Splice Variants and mTOR Signaling Pathway for the Treatment of Castration-Resistant Prostate Cancer von Kato, Minoru, Banuelos, Carmen A, Imamura, Yusuke, Leung, Jacky K, Caley, Daniel P, Wang, Jun, Mawji, Nasrin R, Sadar, Marianne D

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Ligand-independent Activation of the Androgen Receptor by Interleukin-6 and the Role of Steroid Receptor Coactivator-1 in Prostate Cancer Cells von Ueda, Takeshi, Mawji, Nasrin R., Bruchovsky, Nicholas, Sadar, Marianne D.

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Characterization of niphatenones that inhibit androgen receptor N-terminal domain von Banuelos, Carmen A, Lal, Aaron, Tien, Amy H, Shah, Neel, Yang, Yu Chi, Mawji, Nasrin R, Meimetis, Labros G, Park, Jacob, Kunzhong, Jian, Andersen, Raymond J, Sadar, Marianne D

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Niphatenones, Glycerol Ethers from the Sponge Niphates digitalis Block Androgen Receptor Transcriptional Activity in Prostate Cancer Cells: Structure Elucidation, Synthesis, and Bi... von Meimetis, Labros G, Williams, David E, Mawji, Nasrin R, Banuelos, Carmen A, Lal, Aaron A, Park, Jacob J, Tien, Amy H, Fernandez, Javier Garcia, de Voogd, Nicole J, Sadar, Marianne D, Andersen, Raymond J

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Inhibition of androgen receptor by decoy molecules delays progression to castration-recurrent prostate cancer von Myung, Jae-Kyung, Wang, Gang, Chiu, Helen H L, Wang, Jun, Mawji, Nasrin R, Sadar, Marianne D

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Pin1 inhibition improves the efficacy of ralaniten compounds that bind to the N-terminal domain of androgen receptor von Leung, Jacky K., Imamura, Yusuke, Kato, Minoru, Wang, Jun, Mawji, Nasrin R., Sadar, Marianne D.

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Androgen receptor decoy molecules block the growth of prostate cancer von Quayle, Steven N, Mawji, Nasrin R, Wang, Jun, Sadar, Marianne D

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Targeting Androgen Receptor Activation Function-1 with EPI to Overcome Resistance Mechanisms in Castration-Resistant Prostate Cancer von Yang, Yu Chi, Banuelos, Carmen Adriana, Mawji, Nasrin R, Wang, Jun, Kato, Minoru, Haile, Simon, McEwan, Iain J, Plymate, Stephen, Sadar, Marianne D

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Spongian diterpenoids inhibit androgen receptor activity von Yang, Yu Chi, Meimetis, Labros G, Tien, Amy H, Mawji, Nasrin R, Carr, Gavin, Wang, Jun, Andersen, Raymond J, Sadar, Marianne D

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An orthotopic metastatic prostate cancer model in SCID mice via grafting of a transplantable human prostate tumor line von Wang, Yuwei, Xue, Hui, Cutz, Jean-Claude, Bayani, Jane, Mawji, Nasrin R, Chen, Wilfred G, Goetz, Lester J, Hayward, Simon W, Sadar, Marianne D, Gilks, C Blake, Gout, Peter W, Squire, Jeremy A, Cunha, Gerald R, Wang, Yu-Zhuo

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Rational optimization of a transcription factor activation domain inhibitor von Basu, Shaon, Martínez-Cristóbal, Paula, Frigolé-Vivas, Marta, Pesarrodona, Mireia, Lewis, Michael, Szulc, Elzbieta, Bañuelos, C. Adriana, Sánchez-Zarzalejo, Carolina, Bielskutė, Stasė, Zhu, Jiaqi, Pombo-García, Karina, Garcia-Cabau, Carla, Zodi, Levente, Dockx, Hannes, Smak, Jordann, Kaur, Harpreet, Batlle, Cristina, Mateos, Borja, Biesaga, Mateusz, Escobedo, Albert, Bardia, Lídia, Verdaguer, Xavier, Ruffoni, Alessandro, Mawji, Nasrin R., Wang, Jun, Obst, Jon K., Tam, Teresa, Brun-Heath, Isabelle, Ventura, Salvador, Meierhofer, David, García, Jesús, Robustelli, Paul, Stracker, Travis H., Sadar, Marianne D., Riera, Antoni, Hnisz, Denes, Salvatella, Xavier

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Structure–Activity Relationships for the Marine Natural Product Sintokamides: Androgen Receptor N‑Terminus Antagonists of Interest for Treatment of Metastatic Castration-Resistant... von Yan, Luping, Banuelos, Carmen A, Mawji, Nasrin R, Patrick, Brian O, Sadar, Marianne D, Andersen, Raymond J

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Sintokamide A Is a Novel Antagonist of Androgen Receptor That Uniquely Binds Activation Function-1 in Its Amino-terminal Domain von Banuelos, Carmen A, Tavakoli, Iran, Tien, Amy H, Caley, Daniel P, Mawji, Nasrin R, Li, Zhenzhen, Wang, Jun, Yang, Yu Chi, Imamura, Yusuke, Yan, Luping, Wen, Jian Guo, Andersen, Raymond J, Sadar, Marianne D

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Ralaniten Sensitizes Enzalutamide-Resistant Prostate Cancer to Ionizing Radiation in Prostate Cancer Cells that Express Androgen Receptor Splice Variants von Banuelos, Carmen A., Ito, Yusuke, Obst, Jon K., Mawji, Nasrin R., Wang, Jun, Hirayama, Yukiyoshi, Leung, Jacky K., Tam, Teresa, Tien, Amy H., Andersen, Raymond J., Sadar, Marianne D.

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Differential Gene Expression Profiles between N-Terminal Domain and Ligand-Binding Domain Inhibitors of Androgen Receptor Reveal Ralaniten Induction of Metallothionein by a Mechani... von Obst, Jon K, Mawji, Nasrin R, Teskey, Simon J L, Wang, Jun, Sadar, Marianne D

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Osteoblast-Derived Factors Induce Androgen-Independent Proliferation and Expression of Prostate-Specific Antigen in Human Prostate Cancer Cells von BLASZCZYK, Natalie, MASRI, Bassam A, SADAR, Marianne D, MAWJI, Nasrin R, UEDA, Takeshi, MCALINDEN, Gavan, DUNCAN, Clive P, BRUCHOVSKY, Nicholas, SCHWEIKERT, Hans-Udo, SCHNABEL, Doris, JONES, Edward C

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Sintokamides A to E, Chlorinated Peptides from the Sponge Dysidea sp. that Inhibit Transactivation of the N-Terminus of the Androgen Receptor in Prostate Cancer Cells von Sadar, Marianne D, Williams, David E, Mawji, Nasrin R, Patrick, Brian O, Wikanta, Thamrin, Chasanah, Ekowati, Irianto, Hari Eko, Soest, Rob Van, Andersen, Raymond J

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An imaging agent to detect androgen receptor and its active splice variants in prostate cancer von Imamura, Yusuke, Tien, Amy H, Pan, Jinhe, Leung, Jacky K, Banuelos, Carmen A, Jian, Kunzhong, Wang, Jun, Mawji, Nasrin R, Fernandez, Javier Garcia, Lin, Kuo-Shyan, Andersen, Raymond J, Sadar, Marianne D

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