Collective synthesis of natural products by means of organocascade catalysis von Jones, Spencer B., Simmons, Bryon, Mastracchio, Anthony, MacMillan, David W. C.

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Enantioselective Organocatalysis Using SOMO Activation von Beeson, Teresa D, Mastracchio, Anthony, Hong, Jun-Bae, Ashton, Kate, MacMillan, David W.C

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Direct and enantioselective α-allylation of ketones via singly occupied molecular orbital (SOMO) catalysis von Mastracchio, Anthony, Warkentin, Alexander A, Walji, Abbas M, MacMillan, David W.C

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Discovery of a Potent and Selective Covalent p300/CBP Inhibitor von Mastracchio, Anthony, Lai, Chunqiu, Digiammarino, Enrico, Ready, Damien B, Lasko, Loren M, Bromberg, Kenneth D, McClellan, William J, Montgomery, Debra, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Patterson, Melanie J, Sun, Chaohong C, Rosenberg, Saul, Lai, Albert, Michaelides, Michael R

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Selective MCL-1 inhibitor ABBV-467 is efficacious in tumor models but is associated with cardiac troponin increases in patients von Yuda, Junichiro, Will, Christine, Phillips, Darren C., Abraham, Linu, Alvey, Cory, Avigdor, Abraham, Buck, Wayne, Besenhofer, Lauren, Boghaert, Erwin, Cheng, Dong, Cojocari, Dan, Doyle, Kelly, Hansen, T. Matthew, Huang, Kevin, Johnson, Eric F., Judd, Andrew S., Judge, Russell A., Kalvass, John C., Kunzer, Aaron, Lam, Lloyd T., Li, Rachel, Martin, Ruth L., Mastracchio, Anthony, Mitten, Mike, Petrich, Adam, Wang, Jin, Ward, James E., Zhang, Haichao, Wang, Xilu, Wolff, Johannes E., Bell-McGuinn, Katherine M., Souers, Andrew J.

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Crystal Structure of Human Phosphodiesterase 3B:  Atomic Basis for Substrate and Inhibitor Specificity von Scapin, Giovanna, Patel, Sangita B, Chung, Christine, Varnerin, Jeffrey P, Edmondson, Scott D, Mastracchio, Anthony, Parmee, Emma R, Singh, Suresh B, Becker, Joseph W, Van der Ploeg, Lex H. T, Tota, Michael R

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Direct and enantioselective {alpha}-allylation of ketones via singly occupied molecular orbital (SOMO) catalysis von Mastracchio, Anthony, Warkentin, Alexander A, Walji, Abbas M, MacMillan, David W C

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Enabling, Decagram-Scale Synthesis of Macrocyclic MCL‑1 Inhibitor ABBV-467 von Brady, Patrick B., Sorensen, Bryan K., Risi, Roberto M., Curtin, Michael L., Mantei, Robert A., Florjancic, Alan S., Mastracchio, Anthony, Ji, Cheng, Kunzer, Aaron R., Lai, Chunqiu, Storer, Gregory E., Chan, Vincent S., Henry, Rodger F., Souers, Andrew J., Michaelides, Michael R., Judd, Andrew S., Hansen, T. Matthew

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Investigation of biaryl heterocycles as inhibitors of Wee1 kinase (vol 29, pg 1481, 2019) von Mastracchio, Anthony, Lai, Chunqiu, Torrent, Maricel, Bromberg, Kenneth, Buchanan, Fritz G., Ferguson, Debra, Bontcheva, Velitchka, Johnson, Eric F., Lasko, Loren, Maag, David, Shoemaker, Alexander R., Penning, Thomas D.

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Interspecies in vitro metabolism of the phosphodiesterase-4 (PDE4) inhibitor L-454,560 von Bateman, Kevin P., Trimble, Laird, Chauret, Nathalie, Silva, Jose, Day, Stephen, Macdonald, Dwight, Dube, Daniel, Gallant, Michel, Mastracchio, Anthony, Perrier, Helene, Girard, Yves, Nicoll-Griffith, Deborah

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Corrigendum to “Investigation of biaryl heterocycles as inhibitors of Wee1 kinase” [Bioorg. Med. Chem. Lett. 29 (2019) 1481–1486] von Mastracchio, Anthony, Lai, Chunqiu, Torrent, Maricel, Bromberg, Kenneth, Buchanan, Fritz G., Ferguson, Debra, Bontcheva, Velitchka, Johnson, Eric F., Lasko, Loren, Maag, David, Shoemaker, Alexander R., Penning, Thomas D.

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Investigation of biaryl heterocycles as inhibitors of Wee1 kinase von Mastracchio, Anthony, Lai, Chunqiu, Torrent, Maricel, Bromberg, Kenneth, Buchanan, Fritz G., Ferguson, Debra, Bontcheva, Velitchka, Johnson, Eric F., Lasko, Loren, Maag, David, Shoemaker, Alexander R., Penning, Thomas D.

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Collective synthesis of natural products by means of organocascade catalysis von Jones, Spencer B, Simmons, Bryon, Mastracchio, Anthony, MacMillan, David W.C

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Balancing Properties with Carboxylates: A Lead Optimization Campaign for Selective and Orally Active CDK9 Inhibitors von Tong, Yunsong, Florjancic, Alan S, Clark, Rick F, Lai, Chunqiu, Mastracchio, Anthony, Zhu, Gui-dong, Smith, Morey L, Kovar, Peter J, Shaw, Bailin, Albert, Daniel H, Qiu, Wei, Longenecker, Kenton L, Liu, Xiaoqin, Olson, Amanda M, Osterling, Donald J, Tahir, Stephen K, Phillips, Darren C, Leverson, Joel D, Souers, Andrew J, Penning, Thomas D

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(2S,3S)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-N,N-dimethyl-4-oxo-2-(4-[1,2,4]triazolo[1,5-a]- pyridin-6-ylphenyl)butanamide:  A Selective α-Amino Amide Dipeptidyl Peptidase IV In... von Edmondson, Scott D, Mastracchio, Anthony, Mathvink, Robert J, He, Jiafang, Harper, Bart, Park, You-Jung, Beconi, Maria, Di Salvo, Jerry, Eiermann, George J, He, Huaibing, Leiting, Barbara, Leone, Joseph F, Levorse, Dorothy A, Lyons, Kathryn, Patel, Reshma A, Patel, Sangita B, Petrov, Aleksandr, Scapin, Giovanna, Shang, Jackie, Roy, Ranabir Sinha, Smith, Aaron, Wu, Joseph K, Xu, Shiyao, Zhu, Bing, Thornberry, Nancy A, Weber, Ann E

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Palladium-Catalyzed Coupling of Vinylogous Amides with Aryl Halides:  Applications to the Synthesis of Heterocycles von Edmondson, Scott D, Mastracchio, Anthony, Parmee, Emma R

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Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: Close analogs of JANUVIA™ (sitagliptin phosphate) von Kim, Dooseop, Kowalchick, Jennifer E., Edmondson, Scott D., Mastracchio, Anthony, Xu, Jinyou, Eiermann, George J., Leiting, Barbara, Wu, Joseph K., Pryor, KellyAnn D., Patel, Reshma A., He, Huaibing, Lyons, Kathryn A., Thornberry, Nancy A., Weber, Ann E.

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Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors von Edmondson, Scott D., Mastracchio, Anthony, Cox, Jason M., Eiermann, George J., He, Huaibing, Lyons, Kathryn A., Patel, Reshma A., Patel, Sangita B., Petrov, Aleksandr, Scapin, Giovanna, Wu, Joseph K., Xu, Shiyao, Zhu, Bing, Thornberry, Nancy A., Roy, Ranabir Sinha, Weber, Ann E.

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Discovery of potent and selective orally bioavailable β-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors von Edmondson, Scott D., Mastracchio, Anthony, Duffy, Joseph L., Eiermann, George J., He, Huaibing, Ita, Ida, Leiting, Barbara, Leone, Joseph F., Lyons, Kathryn A., Makarewicz, Amanda M., Patel, Reshma A., Petrov, Aleksandr, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.

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Potent and selective proline derived dipeptidyl peptidase IV inhibitors von Edmondson, Scott D., Mastracchio, Anthony, Beconi, Maria, Colwell, Lawrence F., Habulihaz, Bahanu, He, Huaibing, Kumar, Sanjeev, Leiting, Barbara, Lyons, Kathryn A., Mao, Ann, Marsilio, Frank, Patel, Reshma A., Wu, Joseph K., Zhu, Lan, Thornberry, Nancy A., Weber, Ann E., Parmee, Emma R.

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