Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279 von Leit, Silvana, Greenwood, Jeremy, Carriero, Samantha, Mondal, Sayan, Abel, Robert, Ashwell, Mark, Blanchette, Heather, Boyles, Nicholas A., Cartwright, Mark, Collis, Alan, Feng, Shulu, Ghanakota, Phani, Harriman, Geraldine C., Hosagrahara, Vinayak, Kaila, Neelu, Kapeller, Rosanna, Rafi, Salma B., Romero, Donna L., Tarantino, Paul M., Timaniya, Jignesh, Toms, Angela V., Wester, Ronald T., Westlin, William, Srivastava, Bhaskar, Miao, Wenyan, Tummino, Peter, McElwee, Joshua J., Edmondson, Scott D., Masse, Craig E.

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Potent and selective TYK2-JH1 inhibitors highly efficacious in rodent model of psoriasis von Leit, Silvana, Greenwood, Jeremy R., Mondal, Sayan, Carriero, Samantha, Dahlgren, Markus, Harriman, Geraldine C., Kennedy-Smith, Joshua J., Kapeller, Rosana, Lawson, Jon P., Romero, Donna L., Toms, Angela V., Shelley, Mee, Wester, Ronald T., Westlin, William, McElwee, Joshua J., Miao, Wenyan, Edmondson, Scott D., Masse, Craig E.

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Anti‐leukaemic activity of the TYK2 selective inhibitor NDI‐031301 in T‐cell acute lymphoblastic leukaemia von Akahane, Koshi, Li, Zhaodong, Etchin, Julia, Berezovskaya, Alla, Gjini, Evisa, Masse, Craig E., Miao, Wenyan, Rocnik, Jennifer, Kapeller, Rosana, Greenwood, Jeremy R., Tiv, Hong, Sanda, Takaomi, Weinstock, David M., Look, A. Thomas

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Syntheses and Biological Evaluation of (+)-Lactacystin and Analogs von Masse, Craig E., Morgan, Adam J., Adams, Julian, Panek, James S.

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X‑ray Crystal Structures of Escherichia coli RNA Polymerase with Switch Region Binding Inhibitors Enable Rational Design of Squaramides with an Improved Fraction Unbound to Human P... von Molodtsov, Vadim, Fleming, Paul R, Eyermann, Charles J, Ferguson, Andrew D, Foulk, Melinda A, McKinney, David C, Masse, Craig E, Buurman, Ed T, Murakami, Katsuhiko S

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A General Method for the Enantioselective Synthesis of Pantolactone Derivatives von Evans, David A, Wu, Jimmy, Masse, Craig E, MacMillan, David W. C

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Cycloaddition Reactions of Imines with 3-Thiosuccinic Anhydrides:  Synthesis of the Tricyclic Core of Martinellic Acid von Ng, Pui Yee, Masse, Craig E, Shaw, Jared T

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Reversal of Regioselection in the Sharpless Asymmetric Aminohydroxylation of Aryl Ester Substrates von Morgan, Adam J, Masse, Craig E, Panek, James S

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Total Synthesis of (+)-Mycotrienol and (+)-Mycotrienin I:  Application of Asymmetric Crotylsilane Bond Constructions von Masse, Craig E, Yang, Michael, Solomon, Jason, Panek, James S

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The Exceptional Chelating Ability of Dimethylaluminum Chloride and Methylaluminum Dichloride. The Merged Stereochemical Impact of α- and β-Stereocenters in Chelate-Controlled Carbo... von Evans, David A, Allison, Brett D, Yang, Michael G, Masse, Craig E

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C 2 -Symmetric Sc(III)-Complexes as Chiral Lewis Acids. Catalytic Enantioselective Aldol Additions to Glyoxylate Esters von Evans, David A, Masse, Craig E, Wu, Jimmy

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Design and synthesis of deuterated boceprevir analogs with enhanced pharmacokinetic properties von Morgan, Adam J., Nguyen, Sophia, Uttamsingh, Vinita, Bridson, Gary, Harbeson, Scott, Tung, Roger, Masse, Craig E.

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Total Synthesis of (+)-Lactacystin von Panek, James S., Masse, Craig E.

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An Asymmetric Aminohydroxylation Approach to the Azepine Core of (−)-Balanol von Masse, Craig E, Morgan, Adam J, Panek, James S

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Lewis Acid-Mediated Carbocyclization Reactions of Chiral (E)-Crotylsilanes von Masse, Craig E, Dakin, Les A, Knight, Bradford S, Panek, James S

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Total Synthesis of (+)-Mycotrienol and (+)-Mycotrienin I von Panek, James S, Masse, Craig E

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Asymmetric C−N Bond Constructions via Crotylsilane Addition Reactions:  A Stereocontrolled Route to Dipeptide Isosteres von Masse, Craig E, Knight, Bradford S, Stavropoulos, Pericles, Panek, James S

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Anti-Leukemic Activity of the TYK2 Selective Inhibitor Ndi-031301 in T-Cell Acute Lymphoblastic Leukemia von Akahane, Koshi, Li, Zhaodong, Etchin, Julia, Berezovskaya, Alla, Gjini, Evisa, Masse, Craig E, Miao, Wenyan, Rocnik, Jennifer, Kapeller, Rosana, Greenwood, Jeremy R, Tiv, Hong, Sanda, Takaomi, Weinstock, David M, Look, A. Thomas

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An Improved Synthesis of (4S,5S)-2-Phenyl-4-methoxycarbonyl-5-isopropyloxazoline from (S)-Phenylglycinol von Panek, James S, Masse, Craig E

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Enantioselective Nitration of Chiral (E)-Crotylsilanes: A Concise Asymmetric Synthesis of (E)-Olefin Dipeptide Isosteres von Beresis, Richard T, Masse, Craig E, Panek, James S

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