Cypin: A novel target for traumatic brain injury von Swiatkowski, Przemyslaw, Sewell, Emily, Sweet, Eric S., Dickson, Samantha, Swanson, Rachel A., McEwan, Sara A., Cuccolo, Nicholas, McDonnell, Mark E., Patel, Mihir V., Varghese, Nevin, Morrison, Barclay, Reitz, Allen B., Meaney, David F., Firestein, Bonnie L.

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Efficient syntheses of KLS-13019 using palladium mediated cross couplings von Kinney, William A., McDonnell, Mark E., Freeman, Stanley, Simons, Nick, Han, Chao, Yang, Lanyi

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Riluzole prodrugs for melanoma and ALS: Design, synthesis, and in vitro metabolic profiling von McDonnell, Mark E., Vera, Matthew D., Blass, Benjamin E., Pelletier, Jeffrey C., King, Richard C., Fernandez-Metzler, Carmen, Smith, Garry R., Wrobel, Jay, Chen, Suzie, Wall, Brian A., Reitz, Allen B.

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Knockdown siRNA Targeting GPR55 Reveals Significant Differences Between the Anti-inflammatory Actions of KLS-13019 and Cannabidiol von Brenneman, Douglas E., Kinney, William A., McDonnell, Mark E., Ippolito, Michael J., Ward, Sara Jane

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Non-NAD-like PARP-1 inhibitors in prostate cancer treatment von Karpova, Yaroslava, Wu, Chao, Divan, Ali, McDonnell, Mark E., Hewlett, Elizabeth, Makhov, Peter, Gordon, John, Ye, Min, Reitz, Allen B., Childers, Wayne E., Skorski, Tomasz, Kolenko, Vladimir, Tulin, Alexei V.

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Anti-Inflammatory Properties of KLS-13019: a Novel GPR55 Antagonist for Dorsal Root Ganglion and Hippocampal Cultures von Brenneman, Douglas E., Kinney, William A., McDonnell, Mark E., Zhao, Pingei, Abood, Mary E., Ward, Sara Jane

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DART.2: bidirectional synaptic pharmacology with thousandfold cellular specificity von Shields, Brenda C., Yan, Haidun, Lim, Shaun S. X., Burwell, Sasha C. V., Cammarata, Celine M., Fleming, Elizabeth A., Yousefzadeh, S. Aryana, Goldenshtein, Victoria Z., Kahuno, Elizabeth W., Vagadia, Purav P., Loughran, Marie H., Zhiquan, Lei, McDonnell, Mark E., Scalabrino, Miranda L., Thapa, Mishek, Hawley, Tammy M., Field, Greg D., Hull, Court, Schiltz, Gary E., Glickfeld, Lindsey L., Reitz, Allen B., Tadross, Michael R.

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The discovery of azetidine-piperazine di-amides as potent, selective and reversible monoacylglycerol lipase (MAGL) inhibitors von Zhu, Bin, Connolly, Peter J., Zhang, Yue-Mei, McDonnell, Mark E., Bian, Haiyan, Lin, Shu-Chen, Liu, Li, Zhang, Sui-Po, Chevalier, Kristen M., Brandt, Michael R., Milligan, Cynthia M., Flores, Christopher M., Macielag, Mark J.

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Discovery of KLS-13019, a Cannabidiol-Derived Neuroprotective Agent, with Improved Potency, Safety, and Permeability von Kinney, William A, McDonnell, Mark E, Zhong, Hua Marlon, Liu, Chaomin, Yang, Lanyi, Ling, Wei, Qian, Tao, Chen, Yu, Cai, Zhijie, Petkanas, Dean, Brenneman, Douglas E

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Crystal structure of a soluble form of human monoglyceride lipase in complex with an inhibitor at 1.35 Å resolution von Schalk‐Hihi, Céline, Schubert, Carsten, Alexander, Richard, Bayoumy, Shariff, Clemente, Jose C., Deckman, Ingrid, DesJarlais, Renee L., Dzordzorme, Keli C., Flores, Christopher M., Grasberger, Bruce, Kranz, James K., Lewandowski, Frank, Liu, Li, Ma, Hongchang, Maguire, Diane, Macielag, Mark J., McDonnell, Mark E., Mezzasalma Haarlander, Tara, Miller, Robyn, Milligan, Cindy, Reynolds, Charles, Kuo, Lawrence C.

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Novel inhibitors of heat shock protein Hsp70-mediated luciferase refolding that bind to DnaJ von Cassel, Joel A., Ilyin, Sergey, McDonnell, Mark E., Reitz, Allen B.

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Anilino-monoindolylmaleimides as potent and selective JAK3 inhibitors von McDonnell, Mark E, Bian, Haiyan, Wrobel, Jay, Smith, Garry R, Liang, Shuguang, Ma, Haiching, Reitz, Allen B

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Characterization of a series of 4-aminoquinolines that stimulate caspase-7 mediated cleavage of TDP-43 and inhibit its function von Cassel, Joel A., McDonnell, Mark E., Velvadapu, Venkata, Andrianov, Vyacheslav, Reitz, Allen B.

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Intramolecular rearrangement of α-amino acid amide derivatives of 2-aminobenzothiazoles von Pelletier, Jeffrey C., Velvadapu, Venkata, McDonnell, Mark E., Wrobel, Jay E., Reitz, Allen B.

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Facile synthesis of mutagen X (MX): 3-chloro-4-(dichloromethyl)-5-hydroxy-5H-furan-2-one von Velvadapu, Venkata, McDonnell, Mark E., Jaffe, Eileen K., Reitz, Allen B.

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Heteroaryl β-tetralin ureas as novel antagonists of human TRPV1 von Jetter, Michele C., Youngman, Mark A., McNally, James J., McDonnell, Mark E., Zhang, Sui-Po, Dubin, Adrienne E., Nasser, Nadia, Codd, Ellen E., Flores, Christopher M., Dax, Scott L.

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N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1) von Jetter, Michele C., McNally, James J., Youngman, Mark A., McDonnell, Mark E., Dubin, Adrienne E., Nasser, Nadia, Zhang, Sui-Po, Codd, Ellen E., Colburn, Ray W., Stone, Dennis R., Brandt, Michael R., Flores, Christopher M., Dax, Scott L.

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Diabetogenic Effect of a Series of Tricyclic Delta Opioid Agonists Structurally Related to Cyproheptadine von Codd, Ellen E., Baker, Judith, Brandt, Michael R., Bryant, Stewart, Cai, Chaozhong, Carson, John R., Chevalier, Kristen M., Colburn, Raymond W., Coogan, Timothy P., Dax, Scott L., DeCorte, Bart, Kemmerer, Michael, LeGrand, Edmund K., Lenhard, James M., Leone, Angelique M., Lin, Ling, Mabus, John R., McDonnell, Mark E., McMillian, Michael K., McNally, James J., Stone, Dennis J., Wang, Charles Y., Zhang, Sui-Po, Flores, Christopher M.

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Synthesis and in vitro evaluation of a novel iodinated resiniferatoxin derivative that is an agonist at the human vanilloid VR1 receptor von MCDONNELL, Mark E, ZHANG, Sui-Po, DUBIN, Adrienne E, DAX, Scott L

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7-Hydroxynaphthalen-1-yl-urea and -amide antagonists of human vanilloid receptor 1 von McDonnell, Mark E., Zhang, Sui-Po, Nasser, Nadia, Dubin, Adrienne E., Dax, Scott L.

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