Palladium-Catalyzed Synthesis of Functionalized Tetraarylphosphonium Salts von Marcoux, David, Charette, André B

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Nickel‐Catalyzed Synthesis of Phosphonium Salts from Aryl Halides and Triphenylphosphine von Marcoux, David, Charette, André B.

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General Method for the Synthesis of Phenyliodonium Ylides from Malonate Esters: Easy Access to 1,1-Cyclopropane Diesters von Goudreau, Sébastien R, Marcoux, David, Charette, André B

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trans-Directing Ability of the Amide Group: Enabling the Enantiocontrol in the Synthesis of 1,1-Dicarboxy Cyclopropanes. Reaction Development, Scope, and Synthetic Applications von Marcoux, David, Goudreau, Sébastien R, Charette, André B

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Use of achiral additives to increase the stereoselectivity in Rh(II)-catalyzed cyclopropanations von Marcoux, David, Lindsay, Vincent N G, Charette, André B

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Removal, Recovery, and Recycling of Triarylphosphonium-Supported Tin Reagents for Various Organic Transformations von Poupon, Jean-Christophe, Marcoux, David, Cloarec, Jean-Manuel, Charette, André B

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TfNH2 as Achiral Hydrogen-Bond Donor Additive to Enhance the Selectivity of a Transition Metal Catalyzed Reaction. Highly Enantio- and Diastereoselective Rhodium-Catalyzed Cyclopro... von Marcoux, David, Azzi, Soula, Charette, André B

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Tricyclic-Carbocyclic RORγt Inverse AgonistsDiscovery of BMS-986313 von Yang, Michael G, Beaudoin-Bertrand, Myra, Xiao, Zili, Marcoux, David, Weigelt, Carolyn A, Yip, Shiuhang, Wu, Dauh-Rurng, Ruzanov, Max, Sack, John S, Wang, Jinhong, Yarde, Melissa, Li, Sha, Shuster, David J, Xie, Jenny H, Sherry, Tara, Obermeier, Mary T, Fura, Aberra, Stefanski, Kevin, Cornelius, Georgia, Khandelwal, Purnima, Karmakar, Ananta, Basha, Mushkin, Babu, Venkatesh, Gupta, Arun Kumar, Mathur, Arvind, Salter-Cid, Luisa, Denton, Rex, Zhao, Qihong, Dhar, T. G. Murali

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Rationally Designed, Conformationally Constrained Inverse Agonists of RORγtIdentification of a Potent, Selective Series with Biologic-Like in Vivo Efficacy von Marcoux, David, Duan, James J.-W, Shi, Qing, Cherney, Robert J, Srivastava, Anurag S, Cornelius, Lyndon, Batt, Douglas G, Liu, Qingjie, Beaudoin-Bertrand, Myra, Weigelt, Carolyn A, Khandelwal, Purnima, Vishwakrishnan, Sureshbabu, Selvakumar, Kumaravel, Karmakar, Ananta, Gupta, Arun Kumar, Basha, Mushkin, Ramlingam, Sridharan, Manjunath, Naveen, Vanteru, Sridhar, Karmakar, Sukhen, Maddala, Nageswara, Vetrichelvan, Muthalagu, Gupta, Anuradha, Rampulla, Richard A, Mathur, Arvind, Yip, Shiuhang, Li, Peng, Wu, Dauh-Rurng, Khan, Javed, Ruzanov, Max, Sack, John S, Wang, Jinhong, Yarde, Melissa, Cvijic, Mary Ellen, Li, Sha, Shuster, David J, Borowski, Virna, Xie, Jenny H, McIntyre, Kim W, Obermeier, Mary T, Fura, Aberra, Stefanski, Kevin, Cornelius, Georgia, Hynes, John, Tino, Joseph A, Macor, John E, Salter-Cid, Luisa, Denton, Rex, Zhao, Qihong, Carter, Percy H, Dhar, T. G. Murali

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One-Step Diastereoselective Pyrrolidine Synthesis Using a Sulfinamide Annulating Reagent von Shi, Qing, Greenwood, Nathaniel S, Meehan, Mariah C, Park, Hyunsoo, Galella, Michael, Sandhu, Bhupinder, Khandelwal, Purnima, Coombs, John R, Gallagher, William P, Guerrero, Carlos A, Hynes, John, Dhar, T. G. Murali, Gonzalez Bobes, Francisco, Marcoux, David

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trans-Directing Ability of Amide Groups in Cyclopropanation: Application to the Asymmetric Cyclopropanation of Alkenes with Diazo Reagents Bearing Two Carboxy Groups von Marcoux, David, Charette, André B

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Discovery of Annulating Reagents Enabling the One-Step and Highly Stereoselective Synthesis of Cyclopentyl and Cyclohexyl Cores von McDaniel, Jade, Farley, Christopher A, Ramirez, Antonio, Sandhu, Bhupinder, Sarjeant, Amy, Shi, Qing, Han, Arthur, Gallagher, William P, Hynes, John, Dhar, T. G. Murali, Gonzalez-Bobes, Francisco, Coombs, John R, Marcoux, David

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Annulation reaction enables the identification of an exocyclic amide tricyclic chemotype as retinoic acid Receptor-Related orphan receptor gamma (RORγ/RORc) inverse agonists von Marcoux, David, Bertrand, Myra Beaudoin, Weigelt, Carolyn A., Yip, Shiuhang, Galella, Michael, Park, Hyunsoo, Wu, Dauh-Rurng, Wang, Jinhong, Yarde, Melissa, Cvijic, Mary Ellen, Li, Sha, Hynes, John, Tino, Joseph A., Zhao, Qihong, Dhar, T.G. Murali

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Protected Chloroethyl and Chloropropyl Amines as Conformationally Unrestricted Annulating Reagents von Shi, Qing, Meehan, Mariah C, Galella, Michael, Park, Hyunsoo, Khandelwal, Purnima, Hynes, John, Dhar, T. G. Murali, Marcoux, David

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Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist von Cherney, Robert J., Cornelius, Lyndon A. M., Srivastava, Anurag, Weigelt, Carolyn A., Marcoux, David, Duan, James J.-W., Shi, Qing, Batt, Douglas G., Liu, Qingjie, Yip, Shiuhang, Wu, Dauh-Rurng, Ruzanov, Max, Sack, John, Khan, Javed, Wang, Jinhong, Yarde, Melissa, Cvijic, Mary Ellen, Mathur, Arvind, Li, Sha, Shuster, David, Khandelwal, Purnima, Borowski, Virna, Xie, Jenny, Obermeier, Mary, Fura, Aberra, Stefanski, Kevin, Cornelius, Georgia, Tino, Joseph A., Macor, John E., Salter-Cid, Luisa, Denton, Rex, Zhao, Qihong, Carter, Percy H., Dhar, T. G. Murali

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Tricyclic sulfones as potent, selective and efficacious RORγt inverse agonists – Exploring C6 and C8 SAR using late-stage functionalization von Shi, Qing, Xiao, Zili, Yang, Michael G., Marcoux, David, Cherney, Robert J., Yip, Shiuhang, Li, Peng, Wu, Dauh-Rurng, Weigelt, Carolyn A., Sack, John, Khan, Javed, Ruzanov, Max, Wang, Jinhong, Yarde, Melissa, Ellen Cvijic, Mary, Li, Sha, Shuster, David J., Xie, Jenny, Sherry, Tara, Obermeier, Mary, Fura, Aberra, Stefanski, Kevin, Cornelius, Georgia, Chacko, Silvi, Shu, Yue-Zhong, Khandelwal, Purnima, Hynes, John, Tino, Joseph A., Salter-Cid, Luisa, Denton, Rex, Zhao, Qihong, Dhar, T.G. Murali

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Identification of highly potent and selective PI3Kδ inhibitors von Marcoux, David, Qin, Lan-Ying, Ruan, Zheming, Shi, Qing, Ruan, Qian, Weigelt, Carolyn, Qiu, Hongchen, Schieven, Gary, Hynes, John, Bhide, Rajeev, Poss, Michael, Tino, Joseph

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Angiographic Selective Methylene Blue Staining of an Occult Small-Bowel Arteriovenous Malformation von Schechter, Steven, Deorchis, Douglas, Bass, James, Marcoux, David A.

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TfNH 2 as Achiral Hydrogen-Bond Donor Additive to Enhance the Selectivity of a Transition Metal Catalyzed Reaction. Highly Enantio- and Diastereoselective Rhodium-Catalyzed Cyclopr... von Marcoux, David, Azzi, Soula, Charette, André B.

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Aryl Ether-Derived Sphingosine-1-Phosphate Receptor (S1P1) Modulators: Optimization of the PK, PD, and Safety Profiles von Xiao, Zili, Yang, Michael G, Dhar, T. G. Murali, Xiao, Hai-Yun, Gilmore, John L, Marcoux, David, McIntyre, Kim W, Taylor, Tracy L, Shi, Hong, Levesque, Paul C, Marino, Anthony M, Cornelius, Georgia, Mathur, Arvind, Shen, Ding Ren, Cvijic, Mary Ellen, Lehman-McKeeman, Lois D, Sun, Huadong, Xie, Jenny H, Carter, Percy H, Dyckman, Alaric J

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