Metal‐Free Cross‐Dehydrogenative Coupling (CDC): Molecular Iodine as a Versatile Catalyst/Reagent for CDC Reactions von Parvatkar, Prakash T., Manetsch, Roman, Banik, Bimal K.

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The emergence of sulfo-click amidation in kinetic target-guided synthesis von Parvatkar, Prakash T., Manetsch, Roman

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Total synthesis of (±)-decursivine via BINOL-phosphoric acid catalyzed tandem oxidative cyclization von Parvatkar, Prakash T., Smotkin, Eugene S., Manetsch, Roman

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Sulfo-click reaction via in situ generated thioacids and its application in kinetic target-guided synthesis von Namelikonda, Niranjan Kumar, Manetsch, Roman

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In Situ Selection of Lead Compounds by Click Chemistry:  Target-Guided Optimization of Acetylcholinesterase Inhibitors von Krasiński, Antoni, Radić, Zoran, Manetsch, Roman, Raushel, Jessica, Taylor, Palmer, Sharpless, K. Barry, Kolb, Hartmuth C.

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Streptothricin F is a bactericidal antibiotic effective against highly drug-resistant gram-negative bacteria that interacts with the 30S subunit of the 70S ribosome von Morgan, Christopher E, Kang, Yoon-Suk, Green, Alex B, Smith, Kenneth P, Dowgiallo, Matthew G, Miller, Brandon C, Chiaraviglio, Lucius, Truelson, Katherine A, Zulauf, Katelyn E, Rodriguez, Shade, Kang, Anthony D, Manetsch, Roman, Yu, Edward W, Kirby, James E

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Evaluating protein cross-linking as a therapeutic strategy to stabilize SOD1 variants in a mouse model of familial ALS von Hossain, Md Amin, Sarin, Richa, Donnelly, Daniel P, Miller, Brandon C, Weiss, Alexandra, McAlary, Luke, Antonyuk, Svetlana V, Salisbury, Joseph P, Amin, Jakal, Conway, Jeremy B, Watson, Samantha S, Winters, Jenifer N, Xu, Yu, Alam, Novera, Brahme, Rutali R, Shahbazian, Haneyeh, Sivasankar, Durgalakshmi, Padmakumar, Swathi, Sattarova, Aziza, Ponmudiyan, Aparna C, Gawde, Tanvi, Verrill, David E, Yang, Wensheng, Kannapadi, Sunanda, Plant, Leigh D, Auclair, Jared R, Makowski, Lee, Petsko, Gregory A, Ringe, Dagmar, Agar, Nathalie Y R, Greenblatt, David J, Ondrechen, Mary Jo, Chen, Yunqiu, Yerbury, Justin J, Manetsch, Roman, Hasnain, S Samar, Brown, Jr, Robert H, Agar, Jeffrey N

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Progress in the Optimization of 4(1 H )-Quinolone Derivatives as Antimalarials Targeting the Erythrocytic, the Exoerythrocytic and the Transmitting Stages of the Malaria Parasite von Brockmeyer, Fabian, Manetsch, Roman

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Antileishmanial activity of a series of N²,N⁴-disubstituted quinazoline-2,4-diamines von Van Horn, Kurt S, Zhu, Xiaohua, Pandharkar, Trupti, Yang, Sihyung, Vesely, Brian, Vanaerschot, Manu, Dujardin, Jean-Claude, Rijal, Suman, Kyle, Dennis E, Wang, Michael Zhuo, Werbovetz, Karl A, Manetsch, Roman

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Naegleria fowleri: Protein structures to facilitate drug discovery for the deadly, pathogenic free-living amoeba von Tillery, Logan, Barrett, Kayleigh, Goldstein, Jenna, Lassner, Jared W, Osterhout, Bram, Tran, Nathan L, Xu, Lily, Young, Ryan M, Craig, Justin, Chun, Ian, Dranow, David M, Abendroth, Jan, Delker, Silvia L, Davies, Douglas R, Mayclin, Stephen J, Calhoun, Brandy, Bolejack, Madison J, Staker, Bart, Subramanian, Sandhya, Phan, Isabelle, Lorimer, Donald D, Myler, Peter J, Edwards, Thomas E, Kyle, Dennis E, Rice, Christopher A, Morris, James C, Leahy, James W, Manetsch, Roman, Barrett, Lynn K, Smith, Craig L, Van Voorhis, Wesley C

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Efficient Biomimetic Total Synthesis, Characterization, and Antioxidant Activity of Ommatins von Huang, Lili, Kim, Taehwan, Armendarez, Olivia J., Deravi, Leila F., Parvatkar, Prakash T., Manetsch, Roman

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Design, synthesis and photoactivation studies of fluorous photolabels von Kumar, Arun Babu, Anderson, Jordan Micheal, Manetsch, Roman

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A Phenotypic Screen for the Liver Stages of Plasmodium vivax von Maher, Steven P, Vantaux, Amélie, Cooper, Caitlin A, Chasen, Nathan M, Cheng, Wayne T, Joyner, Chester J, Manetsch, Roman, Witkowski, Benoît, Kyle, Dennis

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4-(1H)-Quinolones and 1,2,3,4-Tetrahydroacridin-9(10H)-Ones Prevent the Transmission of Plasmodium falciparum to Anopheles freeborni von SAENZ, Fabián E, LACRUE, Alexis N, CROSS, R. Matthew, MAIGNAN, Jordany R, UDENZE, Kenneth O, MANETSCH, Roman, KYLE, Dennis E

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Screening of Protein–Protein Interaction Modulators via Sulfo-Click Kinetic Target-Guided Synthesis von Kulkarni, Sameer S, Hu, Xiangdong, Doi, Kenichiro, Wang, Hong-Gang, Manetsch, Roman

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Synthesis and structure–activity relationship studies of 1,3-disubstituted 2-propanols as BACE-1 inhibitors von Kumar, Arun Babu, Anderson, Jordan Micheal, Melendez, Anthony Lester, Manetsch, Roman

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4(1H)-Quinolones with Liver Stage Activity against Plasmodium berghei von LACRUE, Alexis N, SAENZ, Fabián E, CROSS, R. Matthew, UDENZE, Kenneth O, MONASTYRSKYI, Andrii, STEIN, Steven, MUTKA, Tina S, MANETSCH, Roman, KYLE, Dennis E

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Antibacterial activity of a series of N2,N4-disubstituted quinazoline-2,4-diamines von Van Horn, Kurt S, Burda, Whittney N, Fleeman, Renee, Shaw, Lindsey N, Manetsch, Roman

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Kinetic target-guided synthesis von Hu, Xiangdong, Manetsch, Roman

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Synthesis and evaluation of a novel adenosine-ribose probe for global-scale profiling of nucleoside and nucleotide-binding proteins von Mahajan, Shikha, Manetsch, Roman, Merkler, David J, Stevens, Jr, Stanley M

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