Novel Peptidyl Phosphorus Derivatives as Inhibitors of Human Calpain I von Tao, Ming, Bihovsky, Ron, Wells, Gregory J, Mallamo, John P

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Neurotrophic 3,9-Bis[(alkylthio)methyl]- and -Bis(alkoxymethyl)-K-252a Derivatives von Kaneko, Masami, Saito, Yutaka, Saito, Hiromitsu, Matsumoto, Tadashi, Matsuda, Yuzuru, Vaught, Jeffry L, Dionne, Craig A, Angeles, Thelma S, Glicksman, Marcie A, Neff, Nicola T, Rotella, David P, Kauer, James C, Mallamo, John P, Hudkins, Robert L, Murakata, Chikara

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d-Amino Acid Containing, High-Affinity Inhibitors of Recombinant Human Calpain I von Chatterjee, Sankar, Gu, Zi-Qiang, Dunn, Derek, Tao, Ming, Josef, Kurt, Tripathy, Rabindranath, Bihovsky, Ron, Senadhi, Shobha E, O'Kane, Teresa M, McKenna, Beth Ann, Mallya, Satish, Ator, Mark A, Bozyczko-Coyne, Donna, Siman, Robert, Mallamo, John P

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Synthesis and Biological Activity of a Series of Potent Fluoromethyl Ketone Inhibitors of Recombinant Human Calpain I von Chatterjee, Sankar, Ator, Mark A, Bozyczko-Coyne, Donna, Josef, Kurt, Wells, Gregory, Tripathy, Rabindranath, Iqbal, Mohamed, Bihovsky, Ron, Senadhi, Shobha E, Mallya, Satish, O'Kane, Teresa M, McKenna, Beth Ann, Siman, Robert, Mallamo, John P

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Antipicornavirus activity of tetrazole analogs related to disoxaril von Diana, Guy D, Cutcliffe, David, Volkots, Deborah L, Mallamo, John P, Bailey, Thomas R, Vescio, Niranjan, Oglesby, Richard C, Nitz, Theodore J, Wetzel, Joseph

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Prodrug esters of the indolocarbazole CEP-751 (KT-6587) von Hudkins, Robert L., Iqbal, Mohamed, Park, Chung-Ho, Goldstein, Joel, Herman, Joseph L., Shek, Efraim, Murakata, Chikara, Mallamo, John P.

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Knowledge-based chemoinformatic approaches to drug discovery von Ghose, Arup K., Herbertz, Torsten, Salvino, Joseph M., Mallamo, John P.

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WIN 63480, a hydrophilic TCP-site ligand, has reduced agonist-independent NMDA ion channel access compared to MK-801 and phencyclidine von Ault, B., Miller, M.S., Kelly, M.D., Hildebrand, L.M., Earley, W.G., Luttinger, D., Mallamo, J.P., Ward, S.J.

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P2-ACHIRAL, P'-extended α-ketoamide inhibitors of calpain I von CHATTERJEE, S, DUNN, D, MING TAO, WELLS, G, GU, Z.-Q, BIHOVSKY, R, ATOR, M. A, SIMAN, R, MALLAMO, J. P

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Synthesis and Mixed Lineage Kinase Activity of Pyrrolocarbazole and Isoindolone Analogs of (+)K-252a von Hudkins, Robert L, Johnson, Neil W, Angeles, Thelma S, Gessner, George W, Mallamo, John P

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Novel Benzo[b]quinolizinium Cations as Uncompetitive N-Methyl-D-aspartic Acid (NMDA) Antagonists: The Relationship between log D and Agonist Independent (Closed) NMDA Channel Block von Earley, William G, Kumar, Virendra, Mallamo, John P, Subramanyam, Chakrapani, Dority, John A, Miller, Matthew S, DeHaven-Hudkins, Diane L, Aimone, Lisa D, Kelly, Michael D, Ault, Brian

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Identification, Synthesis, and Characterization of a Unique Class of N-Methyl-D-aspartate Antagonists. The 6,11-Ethanobenzo[b]quinolizinium Cation von Mallamo, John P, Earley, William G, Kumar, Virendra, Subramanyam, Chakrapani, Dority, John A. Jr, Miller, Matthew S, DeHaven-Hudkins, Diane L, Ault, Brian, Herrmann, John L

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Knowledge-Based, Central Nervous System (CNS) Lead Selection and Lead Optimization for CNS Drug Discovery von Ghose, Arup K, Herbertz, Torsten, Hudkins, Robert L, Dorsey, Bruce D, Mallamo, John P

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Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles von Mallamo, John P, Pilling, Garry M, Wetzel, Joseph R, Kowalczyk, Paul J, Bell, Malcolm R, Kullnig, Rudolph K, Batzold, Frederick H, Juniewicz, Paul E, Winneker, Richard C, Luss, Henry R

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Synthesis and structure-activity studies of some disubstituted phenylisoxazoles against human picornavirus von Diana, Guy D, Cutcliffe, David, Oglesby, Richard C, Otto, Michael J, Mallamo, John P, Akullian, Vahan, McKinlay, Mark A

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Calpain inhibitors based on the quiescent affinity label concept: high rates of calpain inactivation with leaving groups derived from N-hydroxy peptide coupling reagents von Tripathy, Rabindranath, Ator, Mark A., Mallamo, John P.

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An Evaluation of the Antirhinoviral Activity of Acylfuran Replacements for 3-Methylisoxazoles. Are 2-Acetylfurans Bioisosteres for 3-Methylisoxazoles? von Bailey, Thomas R, Diana, Guy D, Mallamo, John P, Vescio, Niranjan, Draper, Tandy L, Carabateas, Philip M, Long, Melody A, Giranda, Vincent L, Dutko, Frank J, Pevear, Daniel C

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Synthesis and Evaluation of 6,11-Ethanohexahydrobenzo[b]quinolizidines: A New Class of Noncompetitive N-Methyl-D-aspartate Antagonists von Subramanyam, Chakrapani, Mallamo, John P, Pilling, Gary M, Earley, William G, Carabateas, Philip M, Wetzel, Joseph R, DeHaven-Hudkins, Diane, Allen, Timothy, Kullnig, Rudolph K

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Novel NMDA Antagonists: Replacement of the Pyridinium Ring of 6,11-Ethanobenzo[b]quinolizinium Cations with Heteroisoquinolinium Cations von Kumar, Virendra, Carabateas, Phil M, Dority, John A, Earley, William G, Mallamo, John P, Subramanyam, Chakrapani, Aimone, Lisa D, Ault, Brian, Hudkins, Diane L. DeHaven, Miller, Matthew S

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Antiandrogenic steroidal sulfonylpyrazoles von Christiansen, Robert G, Bell, Malcolm R, D'Ambra, Thomas E, Mallamo, John P, Herrmann, John L, Ackerman, James H, Opalka, Chester J, Kullnig, Rudolph K, Winneker, Richard C

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