High-Throughput Optimization of Ir-Catalyzed C–H Borylation: A Tutorial for Practical Applications von Preshlock, Sean M, Ghaffari, Behnaz, Maligres, Peter E, Krska, Shane W, Maleczka, Robert E, Smith, Milton R

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A Traceless Directing Group for CH Borylation von Preshlock, Sean M., Plattner, Donald L., Maligres, Peter E., Krska, Shane W., Maleczka Jr, Robert E., Smith III, Milton R.

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Asymmetric Synthesis of Cyclic Indole Aminals via 1,3-Stereoinduction von Li, Hongmei, Chen, Cheng-yi, Nguyen, Hoa, Cohen, Ryan, Maligres, Peter E, Yasuda, Nobuyoshi, Mangion, Ian, Zavialov, Ilia, Reibarkh, Mikhail, Chung, John Y. L

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Engineered Ribosyl-1-Kinase Enables Concise Synthesis of Molnupiravir, an Antiviral for COVID-19 von McIntosh, John A, Benkovics, Tamas, Silverman, Steven M, Huffman, Mark A, Kong, Jongrock, Maligres, Peter E, Itoh, Tetsuji, Yang, Hao, Verma, Deeptak, Pan, Weilan, Ho, Hsing-I, Vroom, Jonathan, Knight, Anders M, Hurtak, Jessica A, Klapars, Artis, Fryszkowska, Anna, Morris, William J, Strotman, Neil A, Murphy, Grant S, Maloney, Kevin M, Fier, Patrick S

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Organocatalytic Conversion of Nucleosides to Furanoid Glycals von Mao, Edna, Chung, Cheol K, Ji, Yining, Lam, Yu-hong, Maligres, Peter E

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Silyl Phosphorus and Nitrogen Donor Chelates for Homogeneous Ortho Borylation Catalysis von Ghaffari, Behnaz, Preshlock, Sean M, Plattner, Donald L, Staples, Richard J, Maligres, Peter E, Krska, Shane W, Maleczka, Robert E, Smith, Milton R

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CO Cross-Coupling of Activated Aryl and Heteroaryl Halides with Aliphatic Alcohols von Maligres, Peter E., Li, Jing, Krska, Shane W., Schreier, John D., Raheem, Izzat T.

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Bismuth Acetate as a Catalyst for the Sequential Protodeboronation of Di- and Triborylated Indoles von Shen, Fangyi, Tyagarajan, Sriram, Perera, Damith, Krska, Shane W, Maligres, Peter E, Smith, Milton R, Maleczka, Robert E

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Discovery and Development of an Unusual Organocatalyst for the Conversion of Thymidine to Furanoid Glycal von Maligres, Peter E, Chung, Cheol K, Dance, Zachary E. X, Mattern, Keith A, Phillips, Eric M, Poirier, Marc, Sirk, Kevin M, Wright, Timothy J

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A Soluble Copper(I) Source and Stable Salts of Volatile Ligands for Copper-Catalyzed C–X Couplings von Maligres, Peter E, Krska, Shane W, Dormer, Peter G

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Enantioselective Synthesis of α‑Methyl-β-cyclopropyldihydrocinnamates von Christensen, Melodie, Nolting, Andrew, Shevlin, Michael, Weisel, Mark, Maligres, Peter E, Lee, Joshua, Orr, Robert K, Plummer, Christopher W, Tudge, Matthew T, Campeau, Louis-Charles, Ruck, Rebecca T

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Efficient synthesis of antiviral agent uprifosbuvir enabled by new synthetic methods von Klapars, Artis, Chung, John Y. L, Limanto, John, Calabria, Ralph, Campeau, Louis-Charles, Campos, Kevin R, Chen, Wenyong, Dalby, Stephen M, Davis, Tyler A, DiRocco, Daniel A, Hyde, Alan M, Kassim, Amude M, Larsen, Mona Utne, Liu, Guiquan, Maligres, Peter E, Moment, Aaron, Peng, Feng, Ruck, Rebecca T, Shevlin, Michael, Simmons, Bryon L, Song, Zhiguo Jake, Tan, Lushi, Wright, Timothy J, Zultanski, Susan L

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Diverse Catalytic Reactions for the Stereoselective Synthesis of Cyclic Dinucleotide MK-1454 von Benkovics, Tamas, Peng, Feng, Phillips, Eric M, An, Chihui, Bade, Rachel S, Chung, Cheol K, Dance, Zachary E. X, Fier, Patrick S, Forstater, Jacob H, Liu, Zhijian, Liu, Zhuqing, Maligres, Peter E, Marshall, Nicholas M, Salehi Marzijarani, Nastaran, McIntosh, John A, Miller, Steven P, Moore, Jeffrey C, Neel, Andrew J, Obligacion, Jennifer V, Pan, Weilan, Pirnot, Michael T, Poirier, Marc, Reibarkh, Mikhail, Sherry, Benjamin D, Song, Zhiguo Jake, Tan, Lushi, Turnbull, Ben W. H, Verma, Deeptak, Waldman, Jacob H, Wang, Lu, Wang, Tao, Winston, Matthew S, Xu, Feng

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A Synthesis of a Spirocyclic Macrocyclic Protease Inhibitor for the Treatment of Hepatitis C von Chung, Cheol K, Cleator, Ed, Dumas, Aaron M, Hicks, Jacqueline D, Humphrey, Guy R, Maligres, Peter E, Nolting, Andrew F, Rivera, Nelo, Ruck, Rebecca T, Shevlin, Michael

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An approach to heterodiarylmethanes via sp2–sp3 Suzuki−Miyaura cross-coupling von Stewart, Gavin W., Maligres, Peter E., Baxter, Carl A., Junker, Ellyn M., Krska, Shane W., Scott, Jeremy P.

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Development of a Second-Generation, Highly Efficient Manufacturing Route for the HIV Integrase Inhibitor Raltegravir Potassium von Humphrey, Guy R, Pye, Philip J, Zhong, Yong-Li, Angelaud, Remy, Askin, David, Belyk, Kevin M, Maligres, Peter E, Mancheno, Danny E, Miller, Ross A, Reamer, Robert A, Weissman, Steven A

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A highly catalytic robust palladium catalyzed cyanation of aryl bromides von Maligres, Peter E., Waters, Marjorie S., Fleitz, Fred, Askin, David

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Selective Synthesis of N 6,3′,5′-Tripivaloyladenosine via Dynamic Kinetic Crystallization and Regioselective Preparation of Pivalated 2′-Deoxy-2′-fluoroarabinoadenosines von Maligres, Peter E., Song, Zhiguo Jake, Chen, Lu, Kosjek, Birgit, Ad, Omer, Chung, Cheol K.

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Highly Regioselective DABCO-Catalyzed Nucleophilic Aromatic Substitution (SNAr) Reaction of Methyl 2,6-Dichloronicotinate with Phenols von Shi, Yao-Jun, Humphrey, Guy, Maligres, Peter E., Reamer, Robert A., Williams, J. Michael

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Practical, Highly Convergent, Asymmetric Synthesis of a Selective PPARγ Modulator von Maligres, Peter E, Humphrey, Guy R, Marcoux, Jean-François, Hillier, Michael C, Zhao, Dalian, Krska, Shane, Grabowski, Edward J. J

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