Directed Remote Aromatic Metalations: Mechanisms and Driving Forces von Tilly, David, Magolan, Jakob, Mortier, Jacques

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Uncovering the Hidden Antibiotic Potential of Cannabis von Farha, Maya A, El-Halfawy, Omar M, Gale, Robert T, MacNair, Craig R, Carfrae, Lindsey A, Zhang, Xiong, Jentsch, Nicholas G, Magolan, Jakob, Brown, Eric D

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A platform for predicting mechanism of action based on bacterial transcriptional responses identifies an unusual DNA gyrase inhibitor von French, Shawn, Guo, Amelia Bing Ya, Ellis, Michael J., Deisinger, Julia P., Johnson, Jarrod W., Rachwalski, Kenneth, Piquette, Zoë A., Lluka, Telmah, Zary, Miranda, Gamage, Sineli, Magolan, Jakob, Brown, Eric D.

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Combined Pd/C and Montmorillonite Catalysis for One-Pot Synthesis of Benzimidazoles von Weires, Nicholas A., Boster, Jared, Magolan, Jakob

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Bromination of Olefins with HBr and DMSO von Karki, Megha, Magolan, Jakob

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Evaluation of synthetic coumarins for antiausterity cytotoxicity against pancreatic cancers von Farley, Conner M., Dibwe, Dya Fita, Ueda, Jun-ya, Hall, Eric A., Awale, Suresh, Magolan, Jakob

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Expanding the Scope of Mn(OAc)3-Mediated Cyclizations:  Synthesis of the Tetracyclic Core of Tronocarpine von Magolan, Jakob, Kerr, Michael A

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Dimethyl Sulfoxide as a Synthon in Organic Chemistry von Jones-Mensah, Ebenezer, Karki, Megha, Magolan, Jakob

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A screen for cell envelope stress uncovers an inhibitor of prolipoprotein diacylglyceryl transferase, Lgt, in Escherichia coli von Rachwalski, Kenneth, Madden, Sean J., Ritchie, Nicole, French, Shawn, Bhando, Timsy, Girgis-Gabardo, Adele, Tu, Megan, Gordzevich, Rodion, Ives, Rowan, Guo, Amelia B.Y., Johnson, Jarrod W., Xu, Yiming, Kapadia, Sharookh B., Magolan, Jakob, Brown, Eric D.

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Aryl methyl sulfides via SNAr using DMSO as the source of the thiomethyl moiety von Jones-Mensah, Ebenezer, Magolan, Jakob

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Novel caffeine derivatives mitigate hyperlipidemia by reducing PCSK9 expression and secretion von Stouth, Derek, Magolan, Jakob, Pare, Guillaume, Tarnopolsky, Mark, Macdonald, Melissa, Sguazzin, Matthew, Austin, Richard

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Use of Vinyl Sulfides in Fischer Indole Reactions von Pal, Parul, Fragis, Meghan, Dharavath, Srinivas, Johnson, Jarrod W., Magolan, Jakob

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Allosteric inhibition of tRNA synthetase Gln4 by N-pyrimidinyl-β-thiophenylacrylamides exerts highly selective antifungal activity von Puumala, Emily, Sychantha, David, Lach, Elizabeth, Reeves, Shawn, Nabeela, Sunna, Fogal, Meea, Nigam, AkshatKumar, Johnson, Jarrod W., Aspuru-Guzik, Alán, Shapiro, Rebecca S., Uppuluri, Priya, Kalyaanamoorthy, Subha, Magolan, Jakob, Whitesell, Luke, Robbins, Nicole, Wright, Gerard D., Cowen, Leah E.

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Bioactivity of the cannabigerol cannabinoid and its analogues - the role of 3-dimensional conformation von Salha, Mohammed, Adenusi, Henry, Dupuis, John H, Bodo, Enrico, Botta, Bruno, McKenzie, Iain, Yada, Rickey Y, Farrar, David H, Magolan, Jakob, Tian, Kun V, Chass, Gregory A

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Total Synthesis of (+)-Angelmarin von Magolan, Jakob, Coster, Mark J

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Targeting SUMOylation dependency in human cancer stem cells through a unique SAE2 motif revealed by chemical genomics von Benoit, Yannick D., Mitchell, Ryan R., Wang, Wenliang, Orlando, Luca, Boyd, Allison L., Tanasijevic, Borko, Aslostovar, Lili, Shapovalova, Zoya, Doyle, Meaghan, Bergin, Christopher J., Vojnits, Kinga, Casado, Fanny L., Di Lu, Justin, Porras, Deanna P., García-Rodriguez, Juan Luis, Russell, Jennifer, Zouggar, Aïcha, Masibag, Angelique N., Caba, Cody, Koteva, Kalinka, Kinthada, Lakshmana K., Patel, Jagdish Suresh, Andres, Sara N., Magolan, Jakob, Collins, Tony J., Wright, Gerard D., Bhatia, Mickie

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Biaryl Ketones by Suzuki-Miyaura Cross-Coupling of Organotrifluoroborates and Acyl Chlorides von Forbes, Alaina M., Meier, G. Patrick, Jones-Mensah, Ebenezer, Magolan, Jakob

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QSAR models reveal new EPAC-selective allosteric modulators von Mohamed, Hebatallah, Shao, Hongzhao, Akimoto, Madoka, Darveau, Patrick, MacKinnon, Marc R, Magolan, Jakob, Melacini, Giuseppe

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BSCI-13 DEVELOPMENT OF NOVEL ANTI-BRAIN METASTASIS INHIBITORS von Kieliszek, Agata, Mobilio, Daniel, Bassey-Archibong, Blessing, Johnson, Jarrod, McKenna, Dillon, Venugopal, Chitra, Magolan, Jakob, Singh, Sheila

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A screen for cell envelope stress uncovers an inhibitor of prolipoprotein diacylglyceryl transferase, Lgt, in Escherichiacoli von Rachwalski, Kenneth, Madden, Sean J., Ritchie, Nicole, French, Shawn, Bhando, Timsy, Girgis-Gabardo, Adele, Tu, Megan, Gordzevich, Rodion, Ives, Rowan, Guo, Amelia B.Y., Johnson, Jarrod W., Xu, Yiming, Kapadia, Sharookh B., Magolan, Jakob, Brown, Eric D.

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