Role of tyrosyl-DNA phosphodiesterase (TDP1) in mitochondria von Das, Benu Brata, Dexheimer, Thomas S., Maddali, Kasthuraiah, Pommier, Yves, Nash, Howard

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Resistance to integrase inhibitors von Métifiot, Mathieu, Marchand, Christophe, Maddali, Kasthuraiah, Pommier, Yves

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Probing chelation motifs in HIV integrase inhibitors von Agrawal, Arpita, DeSoto, Jamie, Fullagar, Jessica L, Maddali, Kasthuraiah, Rostami, Shahrzad, Richman, Douglas D, Pommier, Yves, Cohen, Seth M

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HIV-1 Integrase-Targeted Short Peptides Derived from a Viral Protein R Sequence von Zhao, Xue Zhi, Métifiot, Mathieu, Kiselev, Evgeny, Kessl, Jacques J, Maddali, Kasthuraiah, Marchand, Christophe, Kvaratskhelia, Mamuka, Pommier, Yves, Burke, Jr, Terrence R

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Peptidic HIV integrase inhibitors derived from HIV gene products: Structure–activity relationship studies von Suzuki, Shintaro, Maddali, Kasthuraiah, Hashimoto, Chie, Urano, Emiko, Ohashi, Nami, Tanaka, Tomohiro, Ozaki, Taro, Arai, Hiroshi, Tsutsumi, Hiroshi, Narumi, Tetsuo, Nomura, Wataru, Yamamoto, Naoki, Pommier, Yves, Komano, Jun A., Tamamura, Hirokazu

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3-Hydroxypyrimidine-2,4-diones as an Inhibitor Scaffold of HIV Integrase von Tang, Jing, Maddali, Kasthuraiah, Metifiot, Mathieu, Sham, Yuk Y, Vince, Robert, Pommier, Yves, Wang, Zhengqiang

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Elvitegravir overcomes resistance to raltegravir induced by integrase mutation Y143 von METIFIOT, Mathieu, VANDEGRAAFF, Nick, MADDALI, Kasthuraiah, NAUMOVA, Alena, XUEMIN ZHANG, RHODES, David, MARCHAND, Christophe, POMMIER, Yves

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Biochemical and Pharmacological Analyses of HIV-1 Integrase Flexible Loop Mutants Resistant to Raltegravir von Métifiot, Mathieu, Maddali, Kasthuraiah, Naumova, Alena, Zhang, Xuemin, Marchand, Christophe, Pommier, Yves

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Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase von Costi, Roberta, Métifiot, Mathieu, Chung, Suhman, Cuzzucoli Crucitti, Giuliana, Maddali, Kasthuraiah, Pescatori, Luca, Messore, Antonella, Madia, Valentina Noemi, Pupo, Giovanni, Scipione, Luigi, Tortorella, Silvano, Di Leva, Francesco Saverio, Cosconati, Sandro, Marinelli, Luciana, Novellino, Ettore, Le Grice, Stuart F. J, Corona, Angela, Pommier, Yves, Marchand, Christophe, Di Santo, Roberto

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Preparation And Characterization Of Phospholanes And Phospha Sugars As Novel Anti-Cancer Agents von Ito, Satoru, Yamashita, Mitsuji, Niimi, Taishi, Fujie, Michio, Reddy, Valluru Krishna, Totsuka, Hirono, Haritha, Buchammagari, Maddali, Kasthuraiah, Nakamura, Satoki, Asai, Kazuhide, Suyama, Takuya, Yamashita, Junko, Iguchi, Yukiko, Yu, Gang, Oshikawa, Tatsuo

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Activities, Crystal Structures, and Molecular Dynamics of Dihydro-1 H -isoindole Derivatives, Inhibitors of HIV-1 Integrase von Métifiot, Mathieu, Maddali, Kasthuraiah, Johnson, Barry C., Hare, Stephen, Smith, Steven J., Zhao, Xue Zhi, Marchand, Christophe, Burke, Terrence R., Hughes, Stephen H., Cherepanov, Peter, Pommier, Yves

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Cell-Permeable Stapled Peptides Based on HIV‑1 Integrase Inhibitors Derived from HIV‑1 Gene Products von Nomura, Wataru, Aikawa, Haruo, Ohashi, Nami, Urano, Emiko, Métifiot, Mathieu, Fujino, Masayuki, Maddali, Kasthuraiah, Ozaki, Taro, Nozue, Ami, Narumi, Tetsuo, Hashimoto, Chie, Tanaka, Tomohiro, Pommier, Yves, Yamamoto, Naoki, Komano, Jun A, Murakami, Tsutomu, Tamamura, Hirokazu

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6-Benzoyl-3-hydroxypyrimidine-2,4-diones as dual inhibitors of HIV reverse transcriptase and integrase von Tang, Jing, Maddali, Kasthuraiah, Dreis, Christine D., Sham, Yuk Y., Vince, Robert, Pommier, Yves, Wang, Zhengqiang

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Scaffold rearrangement of dihydroxypyrimidine inhibitors of HIV integrase: Docking model revisited von Tang, Jing, Maddali, Kasthuraiah, Pommier, Yves, Sham, Yuk Y., Wang, Zhengqiang

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Diketoacid-genre HIV-1 integrase inhibitors containing enantiomeric arylamide functionality von Zhao, Xue Zhi, Maddali, Kasthuraiah, Marchand, Christophe, Pommier, Yves, Burke, Terrence R.

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N-3 Hydroxylation of Pyrimidine-2,4-diones Yields Dual Inhibitors of HIV Reverse Transcriptase and Integrase von Tang, Jing, Maddali, Kasthuraiah, Dreis, Christine D, Sham, Yuk Y, Vince, Robert, Pommier, Yves, Wang, Zhengqiang

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Studies of HIV-1 Integrase Inhibitory Activity of Wrightia tinctoria von Selvam, Periyasamy, Maddali, Kasthuraiah, Pommier, Yves

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2,3-Dihydro-6,7-dihydroxy-1H-isoindol-1-one-Based HIV-1 Integrase Inhibitors von Zhao, Xue Zhi, Semenova, Elena A, Vu, B. Christie, Maddali, Kasthuraiah, Marchand, Christophe, Hughes, Stephen H, Pommier, Yves, Burke, Terrence R

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Studies of HIV Integrase Inhibitory Activity of Novel Isatine Derivatives von Selvam, Periyasamy, Maddali, Kasthuraiah, Marchand, Christophe, Pommier, Yves

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6,7-Dihydroxy-1-oxoisoindoline-4-sulfonamide-containing HIV-1 integrase inhibitors von Zhao, Xue Zhi, Maddali, Kasthuraiah, Smith, Steven J., Métifiot, Mathieu, Johnson, Barry C., Marchand, Christophe, Hughes, Stephen H., Pommier, Yves, Burke, Terrence R.

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