Cardioprotective Angiotensin-(1–7) Peptide Acts as a Natural-Biased Ligand at the Angiotensin II Type 1 Receptor von Galandrin, Ségolène, Denis, Colette, Boularan, Cédric, Marie, Jacky, M’Kadmi, Céline, Pilette, Claire, Dubroca, Caroline, Nicaise, Yvan, Seguelas, Marie-Hélène, N’Guyen, Du, Banères, Jean-Louis, Pathak, Atul, Sénard, Jean-Michel, Galés, Céline

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Structure and dynamics of G protein-coupled receptor–bound ghrelin reveal the critical role of the octanoyl chain von Ferré, Guillaume, Louet, Maxime, Saurel, Oliver, Delort, Bartholomé, Czaplicki, Georges, M’Kadmi, Céline, Damian, Marjorie, Renault, Pedro, Cantel, Sonia, Gavara, Laurent, Demange, Pascal, Marie, Jacky, Fehrentz, Jean-Alain, Floquet, Nicolas, Milon, Alain, Banères, Jean-Louis

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Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex von Damian, Marjorie, Mary, Sophie, Maingot, Mathieu, M’Kadmi, Céline, Gagne, Didier, Leyris, Jean-Philippe, Denoyelle, Séverine, Gaibelet, Gérald, Gavara, Laurent, de Souza Costa, Mauricio Garcia, Perahia, David, Trinquet, Eric, Mouillac, Bernard, Galandrin, Ségolène, Galès, Céline, Fehrentz, Jean-Alain, Floquet, Nicolas, Martinez, Jean, Marie, Jacky, Banères, Jean-Louis

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Concerted conformational dynamics and water movements in the ghrelin G protein-coupled receptor von Louet, Maxime, Casiraghi, Marina, Damian, Marjorie, Costa, Mauricio G. S., Renault, Pedro, Gomes, Antoniel A. S., Batista, Paulo R., M'Kadmi, Celine, Mary, Sophie, Cantel, Sonia, Denoyelle, Severine, Salah, Khoubaib Ben Haj, Perahia, David, Bisch, Paulo M., Fehrentz, Jean-Alain, Catoire, Laurent J., Floquet, Nicolas, Baneres, Jean-Louis

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Development of Nonpeptidic Inverse Agonists of the Ghrelin Receptor (GHSR) Based on the 1,2,4-Triazole Scaffold von Haj Salah, Khoubaib Ben, Maingot, Mathieu, Blayo, Anne-Laure, M’Kadmi, Céline, Damian, Marjorie, Mary, Sophie, Cantel, Sonia, Neasta, Jérémie, Oiry, Catherine, Péraldi-Roux, Sylvie, Fernandez, Gimena, Romero, Guadalupe García, Perello, Mario, Marie, Jacky, Banères, Jean-Louis, Fehrentz, Jean-Alain, Denoyelle, Séverine

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Evidence Supporting a Role for Constitutive Ghrelin Receptor Signaling in Fasting-Induced Hyperphagia in Male Mice von Fernandez, Gimena, Cabral, Agustina, Andreoli, María F, Labarthe, Alexandra, M'Kadmi, Céline, Ramos, Jorge G, Marie, Jacky, Fehrentz, Jean-Alain, Epelbaum, Jacques, Tolle, Virginie, Perello, Mario

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The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist von Moulin, Aline, Brunel, Luc, Boeglin, Damien, Demange, Luc, Ryan, Johanne, M’Kadmi, Céline, Denoyelle, Séverine, Martinez, Jean, Fehrentz, Jean-Alain

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Development of a novel fluorescent ligand of growth hormone secretagogue receptor based on the N-Terminal Leap2 region von Barrile, Franco, M'Kadmi, Céline, De Francesco, Pablo N., Cabral, Agustina, García Romero, Guadalupe, Mustafá, Emilio R., Cantel, Sonia, Damian, Marjorie, Mary, Sophie, Denoyelle, Séverine, Banères, Jean-Louis, Marie, Jacky, Raingo, Jesica, Fehrentz, Jean-Alain, Perelló, Mario

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Design and characterization of a triazole-based growth hormone secretagogue receptor modulator inhibiting the glucoregulatory and feeding actions of ghrelin von Péraldi-Roux, Sylvie, Bayle, Morgane, M'Kadmi, Céline, Damian, Marjorie, Vaillé, Justine, Fernandez, Gimena, Cornejo, Maria Paula, Marie, Jacky, Banères, Jean-Louis, Ben Haj Salah, Khoubaib, Fehrentz, Jean-Alain, Cantel, Sonia, Perello, Mario, Denoyelle, Séverine, Oiry, Catherine, Neasta, Jérémie

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N‑Terminal Liver-Expressed Antimicrobial Peptide 2 (LEAP2) Region Exhibits Inverse Agonist Activity toward the Ghrelin Receptor von M’Kadmi, Céline, Cabral, Agustina, Barrile, Franco, Giribaldi, Julien, Cantel, Sonia, Damian, Marjorie, Mary, Sophie, Denoyelle, Séverine, Dutertre, Sébastien, Péraldi-Roux, Sylvie, Neasta, Jérémie, Oiry, Catherine, Banères, Jean-Louis, Marie, Jacky, Perello, Mario, Fehrentz, Jean-Alain

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Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a von Leyris, Jean-Philippe, Roux, Thomas, Trinquet, Eric, Verdié, Pascal, Fehrentz, Jean-Alain, Oueslati, Nadia, Douzon, Stéphanie, Bourrier, Emmanuel, Lamarque, Laurent, Gagne, Didier, Galleyrand, Jean-Claude, M’kadmi, Céline, Martinez, Jean, Mary, Sophie, Banères, Jean-Louis, Marie, Jacky

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Allosteric modulation of ghrelin receptor signaling by lipids von Damian, Marjorie, Louet, Maxime, Gomes, Antoniel Augusto Severo, M’Kadmi, Céline, Denoyelle, Séverine, Cantel, Sonia, Mary, Sophie, Bisch, Paulo M., Fehrentz, Jean-Alain, Catoire, Laurent J., Floquet, Nicolas, Banères, Jean-Louis

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Detergent-free Isolation of Functional G Protein-Coupled Receptors into Nanometric Lipid Particles von Logez, Christel, Damian, Marjorie, Legros, Céline, Dupré, Clémence, Guéry, Mélody, Mary, Sophie, Wagner, Renaud, M’Kadmi, Céline, Nosjean, Olivier, Fould, Benjamin, Marie, Jacky, Fehrentz, Jean-Alain, Martinez, Jean, Ferry, Gilles, Boutin, Jean A, Banères, Jean-Louis

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Quantitative MALDI-MS Binding Assays: An Alternative to Radiolabeling von Rossato, Maxime, Miralles, Guillaume, M'Kadmi, Céline, Maingot, Mathieu, Amblard, Muriel, Mouillac, Bernard, Gagne, Didier, Martinez, Jean, Subra, Gilles, Enjalbal, Christine, Cantel, Sonia

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Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling von M'Kadmi, Céline, Leyris, Jean-Philippe, Onfroy, Lauriane, Galés, Céline, Saulière, Aude, Gagne, Didier, Damian, Marjorie, Mary, Sophie, Maingot, Mathieu, Denoyelle, Séverine, Verdié, Pascal, Fehrentz, Jean-Alain, Martinez, Jean, Banères, Jean-Louis, Marie, Jacky

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New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center von Maingot, Mathieu, Blayo, Anne-Laure, Denoyelle, Séverine, M’Kadmi, Céline, Damian, Marjorie, Mary, Sophie, Gagne, Didier, Sanchez, Pierre, Aicher, Babette, Schmidt, Peter, Müller, Gilbert, Teifel, Michael, Günther, Eckhard, Marie, Jacky, Banères, Jean-Louis, Martinez, Jean, Fehrentz, Jean-Alain

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GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation von Damian, Marjorie, Pons, Véronique, Renault, Pedro, M’Kadmi, Céline, Delort, Bartholomé, Hartmann, Lucie, Kaya, Ali I., Louet, Maxime, Gagne, Didier, Salah, Khoubaib Ben Haj, Denoyelle, Séverine, Ferry, Gilles, Boutin, Jean A., Wagner, Renaud, Fehrentz, Jean-Alain, Martinez, Jean, Marie, Jacky, Floquet, Nicolas, Galès, Céline, Mary, Sophie, Hamm, Heidi E., Banères, Jean-Louis

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The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release von Neasta, Jérémie, Valmalle, Charlène, Coyne, Anne‐Claire, Carnazzi, Eric, Subra, Gilles, Galleyrand, Jean‐Claude, Gagne, Didier, M'Kadmi, Céline, Bernad, Nicole, Bergé, Gilbert, Cantel, Sonia, Marin, Philippe, Marie, Jacky, Banères, Jean‐Louis, Kemel, Marie‐Lou, Daugé, Valérie, Puget, Karine, Martinez, Jean

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α-Tocopherol and α-tocopheryl phosphate interact with the cannabinoid system in the rodent hippocampus von Crouzin, Nadine, de Jesus Ferreira, Marie-Céleste, Cohen-Solal, Catherine, M'Kadmi, Céline, Bernad, Nicole, Martinez, Jean, Barbanel, Gérard, Vignes, Michel, Guiramand, Janique

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Involvement of tryptophan W276 and of two surrounding amino acid residues in the high constitutive activity of the ghrelin receptor GHS-R1a von Gozé, Catherine, Bergé, Gilbert, M'Kadmi, Céline, Floquet, Nicolas, Gagne, Didier, Galleyrand, Jean-Claude, Fehrentz, Jean-Alain, Martinez, Jean

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