Expression, Crystallization, and Three-dimensional Structure of the Catalytic Domain of Human Plasma Kallikrein von Tang, Jie, Yu, Christine Luong, Williams, Steven R., Springman, Eric, Jeffery, Douglas, Sprengeler, Paul A., Estevez, Alberto, Sampang, Jun, Shrader, William, Spencer, Jeff, Young, Wendy, McGrath, Mary, Katz, Bradley A.

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Development of Serine Protease Inhibitors Displaying a Multicentered Short (<2.3 Å) Hydrogen Bond Binding Mode:  Inhibitors of Urokinase-Type Plasminogen Activator and Factor Xa von Verner, Erik, Katz, Bradley A, Spencer, Jeffrey R, Allen, Darin, Hataye, Jason, Hruzewicz, Witold, Hui, Hon C, Kolesnikov, Aleksandr, Li, Yong, Luong, Christine, Martelli, Arnold, Radika, Kesavan, Rai, Roopa, She, Miles, Shrader, William, Sprengeler, Paul A, Trapp, Sean, Wang, Jing, Young, Wendy B, Mackman, Richard L

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The Structure of the Extracellular Region of Human Hepsin Reveals a Serine Protease Domain and a Novel Scavenger Receptor Cysteine-Rich (SRCR) Domain von Somoza, John R, Ho, Joseph D, Luong, Christine, Ghate, Manjiri, Sprengeler, Paul A, Mortara, Kyle, Shrader, William D, Sperandio, David, Chan, Hedy, McGrath, Mary E, Katz, Bradley A

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Design of potent selective zinc-mediated serine protease inhibitors von Katz, Bradley A., Clark, James M., Finer-Moore, Janet S., Jenkins, Thomas E., Johnson, Charles R., Ross, Michael J., Luong, Christine, Moore, William R., Stroud, Robert M.

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Flexibility of the NSAID binding site in the structure of human cyclooxygenase-2 von Luong, Christine, Miller, Aaron, Barnett, Jim, Chow, Joan, Ramesha, Chakk, Browner, Michelle F.

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Structural Snapshots of Human HDAC8 Provide Insights into the Class I Histone Deacetylases von Somoza, John R, Skene, Robert J, Katz, Bradley A, Mol, Clifford, Ho, Joseph D, Jennings, Andy J, Luong, Christine, Arvai, Andrew, Buggy, Joseph J, Chi, Ellen, Tang, Jie, Sang, Bi-Ching, Verner, Erik, Wynands, Robert, Leahy, Ellen M, Dougan, Douglas R, Snell, Gyorgy, Navre, Marc, Knuth, Mark W, Swanson, Ronald V, McRee, Duncan E, Tari, Leslie W

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Partial Activation of Muscle Phosphorylase by Replacement of Serine 14 with Acidic Residues at the Site of Regulatory Phosphorylation von Buchbinder, Jenny L, Luong, Christine B. H, Browner, Michelle F, Fletterick, Robert J

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Exploiting Subsite S1 of Trypsin-Like Serine Proteases for Selectivity:  Potent and Selective Inhibitors of Urokinase-Type Plasminogen Activator von Mackman, Richard L, Katz, Bradley A, Breitenbucher, J. Guy, Hui, Hon C, Verner, Erik, Luong, Christine, Liu, Liang, Sprengeler, Paul A

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A novel serine protease inhibition motif involving a multi-centered short hydrogen bonding network at the active site von Katz, Bradley A, Elrod, Kyle, Luong, Christine, Rice, Mark J, Mackman, Richard L, Sprengeler, Paul A, Spencer, Jeffrey, Hataye, Jason, Janc, James, Link, John, Litvak, Joane, Rai, Roopa, Rice, Ken, Sideris, Steve, Verner, Erik, Young, Wendy

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Dissecting and Designing Inhibitor Selectivity Determinants at the S1 Site Using an Artificial Ala190 Protease (Ala190 uPA) von Katz, Bradley A., Luong, Christine, Ho, Joseph D., Somoza, John R., Gjerstad, Erik, Tang, Jie, Williams, Steven R., Verner, Erik, Mackman, Richard L., Young, Wendy B., Sprengeler, Paul A., Chan, Hedy, Mortara, Kyle, Janc, James W., McGrath, Mary E.

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Recruiting Zn2+to Mediate Potent, Specific Inhibition of Serine Proteases von Katz, Bradley A., Luong, Christine

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Crystal structures of MMP-1 and -13 reveal the structural basis for selectivity of collagenase inhibitors von Lovejoy, Brett, Welch, Anthony R., Carr, Steven, Luong, Christine, Broka, Chris, Hendricks, R. Than, Campbell, Jeffery A., Walker, Keith A.M., Martin, Robert, Van Wart, Harold, Browner, Michelle F.

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Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-directed Serine Protease Inhibitors von Katz, Bradley A., Elrod, Kyle, Verner, Erik, Mackman, Richard L., Luong, Christine, Shrader, William D., Sendzik, Martin, Spencer, Jeffrey R., Sprengeler, Paul A., Kolesnikov, Aleks, Tai, Vincent W.-F., Hui, Hon C., Guy Breitenbucher, J., Allen, Darin, Janc, James W.

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Contribution of Multicentered Short Hydrogen Bond Arrays to Potency of Active Site-Directed Serine Protease Inhibitors von Katz, Bradley A, Spencer, Jeffrey R, Elrod, Kyle, Luong, Christine, Mackman, Richard L, Rice, Mark, Sprengeler, Paul A, Allen, Darin, Janc, James

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Maize photosystem I. Identification of the subunit which binds plastocyanin von Wynn, R. Max, Christine Luong, Malkin, Richard

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2-(2-Hydroxy-3-alkoxyphenyl)-1H-benzimidazole-5-carboxamidine derivatives as potent and selective urokinase-type plasminogen activator inhibitors von MACKMAN, Richard L, HUI, Hon C, SPRENGELER, Paul A, TARIO, James, VERNER, Erik, JING WANG, BREITENBUCHER, J. Guy, KATZ, Bradley A, LUONG, Christine, MARTELLI, Arnold, MCGEE, Danny, RADIKA, Kesavan, SENDZIK, Martin, SPENCER, Jeffrey R

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4-Aminoarylguanidine and 4-aminobenzamidine derivatives as potent and selective urokinase-type plasminogen activator inhibitors von Spencer, Jeffrey R, McGee, Danny, Allen, Darin, Katz, Bradley A, Luong, Christine, Sendzik, Martin, Squires, Neil, Mackman, Richard L

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Development of potent and selective factor Xa inhibitors von RAI, Roopa, KOLESNIKOV, Aleksandr, ALLEN, Darin, CHEN, Xi, KATZ, Bradley A, LUONG, Christine, ELROD, Kyle, CREGAR, Lynne, YONG LI, YOUNG, Wendy B, LEAHY, Ellen, SPRENGELER, Paul A, VERNER, Erik, SHRADER, William D, BURGESS-HENRY, Jana, SANGALANG, Joan C

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A novel serine protease inhibition motif involving a multi-centered short hydrogen bonding network at the active site11Edited by D. Rees von Katz, Bradley A, Elrod, Kyle, Luong, Christine, Rice, Mark J, Mackman, Richard L, Sprengeler, Paul A, Spencer, Jeffrey, Hataye, Jason, Janc, James, Link, John, Litvak, Joane, Rai, Roopa, Rice, Ken, Sideris, Steve, Verner, Erik, Young, Wendy

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2-(2-Hydroxy-3-alkoxyphenyl)-1 H-benzimidazole-5-carboxamidine derivatives as potent and selective urokinase-type plasminogen activator inhibitors von Mackman, Richard L., Hui, Hon C., Breitenbucher, J.Guy, Katz, Bradley A., Luong, Christine, Martelli, Arnold, McGee, Danny, Radika, Kesavan, Sendzik, Martin, Spencer, Jeffrey R., Sprengeler, Paul A., Tario, James, Verner, Erik, Wang, Jing

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