Orally Absorbed Cyclic Peptides von Nielsen, Daniel S, Shepherd, Nicholas E, Xu, Weijun, Lucke, Andrew J, Stoermer, Martin J, Fairlie, David P

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Improving on Nature: Making a Cyclic Heptapeptide Orally Bioavailable von Nielsen, Daniel S., Hoang, Huy N., Lohman, Rink-Jan, Hill, Timothy A., Lucke, Andrew J., Craik, David J., Edmonds, David J., Griffith, David A., Rotter, Charles J., Ruggeri, Roger B., Price, David A., Liras, Spiros, Fairlie, David P.

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Comparing sixteen scoring functions for predicting biological activities of ligands for protein targets von Xu, Weijun, Lucke, Andrew J., Fairlie, David P.

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Flexibility versus Rigidity for Orally Bioavailable Cyclic Hexapeptides von Nielsen, Daniel S., Lohman, Rink-Jan, Hoang, Huy N., Hill, Timothy A., Jones, Alun, Lucke, Andrew J., Fairlie, David P.

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Achiral Derivatives of Hydroxamate AR-42 Potently Inhibit Class I HDAC Enzymes and Cancer Cell Proliferation von Tng, Jiahui, Lim, Junxian, Wu, Kai-Chen, Lucke, Andrew J., Xu, Weijun, Reid, Robert C., Fairlie, David P.

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HDAC7 Inhibition by Phenacetyl and Phenylbenzoyl Hydroxamates von Mak, Jeffrey Y. W, Wu, Kai-Chen, Gupta, Praveer K, Barbero, Sheila, McLaughlin, Maddison G, Lucke, Andrew J, Tng, Jiahui, Lim, Junxian, Loh, Zhixuan, Sweet, Matthew J, Reid, Robert C, Liu, Ligong, Fairlie, David P

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Antimalarial Activity of the Anticancer Histone Deacetylase Inhibitor SB939 von Sumanadasa, Subathdrage D M, Goodman, Christopher D, Lucke, Andrew J, Skinner-Adams, Tina, Sahama, Ishani, Haque, Ashraful, Do, Tram Anh, McFadden, Geoffrey I, Fairlie, David P, Andrews, Katherine T

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Temporal perturbation of histone deacetylase activity reveals a requirement for HDAC1–3 in mesendoderm cell differentiation von Sinniah, Enakshi, Wu, Zhixuan, Shen, Sophie, Naval-Sanchez, Marina, Chen, Xiaoli, Lim, Junxian, Helfer, Abbigail, Iyer, Abishek, Tng, Jiahui, Lucke, Andrew J., Reid, Robert C., Redd, Meredith A., Nefzger, Christian M., Fairlie, David P., Palpant, Nathan J.

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Identification of brain metastasis genes and therapeutic evaluation of histone deacetylase inhibitors in a clinically relevant model of breast cancer brain metastasis von Kim, Soo-Hyun, Redvers, Richard P, Chi, Lap Hing, Ling, Xiawei, Lucke, Andrew J, Reid, Robert C, Fairlie, David P, Martin, Ana Carolina Baptista Moreno, Anderson, Robin L, Denoyer, Delphine, Pouliot, Normand

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Histone deacetylase inhibitor AR-42 and achiral analogues kill malaria parasites in vitro and in mice von Chua, Ming Jang, Tng, Jiahui, Hesping, Eva, Fisher, Gillian M., Goodman, Christopher D., Skinner-Adams, Tina, Do, Darren, Lucke, Andrew J., Reid, Robert C., Fairlie, David P., Andrews, Katherine T.

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Three Homology Models of PAR2 Derived from Different Templates: Application to Antagonist Discovery von Perry, Samuel R, Xu, Weijun, Wirija, Anna, Lim, Junxian, Yau, Mei-Kwan, Stoermer, Martin J, Lucke, Andrew J, Fairlie, David P

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A Nucleotide Analog Prevents Colitis-Associated Cancer via Beta-Catenin Independently of Inflammation and Autophagy von Sheng, Yong Hua, Giri, Rabina, Davies, Julie, Schreiber, Veronika, Alabbas, Saleh, Movva, Ramya, He, Yaowu, Wu, Andy, Hooper, John, McWhinney, Brett, Oancea, Iulia, Kijanka, Gregor, Hasnain, Sumaira, Lucke, Andrew J., Fairlie, David P., McGuckin, Michael A., Florin, Timothy H., Begun, Jakob

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Insecticidal activities of histone deacetylase inhibitors against a dipteran parasite of sheep, Lucilia cuprina von Bagnall, Neil H., Hines, Barney M., Lucke, Andrew J., Gupta, Praveer K., Reid, Robert C., Fairlie, David P., Kotze, Andrew C.

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Cyclic Penta- and Hexaleucine Peptides without N‑Methylation Are Orally Absorbed von Hill, Timothy A, Lohman, Rink-Jan, Hoang, Huy N, Nielsen, Daniel S, Scully, Conor C. G, Kok, W. Mei, Liu, Ligong, Lucke, Andrew J, Stoermer, Martin J, Schroeder, Christina I, Chaousis, Stephanie, Colless, Barbara, Bernhardt, Paul V, Edmonds, David J, Griffith, David A, Rotter, Charles J, Ruggeri, Roger B, Price, David A, Liras, Spiros, Craik, David J, Fairlie, David P

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Antimalarial histone deacetylase inhibitors containing cinnamate or NSAID components von Wheatley, Nicole C., Andrews, Katherine T., Tran, Truc L., Lucke, Andrew J., Reid, Robert C., Fairlie, David P.

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Design, Synthesis, Potency, and Cytoselectivity of Anticancer Agents Derived by Parallel Synthesis from α-Aminosuberic Acid von Kahnberg, Pia, Lucke, Andrew J, Glenn, Matthew P, Boyle, Glen M, Tyndall, Joel D. A, Parsons, Peter G, Fairlie, David P

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Inhibitors selective for HDAC6 in enzymes and cells von Gupta, Praveer K., Reid, Robert C., Liu, Ligong, Lucke, Andrew J., Broomfield, Steve A., Andrews, Melanie R., Sweet, Matthew J., Fairlie, David P.

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Structural Mimicry of Two Cytochrome b562 Interhelical Loops Using Macrocycles Constrained by Oxazoles and Thiazoles von SINGH, Yogendra, STOERMER, Martin J., LUCKE, Andrew J., GUTHRIE, Tom, FAIRLIE, David P.

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Electrophilic Cleavage of Cyclopropylmethystannanes:  An Experimental Comparison of σ−σ and σ−π Conjugation von Lucke, Andrew J, Young, David J

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Improving on Nature: Making a Cyclic Heptapeptide Orally Bioavailable von Nielsen, Daniel S., Hoang, Huy N., Lohman, Rink-Jan, Hill, Timothy A., Lucke, Andrew J., Craik, David J., Edmonds, David J., Griffith, David A., Rotter, Charles J., Ruggeri, Roger B., Price, David A., Liras, Spiros, Fairlie, David P.

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