Use of the Nitrile Oxide Cycloaddition (NOC) Reaction for Molecular Probe Generation: A New Class of Enzyme Selective Histone Deacetylase Inhibitors (HDACIs) Showing Picomolar Acti... von Kozikowski, Alan P, Tapadar, Subhasish, Luchini, Doris N, Kim, Ki Hwan, Billadeau, Daniel D

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Asef2 Functions as a Cdc42 Exchange Factor and Is Stimulated by the Release of an Autoinhibitory Module from a Concealed C-Terminal Activation Element von Hamann, Michael J., Lubking, Casey M., Luchini, Doris N., Billadeau, Daniel D.

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From a Natural Product Lead to the Identification of Potent and Selective Benzofuran-3-yl-(indol-3-yl)maleimides as Glycogen Synthase Kinase 3β Inhibitors That Suppress Proliferati... von Gaisina, Irina N, Gallier, Franck, Ougolkov, Andrei V, Kim, Ki H, Kurome, Toru, Guo, Songpo, Holzle, Denise, Luchini, Doris N, Blond, Sylvie Y, Billadeau, Daniel D, Kozikowski, Alan P

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Novel acridine-based compounds that exhibit an anti-pancreatic cancer activity are catalytic inhibitors of human topoisomerase II von Oppegard, Lisa M., Ougolkov, Andrei V., Luchini, Doris N., Schoon, Renee A., Goodell, John R., Kaur, Harneet, Billadeau, Daniel D., Ferguson, David M., Hiasa, Hiroshi

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Isoxazole moiety in the linker region of HDAC inhibitors adjacent to the Zn-chelating group: Effects on HDAC biology and antiproliferative activity von Tapadar, Subhasish, He, Rong, Luchini, Doris N., Billadeau, Daniel D., Kozikowski, Alan P.

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Molecular and Cellular Pharmacology: Novel acridine-based compounds that exhibit an anti-pancreatic cancer activity are catalytic inhibitors of human topoisomerase II von Oppegard, Lisa M, Ougolkov, Andrei V, Luchini, Doris N, Schoon, Renee A, Goodell, John R, Kaur, Harneet, Billadeau, Daniel D, Ferguson, David M, Hiasa, Hiroshi

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From a natural product lead to the identification of potent and selective benzofuran-3-yl-(indol-3-yl)maleimides as glycogen synthase kinase 3beta inhibitors that suppress prolifer... von Gaisina, Irina N, Gallier, Franck, Ougolkov, Andrei V, Kim, Ki H, Kurome, Toru, Guo, Songpo, Holzle, Denise, Luchini, Doris N, Blond, Sylvie Y, Billadeau, Daniel D, Kozikowski, Alan P

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