Prolonged and tunable residence time using reversible covalent kinase inhibitors von Bradshaw, J Michael, McFarland, Jesse M, Paavilainen, Ville O, Bisconte, Angelina, Tam, Danny, Phan, Vernon T, Romanov, Sergei, Finkle, David, Shu, Jin, Patel, Vaishali, Ton, Tony, Li, Xiaoyan, Loughhead, David G, Nunn, Philip A, Karr, Dane E, Gerritsen, Mary E, Funk, Jens Oliver, Owens, Timothy D, Verner, Erik, Brameld, Ken A, Hill, Ronald J, Goldstein, David M, Taunton, Jack

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Discovery of the Irreversible Covalent FGFR Inhibitor 8‑(3-(4-Acryloyl­piperazin-1-yl)propyl)-6-(2,6-dichloro-3,5-dimethoxyphenyl)-2-(methylamino)­pyrido[2,3‑d]­pyrimidin-7(8H)‑one... von Brameld, Ken A, Owens, Timothy D, Verner, Erik, Venetsanakos, Eleni, Bradshaw, J. Michael, Phan, Vernon T, Tam, Danny, Leung, Kwan, Shu, Jin, LaStant, Jacob, Loughhead, David G, Ton, Tony, Karr, Dane E, Gerritsen, Mary E, Goldstein, David M, Funk, Jens Oliver

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Novel hexahydropyrrolo[3,4- c]pyrrole CCR5 antagonists von Rotstein, David M., Melville, Chris R., Padilla, Fernando, Cournoyer, Dick, Lee, Eun K., Lemoine, Remy, Petersen, Ann C., Setti, Lina Q., Wanner, Jutta, Chen, Lijing, Filonova, Lubov, Loughhead, David G., Manka, Jason, Lin, Xiao-Fa, Gleason, Shelley, Sankuratri, Surya, Ji, Changhua, deRosier, Andre, Dioszegi, Marianna, Heilek, Gabrielle, Jekle, Andreas, Berry, Pamela, Mau, Cheng-I, Weller, Paul

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Asymmetric Synthesis and Stereochemical Assignment of RS-97613, a Potent Immunosuppressive and Antiinflammatory Agent von Smith, David B, Waltos, Ann Marie, Loughhead, David G, Weikert, Robert J, Morgans, David J, Rohloff, John C, Link, John O, Zhu, Rong-rong

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Structures and Total Synthesis of 2-Aminoimidazoles from a Notodoris Nudibranch von Alvi, K. A, Crews, Phillip, Loughhead, David G

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Synthesis of des-N-methylacronycine and acronycine von Loughhead, David G

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Synthesis of Mexiletine Stereoisomers and Related Compounds via SNAr Nucleophilic Substitution of a Cr(CO)3-Complexed Aromatic Fluoride von Loughhead, David G, Flippin, Lee A, Weikert, Robert J

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2,2-Dimethylcyclopropyl-benzamides: Novel positive allosteric modulators of α7 nAChRs von Maag, Hans, Bois, Daisy Joe Du, Loughhead, David G., Manka, Jason, Misner, Dinah, Sahdeo, Sunil, Smith, David B.

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Synthesis and anthelmintic activity of 3'-benzoylurea derivatives of 6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole von Weikert, Robert J, Bingham, Stanford, Emanuel, Mark A, Fraser-Smith, Elizabeth B, Loughhead, David G, Nelson, Peter H, Poulton, Anthony L

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Preparation and acid-catalyzed rearrangement of a carbon-17 isopropylidene and a carbon-17 isopropenyl sterol von Loughhead, David G

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Synthesis of Mexiletine Stereoisomers and Related Compounds via S(N)Ar Nucleophilic Substitution of a Cr(CO)(3)-Complexed Aromatic Fluoride von Loughhead, David G., Flippin, Lee A., Weikert, Robert J.

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Structure−Activity Relationships for Inhibition of Inosine Monophosphate Dehydrogenase by Nuclear Variants of Mycophenolic Acid von Nelson, Peter H, Carr, Stephen F, Devens, Bruce H, Eugui, Elsie M, Franco, Fidencio, Gonzalez, Carlos, Hawley, Ronald C, Loughhead, David G, Milan, David J, Papp, Eva, Patterson, John W, Rouhafza, Sussan, Sjogren, Eric B, Smith, David B, Stephenson, Rebecca A, Talamas, Francisco X, Waltos, Ann-Marie, Weikert, Robert J, Wu, John C

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Synthesis of Mexiletine Stereoisomers and Related Compounds via S N Ar Nucleophilic Substitution of a Cr(CO) 3 -Complexed Aromatic Fluoride von Loughhead, David G., Flippin, Lee A., Weikert, Robert J.

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The Florisil ® catalyzed [1,3]-sigmatropic shift of allyl phenyl ethers — An entryway into novel mycophenolic acid analogues von Talamás, Francisco X., Smith, David B., Cervantes, Alicia, Franco, Fidencio, Cutler, Serena T., Loughhead, David G., Morgans, David J., Weikert, Robert J.

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Unusual reductions induced by formic acid von Loughhead, David G.

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Preparation and acid-catalyzed rearrangement of C-17 isopropylidene and a C-17 isopropenyl sterol von LOUGHHEAD, D. G

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Ring fused pyrazole derivatives as CRF antagonists von LOUGHHEAD DAVID G, O'YANG COUNDE

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Indazole derivatives as CRF antagonists von LOUGHHEAD DAVID G, O'YANG COUNDE, COURNOYER RICHARD L

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Heterocyclic GABAA subtype selective receptor modulators von LOUGHHEAD DAVID G.,NOVAKOVIC SANJA,O'YANG COUNDE,PUTMAN DAVID G.,SOTH MICHAEL

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Heterocyclic GABAA subtype selective receptor modulators von LOUGHHEAD DAVID G, O'YANG COUNDE, PUTMAN DAVID G, SOTH MICHAEL, NOVAKOVIC SANJA

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