Generation and Cross-Coupling of Organozinc Reagents in Flow von Herath, Ananda, Molteni, Valentina, Pan, Shifeng, Loren, Jon

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One-Pot Electrochemical Nickel-Catalyzed Decarboxylative Sp2–Sp3 Cross-Coupling von Koyanagi, Takaoki, Herath, Ananda, Chong, Ashley, Ratnikov, Maxim, Valiere, Andrew, Chang, Jim, Molteni, Valentina, Loren, Jon

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Synthesis of a D3-symmetric "trefoil" knotted cyclophane von Arias, Karla I, Zysman-Colman, Eli, Loren, Jon C, Linden, Anthony, Siegel, Jay S

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Optimization of Platelet-Derived Growth Factor Receptor (PDGFR) Inhibitors for Duration of Action, as an Inhaled Therapy for Lung Remodeling in Pulmonary Arterial Hypertension von Shaw, Duncan E, Baig, Ferheen, Bruce, Ian, Chamoin, Sylvie, Collingwood, Stephen P, Cross, Sarah, Dayal, Satish, Drückes, Peter, Furet, Pascal, Furminger, Vikki, Haggart, Deborah, Hussey, Martin, Konstantinova, Irena, Loren, Jon C, Molteni, Valentina, Roberts, Sonia, Reilly, John, Saunders, Alex M, Stringer, Rowan, Sviridenko, Lilya, Thomas, Matthew, Thomson, Christopher G, Tomlins, Christine, Wen, Ben, Yeh, Vince, Pearce, Andrew C

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Synthesis of achiral and racemic catenanes based on terpyridine and a directionalized terpyridine mimic, pyridyl-phenanthroline von Loren, Jon C, Gantzel, Peter, Linden, Anthony, Siegel, Jay S

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Synthetic Approaches to a Molecular Borromean Link: Two-Ring Threading with Polypyridine Templates von Loren, Jon C., Yoshizawa, Michito, Haldimann, Richard F., Linden, Anthony, Siegel, Jay S.

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Synthesis and Fluorescence Properties of Manisyl-Substituted Terpyridine, Bipyridine, and Phenanthroline von Loren, Jon C., Siegel, Jay S.

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One-Pot Electrochemical Nickel-Catalyzed Decarboxylative Sp 2 -Sp 3 Cross-Coupling von Koyanagi, Takaoki, Herath, Ananda, Chong, Ashley, Ratnikov, Maxim, Valiere, Andrew, Chang, Jim, Molteni, Valentina, Loren, Jon

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Selective DYRK1A Inhibitor for the Treatment of Type 1 Diabetes: Discovery of 6‑Azaindole Derivative GNF2133 von Liu, Yahu A, Jin, Qihui, Zou, Yefen, Ding, Qiang, Yan, Shanshan, Wang, Zhicheng, Hao, Xueshi, Nguyen, Bao, Zhang, Xiaoyue, Pan, Jianfeng, Mo, Tingting, Jacobsen, Kate, Lam, Thanh, Wu, Tom Y.-H, Petrassi, H. Michael, Bursulaya, Badry, DiDonato, Michael, Gordon, W. Perry, Liu, Bo, Baaten, Janine, Hill, Robert, Nguyen-Tran, Vân, Qiu, Minhua, Zhang, You-Qing, Kamireddy, Anwesh, Espinola, Sheryll, Deaton, Lisa, Ha, Sukwon, Harb, George, Jia, Yong, Li, Jing, Shen, Weijun, Schumacher, Andrew M, Colman, Karyn, Glynne, Richard, Pan, Shifeng, McNamara, Peter, Laffitte, Bryan, Meeusen, Shelly, Molteni, Valentina, Loren, Jon

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Tuning a Protein‐Labeling Reaction to Achieve Highly Site Selective Lysine Conjugation von Pham, Grace H., Ou, Weijia, Bursulaya, Badry, DiDonato, Michael, Herath, Ananda, Jin, Yunho, Hao, Xueshi, Loren, Jon, Spraggon, Glen, Brock, Ansgar, Uno, Tetsuo, Geierstanger, Bernhard H., Cellitti, Susan E.

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TrkB inhibition by GNF-4256 slows growth and enhances chemotherapeutic efficacy in neuroblastoma xenografts von Croucher, Jamie L., Iyer, Radhika, Li, Nanxin, Molteni, Valentina, Loren, Jon, Gordon, W. Perry, Tuntland, Tove, Liu, Bo, Brodeur, Garrett M.

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A Dual Inhibitor of DYRK1A and GSK3β for β‐Cell Proliferation: Aminopyrazine Derivative GNF4877 von Liu, Yahu A., Jin, Qihui, Ding, Qiang, Hao, Xueshi, Mo, Tingting, Yan, Shanshan, Zou, Yefen, Huang, Zhihong, Zhang, Xiaoyue, Gao, Wenqi, Wu, Tom Y.‐H., Li, Chun, Bursalaya, Badry, Di Donato, Michael, Zhang, You‐Qing, Deaton, Lisa, Shen, Weijun, Taylor, Brandon, Kamireddy, Anwesh, Harb, George, Li, Jing, Jia, Yong, Schumacher, Andrew M., Laffitte, Bryan, Glynne, Richard, Pan, Shifeng, McNamara, Peter, Molteni, Valentina, Loren, Jon

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NH-1,2,3-Triazoles from Azidomethyl Pivalate and Carbamates: Base-Labile N-Protecting Groups von Loren, Jon C., Krasiński, Antoni, Fokin, Valery V., Sharpless, K. Barry

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Discovery of GNF-5837, a Selective TRK Inhibitor with Efficacy in Rodent Cancer Tumor Models von Albaugh, Pam, Fan, Yi, Mi, Yuan, Sun, Fangxian, Adrian, Francisco, Li, Nanxin, Jia, Yong, Sarkisova, Yelena, Kreusch, Andreas, Hood, Tami, Lu, Min, Liu, Guoxun, Huang, Shenlin, Liu, Zuosheng, Loren, Jon, Tuntland, Tove, Karanewsky, Donald S, Seidel, H. Martin, Molteni, Valentina

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(R)‑2-Phenylpyrrolidine Substituted Imidazopyridazines: A New Class of Potent and Selective Pan-TRK Inhibitors von Choi, Ha-Soon, Rucker, Paul V, Wang, Zhicheng, Fan, Yi, Albaugh, Pamela, Chopiuk, Greg, Gessier, Francois, Sun, Fangxian, Adrian, Francisco, Liu, Guoxun, Hood, Tami, Li, Nanxin, Jia, Yong, Che, Jianwei, McCormack, Susan, Li, Allen, Li, Jie, Steffy, Auzon, Culazzo, AnneMarie, Tompkins, Celine, Phung, Van, Kreusch, Andreas, Lu, Min, Hu, Bin, Chaudhary, Apurva, Prashad, Mahavir, Tuntland, Tove, Liu, Bo, Harris, Jennifer, Seidel, H. Martin, Loren, Jon, Molteni, Valentina

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The Banert Cascade: A Synthetic Sequence to Polyfunctional NH-1,2,3-Triazoles von Loren, Jon C., Sharpless, K. Barry

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Synthesis of a D3-symmetric “trefoil” knotted cyclophane von Arias, Karla I, Zysman-Colman, Eli, Loren, Jon C, Linden, Anthony, Siegel, Jay S

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Synthesis and Fluorescence Properties of Manisyl-Substituted Terpyridine, Bipyridine, and Phenanthroline Manisyl=4-methoxy-2,6-dimethylphenyl. This work was supported by the US Nat... von Loren, Jon C., Siegel, Jay S.

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The Banert Cascade: A Synthetic Sequence to Polyfunctional N H-1,2,3-Triazoles von Loren, Jon C., Sharpless, K. Barry

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N H-1,2,3-Triazoles from Azidomethyl Pivalate and Carbamates: Base-Labile N - Protecting Groups von Loren, Jon C., Krasiński, Antoni, Fokin, Valery V., Sharpless, K. Barry

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