Non-Classical Inhibition of Carbonic Anhydrase von Lomelino, Carrie L, Supuran, Claudiu T, McKenna, Robert

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Cancer Drug Development of Carbonic Anhydrase Inhibitors beyond the Active Site von Singh, Srishti, Lomelino, Carrie L, Mboge, Mam Y, Frost, Susan C, McKenna, Robert

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Asparagine synthetase: Function, structure, and role in disease von Lomelino, Carrie L., Andring, Jacob T., McKenna, Robert, Kilberg, Michael S.

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4‑Hydroxy-3-nitro-5-ureido-benzenesulfonamides Selectively Target the Tumor-Associated Carbonic Anhydrase Isoforms IX and XII Showing Hypoxia-Enhanced Antiproliferative Profiles von Nocentini, Alessio, Trallori, Elena, Singh, Srishti, Lomelino, Carrie L, Bartolucci, Gianluca, Di Cesare Mannelli, Lorenzo, Ghelardini, Carla, McKenna, Robert, Gratteri, Paola, Supuran, Claudiu T

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Kinetic and X-ray crystallographic investigations on carbonic anhydrase isoforms I, II, IX and XII of a thioureido analog of SLC-0111 von Lomelino, Carrie L., Mahon, Brian P., McKenna, Robert, Carta, Fabrizio, Supuran, Claudiu T.

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The Structure of Carbonic Anhydrase IX Is Adapted for Low-pH Catalysis von Mahon, Brian P., Bhatt, Avni, Socorro, Lilien, Driscoll, Jenna M., Okoh, Cynthia, Lomelino, Carrie L., Mboge, Mam Y., Kurian, Justin J., Tu, Chingkuang, Agbandje-McKenna, Mavis, Frost, Susan C., McKenna, Robert

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Discovery of β‑Adrenergic Receptors Blocker–Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy von Nocentini, Alessio, Ceruso, Mariangela, Bua, Silvia, Lomelino, Carrie L, Andring, Jacob T, McKenna, Robert, Lanzi, Cecilia, Sgambellone, Silvia, Pecori, Riccardo, Matucci, Rosanna, Filippi, Luca, Gratteri, Paola, Carta, Fabrizio, Masini, Emanuela, Selleri, Silvia, Supuran, Claudiu T

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“Seriously Sweet”: Acesulfame K Exhibits Selective Inhibition Using Alternative Binding Modes in Carbonic Anhydrase Isoforms von Murray, Akilah B, Lomelino, Carrie L, Supuran, Claudiu T, McKenna, Robert

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Carbonic anhydrase II does not exhibit Nitrite reductase or Nitrous Anhydrase Activity von Andring, Jacob T., Lomelino, Carrie L., Tu, Chingkuang, Silverman, David N., McKenna, Robert, Swenson, Erik R.

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Carbonic anhydrase II in complex with carboxylic acid‐based inhibitors von Lomelino, Carrie L., McKenna, Robert

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The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII von Bonardi, Alessandro, Bua, Silvia, Combs, Jacob, Lomelino, Carrie, Andring, Jacob, Osman, Sameh Mohamed, Toti, Alessandra, Di Cesare Mannelli, Lorenzo, Gratteri, Paola, Ghelardini, Carla, McKenna, Robert, Nocentini, Alessio, Supuran, Claudiu T

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Crystallography and Its Impact on Carbonic Anhydrase Research von Lomelino, Carrie L., Andring, Jacob T., McKenna, Robert

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Next Generation Sequencing of the Pig αβ TCR Repertoire Identifies the Porcine Invariant NKT Cell Receptor von Yang, Guan, Artiaga, Bianca L, Lomelino, Carrie L, Jayaprakash, Anitha D, Sachidanandam, Ravi, Mckenna, Robert, Driver, John P

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Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous Bases von Nocentini, Alessio, Bua, Silvia, Lomelino, Carrie L, McKenna, Robert, Menicatti, Marta, Bartolucci, Gianluca, Tenci, Barbara, Di Cesare Mannelli, Lorenzo, Ghelardini, Carla, Gratteri, Paola, Supuran, Claudiu T

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Disruption of the Physical Interaction Between Carbonic Anhydrase IX and the Monocarboxylate Transporter 4 Impacts Lactate Transport in Breast Cancer Cells von Combs, Jacob E., Murray, Akilah B., Lomelino, Carrie L., Mboge, Mam Y., Mietzsch, Mario, Horenstein, Nicole A., Frost, Susan C., McKenna, Robert, Becker, Holger M.

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The splicing component ISY1 regulates APE1 in base excision repair von Jaiswal, Aruna S., Williamson, Elizabeth A., Srinivasan, Gayathri, Kong, Kimi, Lomelino, Carrie L., McKenna, Robert, Walter, Christi, Sung, Patrick, Narayan, Satya, Hromas, Robert

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Crystal Structure of Cleaved Serp-1, a Myxomavirus-Derived Immune Modulating Serpin: Structural Design of Serpin Reactive Center Loop Peptides with Improved Therapeutic Function von Mahon, Brian P, Ambadapadi, Sriram, Yaron, Jordan R, Lomelino, Carrie L, Pinard, Melissa A, Keinan, Shahar, Kurnikov, Igor, Macaulay, Colin, Zhang, Liqiang, Reeves, Westley, McFadden, Grant, Tibbetts, Scott, McKenna, Robert, Lucas, Alexandra R

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Characterization of a novel variant in siblings with Asparagine Synthetase Deficiency von Sacharow, Stephanie J., Dudenhausen, Elizabeth E., Lomelino, Carrie L., Rodan, Lance, El Achkar, Christelle Moufawad, Olson, Heather E., Genetti, Casie A., Agrawal, Pankaj B., McKenna, Robert, Kilberg, Michael S.

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Sweet Binders: Carbonic Anhydrase IX in Complex with Sucralose von Lomelino, Carrie L., Murray, Akilah B., Supuran, Claudiu T., McKenna, Robert

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Mapping Selective Inhibition of the Cancer-Related Carbonic Anhydrase IX Using Structure–Activity Relationships of Glucosyl-Based Sulfamates von Mahon, Brian P, Lomelino, Carrie L, Ladwig, Janina, Rankin, Gregory M, Driscoll, Jenna M, Salguero, Antonieta L, Pinard, Melissa A, Vullo, Daniela, Supuran, Claudiu T, Poulsen, Sally-Ann, McKenna, Robert

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