Optimization of the in Vitro and in Vivo Properties of a Novel Series of 2,4,5-Trisubstituted Imidazoles as Potent Cholecystokinin-2 (CCK2) Antagonists von Buck, Ildiko M, Black, James W, Cooke, Tracey, Dunstone, David J, Gaffen, John D, Griffin, Eric P, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Lilley, Elliot J, Linney, Ian D, Low, Caroline M. R, McDonald, Iain M, Pether, Michael J, Roberts, Sonia P, Shankley, Nigel P, Shaxted, Mark E, Steel, Katherine I. M, Sykes, David A, Tozer, Matthew J, Watt, Gillian F, Walker, Martin K, Wright, Laurence, Wright, Paul T

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2,7-Dioxo-2,3,4,5,6,7-hexahydro-1H-benzo[h][1,4]diazonine as a New Template for the Design of CCK2 Receptor Antagonists von McDonald, Iain M, Dunstone, David J, Kalindjian, S. Barret, Linney, Ian D, Low, Caroline M. R, Pether, Michael J, Steel, Katherine I. M, Tozer, Matthew J, Vinter, J. G

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Design, Synthesis, and Structure−Activity Relationships of Novel Non-Imidazole Histamine H3 Receptor Antagonists von Linney, Ian D, Buck, Ildiko M, Harper, Elaine A, Kalindjian, S. Barret, Pether, Michael J, Shankley, Nigel P, Watt, Gillian F, Wright, Paul T

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Partial Reduction of Annulated Heterocycles as a General Route to Medium Rings Containing Oxygen and Nitrogen von Donohoe, Timothy J, Raoof, Ali, Linney, Ian D, Helliwell, Madeleine

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Novel, Achiral 1,3,4-Benzotriazepine Analogues of 1,4-Benzodiazepine-Based CCK2 Antagonists That Display High Selectivity over CCK1 Receptors von McDonald, Iain M, Austin, Carol, Buck, Ildiko M, Dunstone, David J, Griffin, Eric, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Linney, Ian D, Low, Caroline M. R, Pether, Michael J, Spencer, John, Wright, Paul T, Adatia, Trushar, Bashall, Alan

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Optimization of 1,3,4-Benzotriazepine-Based CCK sub(2) Antagonists to Obtain Potent, Orally Active Inhibitors of Gastrin-Mediated Gastric Acid Secretion von McDonald, I M, Black, J W, Buck, I M, Dunstone, D J, Griffin, E P, Harper, E A, Hull, RAD, Kalindjian, S B, Lilley, E J, Linney, I D, Pether, MJ, Roberts, S P, Shaxted, ME, Spencer, J

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Novel, Achiral 1,3,4-Benzotriazepine Analogues of 1,4-Benzodiazepine-Based CCK sub(2) Antagonists That Display High Selectivity over CCK sub(1) Receptors von McDonald, I M, Austin, C, Buck, I M, Dunstone, D J, Griffin, E, Harper, E A, Hull, RAD, Kalindjian, S B, Linney, I D, Low, CMR, Pether, MJ, Spencer, J, Wright, P T, Adatia, T, Bashall, A

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Design, Synthesis, and Structure−Activity Relationships of Novel Non-Imidazole Histamine H 3 Receptor Antagonists von Linney, Ian D., Buck, Ildiko M., Harper, Elaine A., Kalindjian, S. Barret, Pether, Michael J., Shankley, Nigel P., Watt, Gillian F., Wright, Paul T.

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Recoverable chiral sulfoxides for asymmetric synthesis : preparation, regeneration and application to the asymmetric aldol reaction von BUTLIN, R. J, LINNEY, I. D, CRITCHER, D. J, MAHON, M. F, MOLLOY, K. C, WILLS, M

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Dependence of ring closure stereoselectivity on the nature of the leaving group : application to the synthesis of a new class of chiral sulfoxide for the control of asymmetric aldo... von WILLS, M, BUTLIN, R. J, LINNEY, I. D, GIBSON, R. W

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2,7-Dioxo-2,3,4,5,6,7-hexahydro-1H-benzo[h][1,4]diazonine as a new template for the design of CCK(2) receptor antagonists von McDonald, I M, Dunstone, D J, Kalindjian, S B, Linney, I D, Low, C M, Pether, M J, Steel, K I, Tozer, M J, Vinter, J G

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Synthesis of Enantiopure Dihydropyranones:  Aldol-Based Ring Expansion of Dihydrofurans von Donohoe, Timothy J, Raoof, Ali, Freestone, Graeme C, Linney, Ian D, Cowley, Andrew, Helliwell, Madeleine

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Design, synthesis, and structure-activity relationships of novel non-imidazole histamine H(3) receptor antagonists von Linney, I D, Buck, I M, Harper, E A, Kalindjian, S B, Pether, M J, Shankley, N P, Watt, G F, Wright, P T

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The total synthesis of epibatidine von KO, S. Y, LERPINIERE, J, LINNEY, I. D, WRIGGLESWORTH, R

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A new class of recoverable chiral sulphoxide: Application to the asymmetric synthesis of β-hydroxy esters von Wills, Martin, Butlin, Roger J., Linney, Ian D.

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The asymmetric synthesis of allylic alcohols using a recoverable chiral sulphoxide von Linney, Ian D., Tye, Heather, Wills, Martin, Butlin, Roger J.

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A Convenient Synthesis of N-Alkyl-(E)-1-alkenesulfonamides von Tozer, Matthew J., Woolford, Alison J. A., Linney, Ian D.

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ChemInform Abstract: A Convenient Synthesis of N-Alkyl-(E)-1-alkenesulfonamides von TOZER, M. J., WOOLFORD, A. J. A., LINNEY, I. D.

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Gastrin and cholecystokinin receptor ligands von I. M. BUCK, S. B. KALINDJIAN, I. D. LINNEY

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Recoverable chiral sulfoxides for asymmetric synthesis: application to stereoselective carbonyl reduction and the asymmetric synthesis of allylic alcohols von Butlin, Roger J., Linney, Ian D., Mahon, Mary F., Tye, Heather, Wills, Martin

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