Conazoles von Heeres, Jan, Meerpoel, Lieven, Lewi, Paul

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Access to Silylated Pyrazole Derivatives by Palladium-Catalyzed C−H Activation of a TMS group von Mistico, Laetitia, Querolle, Olivier, Meerpoel, Lieven, Angibaud, Patrick, Durandetti, Muriel, Maddaluno, Jacques

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Cobalt-Catalyzed Diastereoselective Synthesis of C‑Furanosides. Total Synthesis of (−)-Isoaltholactone von Nicolas, Lionel, Izquierdo, Eva, Angibaud, Patrick, Stansfield, Ian, Meerpoel, Lieven, Reymond, Sébastien, Cossy, Janine

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Iron-Catalyzed Synthesis of C2 Aryl- and N‑Heteroaryl-Substituted Tetrahydropyrans von Bosset, Cyril, Angibaud, Patrick, Stanfield, Ian, Meerpoel, Lieven, Berthelot, Didier, Guérinot, Amandine, Cossy, Janine

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Tandem Suzuki-Miyaura Coupling/Acid-Catalyzed Cyclization between Vinyl Ether Boronates and Vinyl Halides: A Concise Approach to Polysubstituted Furans von Butkevich, Alexey N, Meerpoel, Lieven, Stansfield, Ian, Angibaud, Patrick, Corbu, Andrei, Cossy, Janine

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Diastereoselective Metal-Catalyzed Synthesis of C-Aryl and C-Vinyl Glycosides von Nicolas, Lionel, Angibaud, Patrick, Stansfield, Ian, Bonnet, Pascal, Meerpoel, Lieven, Reymond, Sébastien, Cossy, Janine

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Direct α-Functionalization of Saturated Cyclic Amines von Mitchell, Emily A., Peschiulli, Aldo, Lefevre, Nicolas, Meerpoel, Lieven, Maes, Bert U. W.

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Organic glasses with tunable liquid-crystalline order through kinetic arrest of end-over-end rotation: the case of saperconazole von Chen, Zhenxuan, Yu, Junguang, Teerakapibal, Rattavut, Meerpoel, Lieven, Richert, Ranko, Yu, Lian

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The Novel Azole R126638 Is a Selective Inhibitor of Ergosterol Synthesis in Candida albicans, Trichophyton spp., and Microsporum canis von VANDEN BOSSCHE, Hugo, AUSMA, Jannie, BOHETS, Hilde, VERMUYTEN, Karen, WILLEMSENS, Gustaaf, MARICHAL, Patrick, MEERPOEL, Lieven, ODDS, Frank, BORGERS, Marcel

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Minisci-Photoredox-Mediated α‑Heteroarylation of N‑Protected Secondary Amines: Remarkable Selectivity of Azetidines von Bosset, Cyril, Beucher, Hélène, Bretel, Guillaume, Pasquier, Elisabeth, Queguiner, Laurence, Henry, Cyril, Vos, Ann, Edwards, James P, Meerpoel, Lieven, Berthelot, Didier

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C-2 Arylation of Piperidines through Directed Transition-Metal-Catalyzed sp3 CH Activation von Prokopcová, Hana, Bergman, Sheba D., Aelvoet, Karel, Smout, Veerle, Herrebout, Wouter, Van der Veken, Benjamin, Meerpoel, Lieven, Maes, Bert U. W.

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Discovery and Pharmacological Characterization of JNJ-64619178, a Novel Small-Molecule Inhibitor of PRMT5 with Potent Antitumor Activity von Brehmer, Dirk, Beke, Lijs, Wu, Tongfei, Millar, Hillary J, Moy, Christopher, Sun, Weimei, Mannens, Geert, Pande, Vineet, Boeckx, An, van Heerde, Erika, Nys, Thomas, Gustin, Emmanuel M, Verbist, Bie, Zhou, Longen, Fan, Yue, Bhargava, Vipul, Safabakhsh, Pegah, Vinken, Petra, Verhulst, Tinne, Gilbert, Angelique, Rai, Sumit, Graubert, Timothy A, Pastore, Friederike, Fiore, Danilo, Gu, Junchen, Johnson, Amy, Philippar, Ulrike, Morschhäuser, Barbara, Walker, David, De Lange, Desiree, Keersmaekers, Vikki, Viellevoye, Marcel, Diels, Gaston, Schepens, Wim, Thuring, Jan Willem, Meerpoel, Lieven, Packman, Kathryn, Lorenzi, Matthew V, Laquerre, Sylvie

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Stereodivergent Synthesis of Biologically Active Spironucleoside Scaffolds via Catalytic Cyclopropanation of 4-exo-Methylene Furanosides von Neouchy, Zeina, Verhoeven, Jonas, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Brambilla, Marta, Van Hecke, Kristof, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido, Winne, Johan

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Regio- and Stereoselective Synthesis of C‑4′ Spirocyclobutyl Ribofuranose Scaffolds and Their Use as Biologically Active Nucleoside Analogues von Jouffroy, Lucile, Verhoeven, Jonas, Brambilla, Marta, Verniest, Guido, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Meerpoel, Lieven, Thuring, Jan Willem, Winne, Johan M

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Synthesis and Reactivity of Spirocarbocycles as Scaffolds for Nucleoside Analogues von Verhoeven, Jonas, Deraet, Xavier, Pande, Vineet, Sun, Weimei, Alonso, Mercedes, De Proft, Frank, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido

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Iron-Catalyzed Synthesis of Sulfur-Containing Heterocycles von Bosset, Cyril, Lefebvre, Gauthier, Angibaud, Patrick, Stansfield, Ian, Meerpoel, Lieven, Berthelot, Didier, Guérinot, Amandine, Cossy, Janine

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Synthesis and transformations of pyrrolo[1,2-a][1,3,5]-triazines von Verhoeven, Jonas, Reddy, B. Narendraprasad, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido

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Correction to “Regio- and Stereoselective Synthesis of C‑4′ Spirocyclobutyl Ribofuranose Scaffolds and Their Use as Biologically Active Nucleoside Analogues” von Jouffroy, Lucile, Verhoeven, Jonas, Brambilla, Marta, Verniest, Guido, Kong, Hanchu, Zhao, Yongbin, Wang, Wenbin, Meerpoel, Lieven, Thuring, Jan Willem, Winne, Johan M

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Discovery of JNJ-63576253: A Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC) von Zhang, Zhuming, Connolly, Peter J, Lim, Heng Keang, Pande, Vineet, Meerpoel, Lieven, Teleha, Christopher, Branch, Jonathan R, Ondrus, Janine, Hickson, Ian, Bush, Tammy, Luistro, Leopoldo, Packman, Kathryn, Bischoff, James R, Ibrahim, Salam, Parrett, Christopher, Chong, Yolanda, Gottardis, Marco M, Bignan, Gilles

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Preparation of 4′‐Spirocyclobutyl Nucleoside Analogues as Novel and Versatile Adenosine Scaffolds von Verhoeven, Jonas, De Vleeschouwer, Freija, Kong, Hanchu, Van Hecke, Kristof, Pande, Vineet, Sun, Weimei, Vos, Ann, Wu, Tongfei, Meerpoel, Lieven, Thuring, Jan Willem, Verniest, Guido

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