Enantioselective Synthesis of 4′-Ethynyl-2-fluoro-2′-deoxyadenosine (EFdA) via Enzymatic Desymmetrization von McLaughlin, Mark, Kong, Jongrock, Belyk, Kevin M, Chen, Billy, Gibson, Andrew W, Keen, Stephen P, Lieberman, David R, Milczek, Erika M, Moore, Jeffrey C, Murray, David, Peng, Feng, Qi, Ji, Reamer, Robert A, Song, Zhiguo J, Tan, Lushi, Wang, Lin, Williams, Michael J

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Syntheses of Indoles via a Palladium-Catalyzed Annulation between Iodoanilines and Ketones von Chen, Cheng-yi, Lieberman, David R, Larsen, Robert D, Verhoeven, Thomas R, Reider, Paul J

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Efficient Synthesis of Losartan, A Nonpeptide Angiotensin II Receptor Antagonist von Larsen, Robert D, King, Anthony O, Chen, Cheng Y, Corley, Edward G, Foster, Bruce S, Roberts, F. Edward, Yang, Chunhua, Lieberman, David R, Reamer, Robert A, Tschaen, David M, Verhoeven, Thomas R, Reider, Paul J, Lo, Young S, Rossano, Lucius T, Brookes, A. Sidney, Meloni, David, Moore, James R, Arnett, John F

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Process Development of the HCV NS5B Site D Inhibitor MK-8876 von Williams, Michael J, Chen, Qinghao, Codan, Lorenzo, Dermenjian, Renee K, Dreher, Spencer, Gibson, Andrew W, He, Xianliang, Jin, Yan, Keen, Stephen P, Lee, Alfred Y, Lieberman, David R, Lin, Wei, Liu, Guiquan, McLaughlin, Mark, Reibarkh, Mikhail, Scott, Jeremy P, Strickfuss, Sophie, Tan, Lushi, Varsolona, Richard J, Wen, Feng

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A Practical Synthesis of a γ-Secretase Inhibitor von Scott, Jeremy P, Lieberman, David R, Beureux, Olivier M, Brands, Karel M. J, Davies, Antony J, Gibson, Andrew W, Hammond, Deborah C, McWilliams, Chris J, Stewart, Gavin W, Wilson, Robert D, Dolling, Ulf-H

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A Novel Crystallization-Induced Diastereomeric Transformation Based on a Reversible Carbon−Sulfur Bond Formation. Application to the Synthesis of a γ-Secretase Inhibitor von Davies, Antony J, Scott, Jeremy P, Bishop, Brian C, Brands, Karel M. J, Brewer, Sarah E, DaSilva, Jimmy O, Dormer, Peter G, Dolling, Ulf-H, Gibb, Andrew D, Hammond, Deborah C, Lieberman, David R, Palucki, Michael, Payack, Joseph F

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A Practical and Efficient Preparation of the Releasable Naphthosultam Side Chain of a Novel Anti-MRSA Carbapenem von Miller, Ross A, Humphrey, Guy R, Lieberman, David R, Ceglia, Scott S, Kennedy, Derek J, Grabowski, Edward J. J, Reider, Paul J

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The conformational bias of aryl, arylsulfonyl geminally substituted tertiary carbon centers: applications in substrate-based stereocontrol von Scott, Jeremy P, Mullens, Peter R, Brewer, Sarah E, Brands, Karel M J, Chilenski, Jennifer R, Davies, Antony J, Gibb, Andrew D, Lieberman, David R, Oliver, Steven F, Dolling, Ulf-H

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Synthesis of the 5-HT1D receptor agonist MK-0462 via a Pd-catalyzed coupling reaction von CHENG-YI CHEN, LIEBERMAN, D. R, LARSEN, R. D, REAMER, R. A, VERHOEVEN, T. R, REIDER, P. J, COTTRELL, I. F, HOUGHTON, P. G

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Practical Asymmetric Synthesis of a Non-Peptidic αvβ3 Antagonist von Keen, Stephen P, Cowden, Cameron J, Bishop, Brian C, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf H, Lieberman, David R, Stewart, Gavin W

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Employment of on-line FT-IR spectroscopy to monitor the deprotection of a 9-fluorenylmethyl protected carboxylic acid peptide conjugate of doxorubicin von Cameron, Mark, Zhou, George X, Hicks, Micheal B, Antonucci, Vincent, Ge, Zhihong, Lieberman, David R, Lynch, Joesph E, Shi, Yao-Jun

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In Situ Moisture Determination of a Cytotoxic Compound During Process Optimization von Hicks, Michael B., Zhou, George X., Lieberman, David R., Antonucci, Vincent, Ge, Zhihong, Shi, Yao‐Jun, Cameron, Mark, Lynch, Joseph E.

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Practical Asymmetric Synthesis of a Non-Peptidic α v β 3 Antagonist von Keen, Stephen P., Cowden, Cameron J., Bishop, Brian C., Brands, Karel M. J., Davies, Antony J., Dolling, Ulf H., Lieberman, David R., Stewart, Gavin W.

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An efficient one-pot synthesis of annulated pyridines utilising a directed ortho-metallation/transmetallation approach von Davies, Antony J., Brands, Karel M.J., Cowden, Cameron J., Dolling, Ulf-H., Lieberman, David R.

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Practical asymmetric synthesis of a non-peptidic alphavbeta3 antagonist von Keen, Stephen P, Cowden, Cameron J, Bishop, Brian C, Brands, Karel M J, Davies, Antony J, Dolling, Ulf H, Lieberman, David R, Stewart, Gavin W

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An Efficient Synthesis of a Doxorubicin-Peptide Conjugate von Shi, Yao-Jun, Cameron, Mark, Dolling, Ulf H., Lieberman, David R., Lynch, Joseph E., Reamer, Robert A., Robbins, Michael A., Volante, R. P., Reider, Paul J.

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PROCESS FOR PREPARING ( (1S, 2S) -2- (5-METHYLPYRIDIN-2-YL) CYCLOPROPYL) -METHANOL von LI, Donglin, SHANG, Gao, SNEAD, David R, XIAO, Chengqian, GIBSON, Andrew W, CHUNG, John Y. L, ZHAO, Xiaxia, LIEBERMAN, David R, LÉVESQUE, François, ZHAO, Zhenbing, TAN, Lushi

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PROCESS FOR PREPARING ((1S,2S)-2-(5-METHYLPYRIDIN-2-YL)CYCLOPROPYL)-METHANOL von LI, Donglin, SHANG, Gao, SNEAD, David R, LEVESQUE, Francois, XIAO, Chengqian, GIBSON, Andrew W, CHUNG, John Y. L, ZHAO, Xiaxia, LIEBERMAN, David R, ZHAO, Zhenbing, TAN, Lushi

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An Efficient Synthesis of aDoxorubicin-Peptide Conjugate von Shi, Yao-Jun, Cameron, Mark, Dolling, Ulf H., Lieberman, David R., Lynch, Joseph E., Reamer, Robert A., Robbins, Michael A., Volante, R. P., Reider, Paul J.

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4'-SUBSTITUTED NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS AND PREPARATIONS THEREOF von CLEATOR, EDWARD, DIEGUEZ VAZQUEZ, ALEJANDRO, SONG, ZHIGUO JAKE, KONG, JONGROCK, KEEN, STEPHEN PHILIP, MOORE, JEFFREY C, GIBSON, ANDREW WILLIAM, LIEBERMAN, DAVID R, WILLIAMS, MICHAEL J, MCLAUGHLIN, MARK, PENG, FENG, GIRIJAVALLABHAN, VINAY M, MILCZEK, ERIKA M, BELYK, KEVIN M

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