INCB054828 (pemigatinib), a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3, displays activity against genetically defined tumor models von Liu, Phillip C C, Koblish, Holly, Wu, Liangxing, Bowman, Kevin, Diamond, Sharon, DiMatteo, Darlise, Zhang, Yue, Hansbury, Michael, Rupar, Mark, Wen, Xiaoming, Collier, Paul, Feldman, Patricia, Klabe, Ronald, Burke, Krista A, Soloviev, Maxim, Gardiner, Christine, He, Xin, Volgina, Alla, Covington, Maryanne, Ruggeri, Bruce, Wynn, Richard, Burn, Timothy C, Scherle, Peggy, Yeleswaram, Swamy, Yao, Wenqing, Huber, Reid, Hollis, Gregory

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A new synthesis of symmetric boraindacene (BODIPY) dyes von Wu, Liangxing, Burgess, Kevin

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Synthesis and Spectroscopic Properties of Rosamines with Cyclic Amine Substituents von Wu, Liangxing, Burgess, Kevin

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Functionalized BF2 chelated azadipyrromethene dyes von Loudet, Aurore, Bandichhor, Rakeshwar, Wu, Liangxing, Burgess, Kevin

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Abstract ND01: Discovery of INCB86550: A potent, orally bioavailable small molecule inhibitor of PDL1 for the treatment of cancer von Wu, Liangxing

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Syntheses of Highly Fluorescent GFP-Chromophore Analogues von Wu, Liangxing, Burgess, Kevin

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Fluorescent Cassettes for Monitoring Three-Component Interactions in Vitro and in Living Cells von Wu, Liangxing, Loudet, Aurore, Barhoumi, Rola, Burghardt, Robert C, Burgess, Kevin

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Rosamines targeting the cancer oxidative phosphorylation pathway von Lim, Siang Hui, Wu, Liangxing, Kiew, Lik Voon, Chung, Lip Yong, Burgess, Kevin, Lee, Hong Boon

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High-contrast fluorescence imaging in fixed and living cells using optimized optical switches von Wu, Liangxing, Dai, Yingrui, Jiang, Xiaoli, Petchprayoon, Chutima, Lee, Jessie E, Jiang, Tao, Yan, Yuling, Marriott, Gerard

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Organelle-selective energy transfer: A fluorescent indicator of intracellular environment von Loudet, Aurore, Ueno, Yuichiro, Wu, Liangxing, Jose, Jiney, Barhoumi, Rola, Burghardt, Robert, Burgess, Kevin

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Fluorescent Amino- and Thiopyronin Dyes von Wu, Liangxing, Burgess, Kevin

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Discovery of Pemigatinib: A Potent and Selective Fibroblast Growth Factor Receptor (FGFR) Inhibitor von Wu, Liangxing, Zhang, Colin, He, Chunhong, Qian, Dingquan, Lu, Liang, Sun, Yaping, Xu, Meizhong, Zhuo, Jincong, Liu, Phillip C. C, Klabe, Ronald, Wynn, Richard, Covington, Maryanne, Gallagher, Karen, Leffet, Lynn, Bowman, Kevin, Diamond, Sharon, Koblish, Holly, Zhang, Yue, Soloviev, Maxim, Hollis, Gregory, Burn, Timothy C, Scherle, Peggy, Yeleswaram, Swamy, Huber, Reid, Yao, Wenqing

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Characterization of INCB086550: A Potent and Novel Small-Molecule PD-L1 Inhibitor von Koblish, Holly K, Wu, Liangxing, Wang, Liang-Chuan S, Liu, Phillip C C, Wynn, Richard, Rios-Doria, Jonathan, Spitz, Susan, Liu, Hao, Volgina, Alla, Zolotarjova, Nina, Kapilashrami, Kanishk, Behshad, Elham, Covington, Maryanne, Yang, Yan-Ou, Li, Jingwei, Diamond, Sharon, Soloviev, Maxim, O'Hayer, Kevin, Rubin, Stephen, Kanellopoulou, Chrysi, Yang, Gengjie, Rupar, Mark, DiMatteo, Darlise, Lin, Luping, Stevens, Christina, Zhang, Yue, Thekkat, Pramod, Geschwindt, Ryan, Marando, Cindy, Yeleswaram, Swamy, Jackson, Jeff, Scherle, Peggy, Huber, Reid, Yao, Wenqing, Hollis, Gregory

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Abstract 1134: The LSD1 inhibitor INCB059872 is a possible therapeutic option for venetoclax-resistant AML von Diamond, Melody, Chadderton, Antony, He, Chunhong, Wu, Liangxing, Yao, Wenqing, Koblish, Holly, Lee, Sang Hyun, Stubbs, Matthew C.

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Inhibition of ALK2 with bicyclic pyridyllactams von Witten, Michael R., Wu, Liangxing, Lai, Cheng-Tsung, Kapilashrami, Kanishk, Pusey, Michelle, Gallagher, Karen, Chen, Yaoyu, Yao, Wenqing

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Discovery of (4-Pyrazolyl)-2-aminopyrimidines as Potent and Selective Inhibitors of Cyclin-Dependent Kinase 2 von Hummel, Joshua R., Xiao, Kai-Jiong, Yang, Jeffrey C., Epling, Leslie B., Mukai, Ken, Ye, Qinda, Xu, Meizhong, Qian, Dingquan, Huo, Lu, Weber, Michael, Roman, Valerie, Lo, Yvonne, Drake, Katherine, Stump, Kristine, Covington, Maryanne, Kapilashrami, Kanishk, Zhang, Guofeng, Ye, Min, Diamond, Sharon, Yeleswaram, Swamy, Macarron, Ricardo, Deller, Marc C., Wee, Susan, Kim, Sunkyu, Wang, Xiaozhao, Wu, Liangxing, Yao, Wenqing

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Optical Control of Calcium Affinity in a Spiroamido-rhodamine Based Calcium Chelator von Wu, Liangxing, Dai, Yingrui, Marriott, Gerard

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Preparation and characterization of ZnTiO3–TiO2/pillared montmorillonite composite catalyst for enhanced photocatalytic activity von Wu, Liangxing, Wu, Pingxiao, Zhu, Yajie, Zhu, Nengwu, Dang, Zhi

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Discovery of 5,7-Dihydro‑6H‑pyrrolo[2,3‑d]pyrimidin-6-ones as Highly Selective CDK2 Inhibitors von Sokolsky, Alexander, Winterton, Sarah, Kennedy, Keith, Drake, Katherine, Stump, Kristine, Huo, Lu, Lo, Yvonne, Ye, Min, Covington, Maryanne, Diamond, Sharon, Yang, Yan-ou, Kim, Sunkyu, Yeleswaram, Swamy, Wu, Liangxing, Yao, Wenqing

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Discovery of 5,7-Dihydro-6 H -pyrrolo[2,3- d ]pyrimidin-6-ones as Highly Selective CDK2 Inhibitors von Sokolsky, Alexander, Winterton, Sarah, Kennedy, Keith, Drake, Katherine, Stump, Kristine, Huo, Lu, Lo, Yvonne, Ye, Min, Covington, Maryanne, Diamond, Sharon, Yang, Yan-ou, Kim, Sunkyu, Yeleswaram, Swamy, Wu, Liangxing, Yao, Wenqing

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