Enantioselective Total Synthesis of (+)-Salvileucalin B von Levin, Sergiy, Nani, Roger R, Reisman, Sarah E

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An Integrated Approach toward NanoBRET Tracers for Analysis of GPCR Ligand Engagement von Killoran, Michael P., Levin, Sergiy, Boursier, Michelle E., Zimmerman, Kristopher, Hurst, Robin, Hall, Mary P., Machleidt, Thomas, Kirkland, Thomas A., Friedman Ohana, Rachel

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Rapid Assembly of the Salvileucalin B Norcaradiene Core von Levin, Sergiy, Nani, Roger R, Reisman, Sarah E

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Equilibrium and Kinetic Measurements of Ligand Binding to HiBiT-tagged GPCRs on the Surface of Living Cells von Boursier, Michelle E, Levin, Sergiy, Hurst, Robin, Ohana, Rachel Friedman

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Scalable Regioselective Synthesis of Rhodamine Dyes von Dwight, Stephen J, Levin, Sergiy

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Target engagement and drug residence time can be observed in living cells with BRET von Robers, Matthew B., Dart, Melanie L., Woodroofe, Carolyn C., Zimprich, Chad A., Kirkland, Thomas A., Machleidt, Thomas, Kupcho, Kevin R., Levin, Sergiy, Hartnett, James R., Zimmerman, Kristopher, Niles, Andrew L., Ohana, Rachel Friedman, Daniels, Danette L., Slater, Michael, Wood, Monika G., Cong, Mei, Cheng, Yi-Qiang, Wood, Keith V.

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The luminescent HiBiT peptide enables selective quantitation of G protein–coupled receptor ligand engagement and internalization in living cells von Boursier, Michelle E., Levin, Sergiy, Zimmerman, Kris, Machleidt, Thomas, Hurst, Robin, Butler, Braeden L., Eggers, Christopher T., Kirkland, Thomas A., Wood, Keith V., Friedman Ohana, Rachel

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Streamlined Target Deconvolution Approach Utilizing a Single Photoreactive Chloroalkane Capture Tag von Friedman Ohana, Rachel, Levin, Sergiy, Hurst, Robin, Rosenblatt, Michael M, Zimmerman, Kristopher, Machleidt, Thomas, Wood, Keith V, Kirkland, Thomas A

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Utilizing a Simple Method for Stoichiometric Protein Labeling to Quantify Antibody Blockade von Friedman Ohana, Rachel, Hurst, Robin, Rosenblatt, Mike, Levin, Sergiy, Machleidt, Thomas, Kirkland, Thomas A., Encell, Lance P., Robers, Matthew B., Wood, Keith V.

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Luminogenic HiBiT Peptide-Based NanoBRET Ligand Binding Assays for Melatonin Receptors von Gbahou, Florence, Levin, Sergiy, Tikhonova, Irina G., Somalo Barranco, Gloria, Izabelle, Charlotte, Ohana, Rachel Friedman, Jockers, Ralf

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Deciphering the Cellular Targets of Bioactive Compounds Using a Chloroalkane Capture Tag von Friedman Ohana, Rachel, Kirkland, Thomas A, Woodroofe, Carolyn C, Levin, Sergiy, Uyeda, H. Tetsuo, Otto, Paul, Hurst, Robin, Robers, Matthew B, Zimmerman, Kris, Encell, Lance P, Wood, Keith V

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Abstract C158: A chemoproteomics strategy for target identification and lead compound optimization using chloroalkane derivatized compounds von Ford, Michael, Jones, Richard, Amunugama, Ravi, Daniels, Danette, Ohana, Rachel, Levin, Sergiy, Kirkland, Thomas, Urh, Marjeta, Wood, Keith

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Abstract B161: Chemoproteomic profiling for target identification using chloroalkane derivatized compounds von Ford, Michael, Jones, Richard, Amunugama, Ravi, Daniels, Danette, Ohana, Rachel, Levin, Sergiy, Kirkland, Thomas, Urh, Marjeta, Wood, Keith

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An Artificial β-Sheet That Dimerizes through Parallel β-Sheet Interactions von Levin, Sergiy, Nowick, James S

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Improved Deconvolution of Protein Targets for Bioactive Compounds Using a Palladium Cleavable Chloroalkane Capture Tag von Friedman Ohana, Rachel, Levin, Sergiy, Wood, Monika G, Zimmerman, Kris, Dart, Melanie L, Schwinn, Marie K, Kirkland, Thomas A, Hurst, Robin, Uyeda, H. Tetsuo, Encell, Lance P, Wood, Keith V

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Abstract 3512: Measuring intracellular target engagement and drug residence time with nanoBRET von Robers, Matthew B., Dart, Melanie, Zimprich, Chad, Kirkland, Thomas, Levin, Sergiy, Machleidt, Thomas, Hartnett, Jim, Zimmerman, Kris, Ohana, Rachel, Daniels, Danette, Cong, Mei, Fan, Frank, Wood, Keith

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Abstract 2446: Decoding phenotypic drug screening targets using a novel chloroalkane capture tag von Friedman Ohana, Rachel, Kirkland, Thomas, Woodroofe, Carolyn, Levin, Sergiy, Hurst, Robin, Otto, Paul, Uyeda, Tetsuo, Ford, Michael, Jones, Richard, Daniels, Danette, Urh, Marjeta, Wood, Keith

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Abstract 2003: Investigating the cellular interactions of BIRB796 analogues using a novel chloroalkane capture tag von Friedman Ohana, Rachel, Hurst, Robin, Kirkland, Thomas, Woodroofe, Carolyn, Levin, Sergiy, Otto, Paul, Uyeda, Tetsuo, Ford, Michael, Jones, Richard, Daniels, Danette, Urh, Marjeta, Wood, Keith

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A New Artificial β-Sheet That Dimerizes through Parallel β-Sheet Interactions von Levin, Sergiy, Nowick, James S

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cationic cysteine-hydrazide as an enrichment tool for the mass spectrometric characterization of bacterial free oligosaccharides von Jang, Kyoung-Soon, Nani, Roger R, Kalli, Anastasia, Levin, Sergiy, Müller, Axel, Hess, Sonja, Reisman, Sarah E, Clemons, William M., Jr

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