Metabotropic glutamate 1 receptor distribution and occupancy in the rat brain: a quantitative autoradiographic study using [ 3H]R214127 von Lavreysen, Hilde, Pereira, Sandrina Nóbrega, Leysen, Joseé E, Langlois, Xavier, Lesage, Anne S.J

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JNJ16259685, a highly potent, selective and systemically active mGlu1 receptor antagonist von Lavreysen, Hilde, Wouters, Ria, Bischoff, François, Nóbrega Pereira, Sandrina, Langlois, Xavier, Blokland, Saskia, Somers, Marijke, Dillen, Lieve, Lesage, Anne S.J.

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Metabotropic glutamate receptor 1 blockade impairs acquisition and retention in a spatial Water maze task von Steckler, Thomas, Oliveira, Ana F.M., Van Dyck, Chistophe, Van Craenendonck, Hansfried, Mateus, Ana M.A., Langlois, Xavier, Lesage, Anne S.J., Prickaerts, Jos

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Characterization of 2-[[4-Fluoro-3-(trifluoromethyl)phenyl]amino]-4-(4-pyridinyl)-5-thiazolemethanol (JNJ-1930942), a Novel Positive Allosteric Modulator of the α7 Nicotinic Acetyl... von Dinklo, Theo, Shaban, Hamdy, Thuring, Jan Willem, Lavreysen, Hilde, Stevens, Karen E., Zheng, Lijun, Mackie, Claire, Grantham, Christopher, Vandenberk, Ine, Meulders, Greet, Peeters, Luc, Verachtert, Hanne, De Prins, Erik, Lesage, Anne S.J.

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Synthesis, Structure−Activity Relationship, and Receptor Pharmacology of a New Series of Quinoline Derivatives Acting as Selective, Noncompetitive mGlu1 Antagonists von Mabire, Dominique, Coupa, Sophie, Adelinet, Christophe, Poncelet, Alain, Simonnet, Yvan, Venet, Marc, Wouters, Ria, Lesage, Anne S. J, Beijsterveldt, Ludy Van, Bischoff, François

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Effects of mGlu1 receptor blockade on anxiety-related behaviour in the rat lick suppression test von Steckler, Thomas, Lavreysen, Hilde, Oliveira, Ana M, Aerts, Nancy, Van Craenendonck, Hansfried, Prickaerts, Jos, Megens, Anton, Lesage, Anne S J

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[3H]R214127: A Novel High-Affinity Radioligand for the mGlu1 Receptor Reveals a Common Binding Site Shared by Multiple Allosteric Antagonists von Lavreysen, Hilde, Janssen, Cor, Bischoff, François, Langlois, Xavier, Leysen, Josée E., Lesage, Anne S.J.

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Synthesis and inhibitory activities at mGluRs of 3-alkylated and N-alkylated cyclopentyl-glutamate analogues von Ung, Alison T., Pyne, Stephen G., Bischoff, François, Lesage, Anne S.J., Skelton, Brian W., White, Allan H.

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Synthesis and Biological Activities of Conformationally Restricted Cyclopentenyl-Glutamate Analogues von Ung, Alison T, Schafer, Karl, Lindsay, Karl B, Pyne, Stephen G, Amornraksa, Kitti, Wouters, Ria, Van der Linden, Ilse, Biesmans, Ilse, Lesage, Anne S. J, Skelton, Brian W, White, Allan H

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Binding of GDNF and neurturin to human GDNF family receptor alpha 1 and 2. Influence of cRET and cooperative interactions von Cik, M, Masure, S, Lesage, A S, Van Der Linden, I, Van Gompel, P, Pangalos, M N, Gordon, R D, Leysen, J E

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Antagonist-induced supersensitivity of mGlu1 receptor signalling in cerebellar granule cells von Lavreysen, Hilde, Willemoens, Tineke, Leysen, Joseé E., Lesage, Anne S. J.

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Synthesis and antagonist activities of 4-aryl-substituted conformationally restricted cyclopentenyl and cyclopentanyl-glutamate analogues von Ung, Alison T., Pyne, Stephen G., Batenburg-Nguyen, Uta, Davis, Andrew S., Sherif, Azlifa, Bischoff, François, Lesage, Anne S.J.

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Mammalian GFRα-4, a Divergent Member of the GFRα Family of Coreceptors for Glial Cell Line-derived Neurotrophic Factor Family Ligands, Is a Receptor for the Neurotrophic Factor Per... von Masure, Stefan, Cik, Miroslav, Hoefnagel, Evert, Nosrat, Christopher A., Van der Linden, Ilse, Scott, Rizaldy, Van Gompel, Paul, Lesage, Anne S.J., Verhasselt, Peter, Ibáñez, Carlos F., Gordon, Robert D.

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Molecular cloning, expression and tissue distribution of glial‐cell‐line‐derived neurotrophic factor family receptor α‐3 (GFRα‐3) von Masure, Stefan, Cik, Miroslav, Pangalos, Menelas N., Bonaventure, Pascal, Verhasselt, Peter, Lesage, Anne S. J., Leysen, Josee E., Gordon, Robert D.

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Supersensitivity of Human Metabotropic Glutamate 1a Receptor Signaling in L929sA Cells von Lavreysen, Hilde, Le Poul, Emmanuel, Van Gompel, Paul, Dillen, Lieve, Leysen, Josée E, Lesage, Anne S J

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Supersensitivity of Human Metabotropic Glutamate 1a Receptor Signaling in L929sA Cells von Hilde, Lavreysen, Emmanuel, Le Poul, Paul, Van Gompel, Dillen, Lieve, Leysen, Josée E., Lesage, Anne S.J.

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Binding of GDNF and Neurturin to Human GDNF Family Receptor α 1 and 2 von Cik, Miroslav, Masure, Stefan, Lesage, Anne S.J., Van der Linden, Ilse, Van Gompel, Paul, Pangalos, Menelas N., Gordon, Robert D., Leysen, Josée E.

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Enovin, a member of the glial cell-line-derived neurotrophic factor (GDNF) family with growth promoting activity on neuronal cells. Existence and tissue-specific expression of diff... von Masure, S, Geerts, H, Cik, M, Hoefnagel, E, Van Den Kieboom, G, Tuytelaars, A, Harris, S, Lesage, A S, Leysen, J E, Van Der Helm, L, Verhasselt, P, Yon, J, Gordon, R D

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Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands von LAVREYSEN HILDE, LESAGE ANNE S.J, BISCHOFF FRANCOIS P, JANSSEN CORNELUS G.M

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Metabotropic glutamate receptor antagonists von COUPA SOPHIE, MABIRE DOMINIQUE J, PONCELET ALAIN P, LESAGE ANNE S.J, VENET MARC G

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