4-(N-Alkyl- and -Acyl-amino)-1,2,4-triazole-3-thione Analogs as Metallo-beta-Lactamase Inhibitors: Impact of 4-Linker on Potency and Spectrum of Inhibition von Gavara, Laurent, Verdirosa, Federica, Legru, Alice, Mercuri, Paola Sandra, Nauton, Lionel, Sevaille, Laurent, Feller, Georges, Berthomieu, Dorothee, Sannio, Filomena, Marcoccia, Francesca, Tanfoni, Silvia, De Luca, Filomena, Gresh, Nohad, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-Francois

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Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1 von Legru, Alice, Batista, Fernando, Puszko, Anna, Bouillon, Anthony, Maurel, Manon, Martinez, Mariano, Ejjoummany, Abdelaziz, Ortega Varga, Laura, Adler, Pauline, Mechaly, Ariel E, Hadjadj, Margot, Sosnowski, Piotr, Hopfgartner, Gérard, Alzari, Pedro, Blondel, Arnaud, Haouz, Ahmed, Barale, Jean-Christophe, Hernandez, Jean-François

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4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors von Gavara, Laurent, Sevaille, Laurent, De Luca, Filomena, Mercuri, Paola, Bebrone, Carine, Feller, Georges, Legru, Alice, Cerboni, Giulia, Tanfoni, Silvia, Baud, Damien, Cutolo, Giuliano, Bestgen, Benoît, Chelini, Giulia, Verdirosa, Federica, Sannio, Filomena, Pozzi, Cecilia, Benvenuti, Manuela, Kwapien, Karolina, Fischer, Marina, Becker, Katja, Frère, Jean-Marie, Mangani, Stefano, Gresh, Nohad, Berthomieu, Dorothée, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François

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1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity von Legru, Alice, Verdirosa, Federica, Hernandez, Jean-François, Tassone, Giusy, Sannio, Filomena, Benvenuti, Manuela, Conde, Pierre-Alexis, Bossis, Guillaume, Thomas, Caitlyn A., Crowder, Michael W., Dillenberger, Melissa, Becker, Katja, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean-Denis, Gavara, Laurent

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Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates von Legru, Alice, Verdirosa, Federica, Vo-Hoang, Yen, Tassone, Giusy, Vascon, Filippo, Thomas, Caitlyn A., Sannio, Filomena, Corsica, Giuseppina, Benvenuti, Manuela, Feller, Georges, Coulon, Rémi, Marcoccia, Francesca, Devente, Savannah Rowane, Bouajila, Ezeddine, Piveteau, Catherine, Leroux, Florence, Deprez-Poulain, Rebecca, Deprez, Benoît, Licznar-Fajardo, Patricia, Crowder, Michael W., Cendron, Laura, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean-Denis, Hernandez, Jean-François, Gavara, Laurent

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1,2,4-Triazole-3-thione analogues with an arylakyl group at position 4 as metallo-β-lactamase inhibitors von Gavara, Laurent, Verdirosa, Federica, Sevaille, Laurent, Legru, Alice, Corsica, Giuseppina, Nauton, Lionel, Sandra Mercuri, Paola, Sannio, Filomena, De Luca, Filomena, Hadjadj, Margot, Cerboni, Giulia, Vo Hoang, Yen, Licznar-Fajardo, Patricia, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François

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Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1 von Legru, Alice, Batista, Fernando A., Puszko, Anna K., Bouillon, Anthony, Maurel, Manon, Martinez, Mariano, Ejjoummany, Abdelaziz, Ortega Varga, Laura, Adler, Pauline, Méchaly, Ariel, Hadjadj, Margot, Sosnowski, Piotr, Hopfgartner, Gérard, Alzari, Pedro M., Blondel, Arnaud, Haouz, Ahmed, Barale, Jean-Christophe, Hernandez, Jean-François

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1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-b-lactamase inhibitors with re-sensitization activity von Legru, Alice, Verdirosa, Federica, Hernandez, Jean-François, Tassone, Giusi, Sannio, Filomena, Benvenuti, Manuela, Conde, Pierre-Alexis, Bossis, Guillaume, Thomas, Caitlyn A, Crowder, Michael, Dillenberger, Melissa, Becker, Katja, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean-Denis, Gavara, Laurent

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4-Alkyl-1,2,4-triazole-3-thione analogues as metallo-β-lactamase inhibitors von Gavara, Laurent, Legru, Alice, Verdirosa, Federica, Sevaille, Laurent, Nauton, Lionel, Corsica, Giuseppina, Mercuri, Paola Sandra, Sannio, Filomena, Feller, Georges, Coulon, Rémi, De Luca, Filomena, Cerboni, Giulia, Tanfoni, Silvia, Chelini, Giulia, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François

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1,2,4‐Triazole‐3‐Thione Analogues with a 2‐Ethylbenzoic Acid at Position 4 as VIM‐type Metallo‐β‐Lactamase Inhibitors von Verdirosa, Federica, Gavara, Laurent, Sevaille, Laurent, Tassone, Giusy, Corsica, Giuseppina, Legru, Alice, Feller, Georges, Chelini, Giulia, Mercuri, Paola Sandra, Tanfoni, Silvia, Sannio, Filomena, Benvenuti, Manuela, Cerboni, Giulia, De Luca, Filomena, Bouajila, Ezeddine, Vo Hoang, Yen, Licznar‐Fajardo, Patricia, Galleni, Moreno, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean‐Denis, Hernandez, Jean‐François

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4-Alkyl-1,2,4-triazole-3-thione analogues as metallo-b-lactamase inhibitors von Gavara, Laurent, Legru, Alice, Verdirosa, Federica, Sevaille, Laurent, Nauton, Lionel, Corsica, Giuseppina, Mercuri, Paola Sandra, Sannio, Filomena, Feller, Georges, Coulon, Rémi, De luca, Filomena, Cerboni, Giulia, Tanfoni, Silvia, Chelini, Giulia, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François

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4--1,2,4-triazole-3-thione Analogs as Metallo-[beta]-Lactamase Inhibitors: Impact of 4-Linker on Potency and Spectrum of Inhibition von Gavara, Laurent, Verdirosa, Federica, Legru, Alice, Mercuri, Paola Sandra, Nauton, Lionel, Sevaille, Laurent, Feller, Georges, Berthomieu, Dorothee, Sannio, Filomena, Marcoccia, Francesca, Tanfoni, Silvia, De Luca, Filomena, Gresh, Nohad, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-Frangois

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INHIBITORS OF METALLO-BETA-LACTAMASES von HERNANDEZ, JEAN-FRANÇOIS, DOCQUIER, JEAN-DENIS, SEVAILLE, LAURENT, GAVARA, LAURENT, LEGRU, ALICE

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INHIBITORS OF METALLO-BETA-LACTAMASES von DOCQUIER, Jean-Denis, SEVAILLE, Laurent, GAVARA, Laurent, LEGRU, Alice, HERNANDEZ, Jean-François

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INHIBITORS OF METALLO-BETA-LACTAMASES von SEVAILLE, LAURENT, DOCQUIER, JEAN-DENIS, GAVARA, LAURENT, HERNANDEZ, JEAN-FRANCOIS, LEGRU, ALICE

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INHIBITORS OF METALLO-BETA-LACTAMASES von DOCQUIER, Jean-Denis, SEVAILLE, Laurent, GAVARA, Laurent, LEGRU, Alice, HERNANDEZ, Jean-François

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INHIBITORS OF METALLO-BETA-LACTAMASES von LEGRU ALICE, HERNANDEZ JEAN-FRANCOIS, SEVAILLE LAURENT, GAVARA LAURENT, DOCQUIER JEAN-DENIS

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