Antibacterial activity of quinoxalines, quinazolines, and 1,5-naphthyridines von Parhi, Ajit K., Zhang, Yongzheng, Saionz, Kurt W., Pradhan, Padmanava, Kaul, Malvika, Trivedi, Kalkal, Pilch, Daniel S., LaVoie, Edmond J.

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Combining the FtsZ-Targeting Prodrug TXA709 and the Cephalosporin Cefdinir Confers Synergy and Reduces the Frequency of Resistance in Methicillin-Resistant Staphylococcus aureus von Kaul, Malvika, Mark, Lilly, Parhi, Ajit K, LaVoie, Edmond J, Pilch, Daniel S

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Structural Flexibility of an Inhibitor Overcomes Drug Resistance Mutations in Staphylococcus aureus FtsZ von Fujita, Junso, Maeda, Yoko, Mizohata, Eiichi, Inoue, Tsuyoshi, Kaul, Malvika, Parhi, Ajit K, LaVoie, Edmond J, Pilch, Daniel S, Matsumura, Hiroyoshi

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An FtsZ-Targeting Prodrug with Oral Antistaphylococcal Efficacy In Vivo von KAUL, Malvika, MARK, Lilly, YONGZHENG ZHANG, PARHI, Ajit K, LAVOIE, Edmond J, PILCH, Daniel S

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Structure-Guided Design of a Fluorescent Probe for the Visualization of FtsZ in Clinically Important Gram-Positive and Gram-Negative Bacterial Pathogens von Ferrer-González, Edgar, Fujita, Junso, Yoshizawa, Takuya, Nelson, Julia M., Pilch, Alyssa J., Hillman, Elani, Ozawa, Mayuki, Kuroda, Natsuko, Al-Tameemi, Hassan M., Boyd, Jeffrey M., LaVoie, Edmond J., Matsumura, Hiroyoshi, Pilch, Daniel S.

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Pharmacokinetics and in vivo antistaphylococcal efficacy of TXY541, a 1-methylpiperidine-4-carboxamide prodrug of PC190723 von Kaul, Malvika, Mark, Lilly, Zhang, Yongzheng, Parhi, Ajit K., LaVoie, Edmond J., Pilch, Daniel S.

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Crystallographic Fragment Screening and Structure-Based Optimization Yields a New Class of Influenza Endonuclease Inhibitors von Bauman, Joseph D, Patel, Disha, Baker, Steven F, Vijayan, R. S. K, Xiang, Amy, Parhi, Ajit K, Martínez-Sobrido, Luis, LaVoie, Edmond J, Das, Kalyan, Arnold, Eddy

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A FtsZ Inhibitor That Can Utilize Siderophore-Ferric Iron Uptake Transporter Systems for Activity against Gram-Negative Bacterial Pathogens von Bryan, Eric J, Qiao, Qi, Wang, Yuxuan, Roberge, Jacques Y, LaVoie, Edmond J, Pilch, Daniel S

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Antibacterial activity of substituted dibenzo[a,g]quinolizin-7-ium derivatives von Parhi, Ajit, Lu, Songfeng, Kelley, Cody, Kaul, Malvika, Pilch, Daniel S., LaVoie, Edmond J.

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Bioisosterism:  A Rational Approach in Drug Design von Patani, George A, LaVoie, Edmond J

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TXH11106: A Third-Generation MreB Inhibitor with Enhanced Activity against a Broad Range of Gram-Negative Bacterial Pathogens von Bryan, Eric J, Sagong, Hye Yeon, Parhi, Ajit K, Grier, Mark C, Roberge, Jacques Y, LaVoie, Edmond J, Pilch, Daniel S

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Enterococcal and streptococcal resistance to PC190723 and related compounds: Molecular insights from a FtsZ mutational analysis von Kaul, Malvika, Zhang, Yongzheng, Parhi, Ajit K., LaVoie, Edmond J., Tuske, Steve, Arnold, Eddy, Kerrigan, John E., Pilch, Daniel S.

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Antimicrobial activity of various 4- and 5-substituted 1-phenylnaphthalenes von Kelley, Cody, Lu, Songfeng, Parhi, Ajit, Kaul, Malvika, Pilch, Daniel S., LaVoie, Edmond J.

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Antioxidative Phenolic Compounds from Sage (Salvia officinalis) von Wang, Mingfu, Li, Jiangang, Rangarajan, Meera, Shao, Yu, LaVoie, Edmond J, Huang, Tzou-Chi, Ho, Chi-Tang

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Genz-644282, a Novel Non-Camptothecin Topoisomerase I Inhibitor for Cancer Treatment von KURTZBERG, Leslie S, ROTH, Stephanie, FEI WANG, SCHMID, Steven M, LAVOIE, Edmond J, TEICHER, Beverly A, KRUMBHOLZ, Roy, CRAWFORD, Jennifer, BORMANN, Christy, DUNHAM, Sarah, MIN YAO, ROULEAU, Cecile, BAGLEY, Rebecca G, YU, Xian-Jie

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Macrocyclic biphenyl tetraoxazoles: Synthesis, evaluation as G-quadruplex stabilizers and cytotoxic activity von Blankson, Gifty A., Pilch, Daniel S., Liu, Angela A., Liu, Leroy F., Rice, Joseph E., LaVoie, Edmond J.

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Determination of the Predominant Catechins in Acacia catechu by Liquid Chromatography/Electrospray Ionization−Mass Spectrometry von Shen, Diandian, Wu, Qingli, Wang, Mingfu, Yang, Yonghong, Lavoie, Edmond J, Simon, James E

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A G-quadruplex Stabilizer Induces M-phase Cell Cycle Arrest von Tsai, Yuan-Chin, Qi, Haiyan, Lin, Chao-Po, Lin, Ren-Kuo, Kerrigan, John E., Rzuczek, Suzanne G., LaVoie, Edmond J., Rice, Joseph E., Pilch, Daniel S., Lyu, Yi Lisa, Liu, Leroy F.

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Macrocyclic pyridyl polyoxazoles: structure-activity studies of the aminoalkyl side-chain on G-quadruplex stabilization and cytotoxic activity von Blankson, Gifty, Rzuczek, Suzanne G, Bishop, Cody, Pilch, Daniel S, Liu, Angela, Liu, Leroy, Lavoie, Edmond J, Rice, Joseph E

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Structure-activity relationships of potentiators of the antibiotic activity of clarithromycin against Escherichia coli von Blankson, Gifty, Parhi, Ajit K., Kaul, Malvika, Pilch, Daniel S., LaVoie, Edmond J.

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