Monitoring G protein-coupled receptor and β-arrestin trafficking in live cells using enhanced bystander BRET von Namkung, Yoon, Le Gouill, Christian, Lukashova, Viktoria, Kobayashi, Hiroyuki, Hogue, Mireille, Khoury, Etienne, Song, Mideum, Bouvier, Michel, Laporte, Stéphane A.

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A new inhibitor of the β-arrestin/AP2 endocytic complex reveals interplay between GPCR internalization and signalling von Beautrait, Alexandre, Paradis, Justine S., Zimmerman, Brandon, Giubilaro, Jenna, Nikolajev, Ljiljana, Armando, Sylvain, Kobayashi, Hiroyuki, Yamani, Lama, Namkung, Yoon, Heydenreich, Franziska M., Khoury, Etienne, Audet, Martin, Roux, Philippe P., Veprintsev, Dmitry B., Laporte, Stéphane A., Bouvier, Michel

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Functional selectivity profiling of the angiotensin II type 1 receptor using pathway-wide BRET signaling sensors von Namkung, Yoon, LeGouill, Christian, Kumar, Sahil, Cao, Yubo, Teixeira, Larissa B, Lukasheva, Viktoriya, Giubilaro, Jenna, Simões, Sarah C, Longpré, Jean-Michel, Devost, Dominic, Hébert, Terence E, Piñeyro, Graciela, Leduc, Richard, Costa-Neto, Claudio M, Bouvier, Michel, Laporte, Stéphane A

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Dynamic spatiotemporal determinants modulate GPCR:G protein coupling selectivity and promiscuity von Sandhu, Manbir, Cho, Aaron, Ma, Ning, Mukhaleva, Elizaveta, Namkung, Yoon, Lee, Sangbae, Ghosh, Soumadwip, Lee, John H., Gloriam, David E., Laporte, Stéphane A., Babu, M. Madan, Vaidehi, Nagarajan

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Manifold roles of β-arrestins in GPCR signaling elucidated with siRNA and CRISPR/Cas9 von Luttrell, Louis M, Wang, Jialu, Plouffe, Bianca, Smith, Jeffrey S, Yamani, Lama, Kaur, Suneet, Jean-Charles, Pierre-Yves, Gauthier, Christophe, Lee, Mi-Hye, Pani, Biswaranjan, Kim, Jihee, Ahn, Seungkirl, Rajagopal, Sudarshan, Reiter, Eric, Bouvier, Michel, Shenoy, Sudha K, Laporte, Stéphane A, Rockman, Howard A, Lefkowitz, Robert J

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Intrinsic bias at non-canonical, β-arrestin-coupled seven transmembrane receptors von Pandey, Shubhi, Kumari, Punita, Baidya, Mithu, Kise, Ryoji, Cao, Yubo, Dwivedi-Agnihotri, Hemlata, Banerjee, Ramanuj, Li, Xaria X., Cui, Cedric S., Lee, John D., Kawakami, Kouki, Maharana, Jagannath, Ranjan, Ashutosh, Chaturvedi, Madhu, Jhingan, Gagan Deep, Laporte, Stéphane A., Woodruff, Trent M., Inoue, Asuka, Shukla, Arun K.

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The experimental power of FR900359 to study Gq-regulated biological processes von Schrage, Ramona, Schmitz, Anna-Lena, Gaffal, Evelyn, Annala, Suvi, Kehraus, Stefan, Wenzel, Daniela, Büllesbach, Katrin M., Bald, Tobias, Inoue, Asuka, Shinjo, Yuji, Galandrin, Ségolène, Shridhar, Naveen, Hesse, Michael, Grundmann, Manuel, Merten, Nicole, Charpentier, Thomas H., Martz, Matthew, Butcher, Adrian J., Slodczyk, Tanja, Armando, Sylvain, Effern, Maike, Namkung, Yoon, Jenkins, Laura, Horn, Velten, Stößel, Anne, Dargatz, Harald, Tietze, Daniel, Imhof, Diana, Galés, Céline, Drewke, Christel, Müller, Christa E., Hölzel, Michael, Milligan, Graeme, Tobin, Andrew B., Gomeza, Jesús, Dohlman, Henrik G., Sondek, John, Harden, T. Kendall, Bouvier, Michel, Laporte, Stéphane A., Aoki, Junken, Fleischmann, Bernd K., Mohr, Klaus, König, Gabriele M., Tüting, Thomas, Kostenis, Evi

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Angiotensin II type 1 receptor variants alter endosomal receptor–β-arrestin complex stability and MAPK activation von Cao, Yubo, Kumar, Sahil, Namkung, Yoon, Gagnon, Laurence, Cho, Aaron, Laporte, Stéphane A.

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Molecular insights into intrinsic transducer-coupling bias in the CXCR4-CXCR7 system von Sarma, Parishmita, Carino, Carlo Marion C., Seetharama, Deeksha, Pandey, Shubhi, Dwivedi-Agnihotri, Hemlata, Rui, Xue, Cao, Yubo, Kawakami, Kouki, Kumari, Poonam, Chen, Yu-Chih, Luker, Kathryn E., Yadav, Prem N., Luker, Gary D., Laporte, Stéphane A., Chen, Xin, Inoue, Asuka, Shukla, Arun K.

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Allosteric modulation of GPCR-induced β-arrestin trafficking and signaling by a synthetic intrabody von Baidya, Mithu, Chaturvedi, Madhu, Dwivedi-Agnihotri, Hemlata, Ranjan, Ashutosh, Devost, Dominic, Namkung, Yoon, Stepniewski, Tomasz Maciej, Pandey, Shubhi, Baruah, Minakshi, Panigrahi, Bhanupriya, Sarma, Parishmita, Yadav, Manish K., Maharana, Jagannath, Banerjee, Ramanuj, Kawakami, Kouki, Inoue, Asuka, Selent, Jana, Laporte, Stéphane A., Hébert, Terence E., Shukla, Arun K.

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Phosphate‐Rich Biomimetic Peptides Shed Light on High‐Affinity Hyperphosphorylated Uranyl Binding Sites in Phosphoproteins von Laporte, Fanny A., Lebrun, Colette, Vidaud, Claude, Delangle, Pascale

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Allosteric and biased g protein-coupled receptor signaling regulation: potentials for new therapeutics von Khoury, Etienne, Clément, Stéphanie, Laporte, Stéphane A

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Differential β-arrestin-dependent conformational signaling and cellular responses revealed by angiotensin analogs von Zimmerman, Brandon, Beautrait, Alexandre, Aguila, Benjamin, Charles, Ricardo, Escher, Emanuel, Claing, Audrey, Bouvier, Michel, Laporte, Stéphane A

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Genetic code expansion and photocross-linking identify different β-arrestin binding modes to the angiotensin II type 1 receptor von Gagnon, Laurence, Cao, Yubo, Cho, Aaron, Sedki, Dana, Huber, Thomas, Sakmar, Thomas P., Laporte, Stéphane A.

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β-Arrestin 2: A Receptor-Regulated MAPK Scaffold for the Activation of JNK3 von McDonald, Patricia H., Chow, Chi-Wing, Miller, William E., Laporte, Stéphane A., Field, Michael E., Lin, Fang-Tsyr, Davis, Roger J., Lefkowitz, Robert J.

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FZD5 is a Gαq-coupled receptor that exhibits the functional hallmarks of prototypical GPCRs von Wright, Shane C, Cañizal Maria Consuelo Alonso, Benkel Tobias, Simon, Katharina, Le Gouill Christian, Matricon Pierre, Yoon, Namkung, Lukasheva Viktoria, König, Gabriele M, Laporte, Stéphane A, Carlsson Jens, Kostenis Evi, Bouvier, Michel, Schulte, Gunnar, Hoffmann, Carsten

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Discovery of a dual Ras and ARF6 inhibitor from a GPCR endocytosis screen von Giubilaro, Jenna, Schuetz, Doris A., Stepniewski, Tomasz M., Namkung, Yoon, Khoury, Etienne, Lara-Márquez, Mónica, Campbell, Shirley, Beautrait, Alexandre, Armando, Sylvain, Radresa, Olivier, Duchaine, Jean, Lamarche-Vane, Nathalie, Claing, Audrey, Selent, Jana, Bouvier, Michel, Marinier, Anne, Laporte, Stéphane A.

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Structure-toxicity relationships of saturated and unsaturated free fatty acids for elucidating the lipotoxic effects in human EndoC-βH1 beta-cells von Plötz, T., von Hanstein, A.S., Krümmel, B., Laporte, A., Mehmeti, I., Lenzen, S.

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Prostaglandin F2α and angiotensin II type 1 receptors exhibit differential cognate G protein coupling regulation von Sedki, Dana, Cho, Aaron, Cao, Yubo, Nikolajev, Ljiljana, Atmuri, N. D. Prasad, Lubell, William D., Laporte, Stéphane A.

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β-Arrestin-mediated Angiotensin II Signaling Controls the Activation of ARF6 Protein and Endocytosis in Migration of Vascular Smooth Muscle Cells von Charles, Ricardo, Namkung, Yoon, Cotton, Mathieu, Laporte, Stéphane A., Claing, Audrey

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