Recent developments and applications of clickable photoprobes in medicinal chemistry and chemical biology von Lapinsky, David J, Johnson, Douglas S

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Tandem photoaffinity labeling–bioorthogonal conjugation in medicinal chemistry von Lapinsky, David J.

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Clickable photoaffinity ligands for the human serotonin transporter based on the selective serotonin reuptake inhibitor (S)-citalopram von Yarravarapu, Nageswari, Geffert, Laura, Surratt, Christopher K., Cascio, Michael, Lapinsky, David J.

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Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 5 Based on Select Acetylenic Negative Allosteric Modulators von Gregory, Karen J, Velagaleti, Ranganadh, Thal, David M, Brady, Ryan M, Christopoulos, Arthur, Conn, P. Jeffrey, Lapinsky, David J

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Structural studies of the human α1 glycine receptor via site-specific chemical cross-linking coupled with mass spectrometry von Veeramachaneni, Rathna J., Donelan, Chelsee A., Tomcho, Kayce A., Aggarwal, Shaili, Lapinsky, David J., Cascio, Michael

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Appendage- and Scaffold-Diverse Electrophilic and Photoreactive Probes for Integrated Phenotypic Screening–Target Identification Campaigns via a Minimalist Bifunctional Isocyanide... von Jackson, Paul A., Kisty, Eleni, Pradhan, Vandan, Swank, Christopher, Bohrer, Luke, Nolan, Tammy L., Weerapana, Eranthie, Lapinsky, David J.

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Appendage and Scaffold Diverse Fully Functionalized Small-Molecule Probes via a Minimalist Terminal Alkyne-Aliphatic Diazirine Isocyanide von Jackson, Paul, Lapinsky, David J

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Differential contribution of metabotropic glutamate receptor 5 common allosteric binding site residues to biased allosteric agonism von Sengmany, Kathy, Hellyer, Shane D., Christopoulos, Arthur, Lapinsky, David J., Leach, Katie, Gregory, Karen J.

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Development of Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 2 Based on Two Positive Allosteric Modulator Chemotypes von Hellyer, Shane D, Aggarwal, Shaili, Chen, Amy N Y, Leach, Katie, Lapinsky, David J, Gregory, Karen J

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Novel Azido-Iodo Photoaffinity Ligands for the Human Serotonin Transporter Based on the Selective Serotonin Reuptake Inhibitor (S)‑Citalopram von Kumar, Vivek, Yarravarapu, Nageswari, Lapinsky, David J., Perley, Danielle, Felts, Bruce, Tomlinson, Michael J., Vaughan, Roxanne A., Henry, L. Keith, Lever, John R., Newman, Amy Hauck

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Bupropion Binds to Two Sites in the Torpedo Nicotinic Acetylcholine Receptor Transmembrane Domain: A Photoaffinity Labeling Study with the Bupropion Analogue [125I]-SADU-3-72 von Pandhare, Akash, Hamouda, Ayman K, Staggs, Brandon, Aggarwal, Shaili, Duddempudi, Phaneendra K, Lever, John R, Lapinsky, David J, Jansen, Michaela, Cohen, Jonathan B, Blanton, Michael P

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Structural and functional interaction of (±)-2-(N-tert-butylamino)-3′-iodo-4′-azidopropiophenone, a photoreactive bupropion derivative, with nicotinic acetylcholine receptors von Arias, Hugo R., Feuerbach, Dominik, Targowska-Duda, Katarzyna M., Aggarwal, Shaili, Lapinsky, David J., Jozwiak, Krzysztof

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Aziridine–allylsilane-mediated synthesis of exocyclic γ-amino olefins and azabicyclo[ x. y.1]-systems von Lapinsky, David J, Bergmeier, Stephen C

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Structure–activity studies with ring E analogues of methyllycaconitine on bovine adrenal α3β4 nicotinic receptors von Bryant, Darrell L, Free, R.Benjamin, Thomasy, Sara M, Lapinsky, David J, Ismail, Khadiga A, McKay, Susan B, Bergmeier, Stephen C, McKay, Dennis B

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Ring E analogs of methyllycaconitine (MLA) as novel nicotinic antagonists von Bergmeier, Stephen C., Lapinsky, David J., Free, R.Benjamin, McKay, Dennis B

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(±)-2-(N-tert-Butylamino)-3′-[125I]-iodo-4′-azidopropiophenone: A dopamine transporter and nicotinic acetylcholine receptor photoaffinity ligand based on bupropion (Wellbutrin, Zyb... von Lapinsky, David J., Aggarwal, Shaili, Nolan, Tammy L., Surratt, Christopher K., Lever, John R., Acharya, Rejwi, Vaughan, Roxanne A., Pandhare, Akash, Blanton, Michael P.

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A Suzuki cross-coupling route to substituted aziridines von Lapinsky, David J, Bergmeier, Stephen C

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Azido-iodo-N-benzyl derivatives of threo-methylphenidate (Ritalin, Concerta): Rational design, synthesis, pharmacological evaluation, and dopamine transporter photoaffinity labelin... von Lapinsky, David J., Velagaleti, Ranganadh, Yarravarapu, Nageswari, Liu, Yi, Huang, Yurong, Surratt, Christopher K., Lever, John R., Foster, James D., Acharya, Rejwi, Vaughan, Roxanne A., Deutsch, Howard M.

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Substitution effects in intramolecular aziridine–allylsilane cyclizations von Lapinsky, David J., Pulipaka, Aravinda B., Bergmeier, Stephen C.

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Inner ear damage in children due to noise exposure from toy cap pistols and firecrackers: a retrospective review of 53 cases von Segal, S, Eviatar, E, Lapinsky, J, Shlamkovitch, N, Kessler, A

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