Enzymatic Late‐Stage Oxidation of Lead Compounds with Solubilizing Biomimetic Docking/Protecting groups von Vickers, Clare, Backfisch, Gisela, Oellien, Frank, Piel, Isabel, Lange, Udo E. W.

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Combining Machine Learning and Molecular Dynamics to Predict P‑Glycoprotein Substrates von Esposito, Carmen, Wang, Shuzhe, Lange, Udo E. W, Oellien, Frank, Riniker, Sereina

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Solid-phase synthesis of 2,3,5-trisubstituted 4H-imidazolones von Lange, Udo E.W

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De Novo Design, Synthesis, and Biological Evaluation of 3,4-Disubstituted Pyrrolidine Sulfonamides as Potent and Selective Glycine Transporter 1 Competitive Inhibitors von Wang, Ying, Zhao, Hongyu, Brewer, Jason T, Li, Huanqiu, Lao, Yanbin, Amberg, Willi, Behl, Berthold, Akritopoulou-Zanze, Irini, Dietrich, Justin, Lange, Udo E. W, Pohlki, Frauke, Hoft, Carolin, Hornberger, Wilfried, Djuric, Stevan W, Sydor, Jens, Mezler, Mario, Relo, Ana Lucia, Vasudevan, Anil

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Emerging technologies for metabolite generation and structural diversification von Cusack, Kevin P., Koolman, Hannes F., Lange, Udo E.W., Peltier, Hillary M., Piel, Isabel, Vasudevan, Anil

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Discovery of Novel Aminotetralines and Aminochromanes as Selective and Competitive Glycine Transporter 1 (GlyT1) Inhibitors von Amberg, Willi, Lange, Udo E. W, Ochse, Michael, Pohlki, Frauke, Behl, Berthold, Relo, Ana Lucia, Hornberger, Wilfried, Hoft, Carolin, Mezler, Mario, Sydor, Jens, Wang, Ying, Zhao, Hongyu, Brewer, Jason T, Dietrich, Justin, Li, Huanqiu, Akritopoulou-Zanze, Irini, Lao, Yanbin, Hannick, Steven M, Ku, Yi-Yin, Vasudevan, Anil

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A new mild method for the synthesis of amidines von Lange, Udo E.W., Schäfer, Bernd, Baucke, Dorit, Buschmann, Ernst, Mack, Helmut

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Synthesis and SAR of N-substituted dibenzazepinone derivatives as novel potent and selective αVβ3 antagonists von KLING, Andreas, BACKFISCH, Gisela, SEITZ, Werner, SUBKOWSKI, Thomas, DELZER, Jürgen, GENESTE, Hervé, GRAEF, Claudia, HOLZENKAMP, Uta, HORNBERGER, Wilfried, LANGE, Udo E. W, LAUTERBACH, Arnulf, MACK, Helmut

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d-Phe-Pro-Arg type thrombin inhibitors: unexpected selectivity by modification of the P1 moiety von Lange, Udo E.W, Baucke, Dorit, Hornberger, Wilfried, Mack, Helmut, Seitz, Werner, Höffken, H.Wolfgang

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Highly potent and selective αvβ3-receptor antagonists: Solid-phase synthesis and SAR of 1-substituted 4-amino-1H-pyrimidin-2-ones von ZECHEL, Christian, BACKFISCH, Gisela, SUBKOWSKI, Thomas, DELZER, Jürgen, GENESTE, Hervé, GRAEF, Claudia, HORNBERGER, Wilfried, KLING, Andreas, LANGE, Udo E. W, LAUTERBACH, Arnulf, SEITZ, Werner

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Solid-Phase synthesis of endothelin receptor antagonists von Lange, Udo E.W, Braje, Wilfried M, Amberg, Willi, Kettschau, Georg

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Highly Enantioselective Imine Hydrosilylation Using (S,S)-Ethylenebis(η5-tetrahydroindenyl)titanium Difluoride von Verdaguer, Xavier, Lange, Udo E. W., Reding, Matthew T., Buchwald, Stephen L.

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Amine Additives Greatly Expand the Scope of Asymmetric Hydrosilylation of Imines von Verdaguer, Xavier, Lange, Udo E. W., Buchwald, Stephen L.

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Orally active thrombin inhibitors. Part 2: Optimization of the P2-moiety von Lange, Udo E.W., Baucke, Dorit, Hornberger, Wilfried, Mack, Helmut, Seitz, Werner, Höffken, H. Wolfgang

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Solid-phase synthesis of 2,3,5-trisubstituted 4 H-imidazolones von Lange, Udo E.W

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Design and synthesis of 1,5- and 2,5-substituted tetrahydrobenzazepinones as novel potent and selective integrin αvβ3antagonists von KLING, Andreas, BACKFISCH, Gisela, DELZER, Jürgen, GENESTE, Herve, GRAEF, Claudia, HORNBERGER, Wilfried, LANGE, Udo E. W, LAUTERBACH, Arnulf, SEITZ, Werner, SUBKOWSKI, Thomas

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Orally active thrombin inhibitors. Part 1: Optimization of the P1-moiety von Mack, Helmut, Baucke, Dorit, Hornberger, Wilfried, Lange, Udo E.W., Seitz, Werner, Höffken, H. Wolfgang

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Synthesis and SAR of highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drugs von KLING, Andreas, LANGE, Udo E. W, UNGER, Liliane, WICKE, Karsten, SCHELLHAAS, Kurt, STEINER, Gerd, MACK, Helmut, BAKKER, Margot H. M, DRESCHER, Karla U, HORNBERGER, Wilfried, HUTCHINS, Charles W, MÖLLER, Achim, MÜLLER, Reinhold, SCHMIDT, Martin

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Technical Scale Synthesis of a New and Highly Potent Thrombin Inhibitor von Bernard, Harald, Bülow, Gerd, Lange, Udo E., Mack, Helmut, Pfeiffer, Thomas, Schäfer, Bernd, Seitz, Werner, Zierke, Thomas

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Solid-phase synthesis of thrombin inhibitors von Lange, Udo E.W., Zechel, Christian

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