Androgen receptor-binding sites are highly mutated in prostate cancer von Morova, Tunç, McNeill, Daniel R., Lallous, Nada, Gönen, Mehmet, Dalal, Kush, Wilson, David M., Gürsoy, Attila, Keskin, Özlem, Lack, Nathan A.

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Moving Towards Precision Urologic Oncology: Targeting Enzalutamide-resistant Prostate Cancer and Mutated Forms of the Androgen Receptor Using the Novel Inhibitor Darolutamide (ODM-... von Borgmann, Hendrik, Lallous, Nada, Ozistanbullu, Deniz, Beraldi, Eliana, Paul, Naman, Dalal, Kush, Fazli, Ladan, Haferkamp, Axel, Lejeune, Pascale, Cherkasov, Artem, Gleave, Martin E.

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Ivermectin inhibits HSP27 and potentiates efficacy of oncogene targeting in tumor models von Nappi, Lucia, Aguda, Adeleke H, Nakouzi, Nader Al, Lelj-Garolla, Barbara, Beraldi, Eliana, Lallous, Nada, Thi, Marisa, Moore, Susan, Fazli, Ladan, Battsogt, Dulguun, Stief, Sophie, Ban, Fuqiang, Nguyen, Nham T, Saxena, Neetu, Dueva, Evgenia, Zhang, Fan, Yamazaki, Takeshi, Zoubeidi, Amina, Cherkasov, Artem, Brayer, Gary D, Gleave, Martin

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Characterization of novel small molecule inhibitors of estrogen receptor-activation function 2 (ER-AF2) von Foo, Jane, Gentile, Francesco, Massah, Shabnam, Morin, Helene, Singh, Kriti, Lee, Joseph, Smith, Jason, Ban, Fuqiang, LeBlanc, Eric, Young, Robert, Strynadka, Natalie, Lallous, Nada, Cherkasov, Artem

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Computer-Aided Discovery of Small Molecules Targeting the RNA Splicing Activity of hnRNP A1 in Castration-Resistant Prostate Cancer von Carabet, Lavinia A, Leblanc, Eric, Lallous, Nada, Morin, Helene, Ghaidi, Fariba, Lee, Joseph, Rennie, Paul S, Cherkasov, Artem

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Computer-aided drug discovery of Myc-Max inhibitors as potential therapeutics for prostate cancer von Carabet, Lavinia A., Lallous, Nada, Leblanc, Eric, Ban, Fuqiang, Morin, Helene, Lawn, Sam, Ghaidi, Fariba, Lee, Joseph, Mills, Ian G., Gleave, Martin E., Rennie, Paul S., Cherkasov, Artem

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Discovery of New Catalytic Topoisomerase II Inhibitors for Anticancer Therapeutics von Matias-Barrios, Victor M, Radaeva, Mariia, Song, Yi, Alperstein, Zaccary, Lee, Ahn R, Schmitt, Veronika, Lee, Joseph, Ban, Fuqiang, Xie, Ning, Qi, Jianfei, Lallous, Nada, Gleave, Martin E, Cherkasov, Artem, Dong, Xuesen

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Targeting alternative sites on the androgen receptor to treat castration-resistant prostate cancer von Lallous, Nada, Dalal, Kush, Cherkasov, Artem, Rennie, Paul S

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Reformation of the chondroitin sulfate glycocalyx enables progression of AR-independent prostate cancer von Al-Nakouzi, Nader, Wang, Chris Kedong, Oo, Htoo Zarni, Nelepcu, Irina, Lallous, Nada, Spliid, Charlotte B., Khazamipour, Nastaran, Lo, Joey, Truong, Sarah, Collins, Colin, Hui, Desmond, Esfandnia, Shaghayegh, Adomat, Hans, Clausen, Thomas Mandel, Gustavsson, Tobias, Choudhary, Swati, Dagil, Robert, Corey, Eva, Wang, Yuzhuo, Chauchereau, Anne, Fazli, Ladan, Esko, Jeffrey D., Salanti, Ali, Nelson, Peter S., Gleave, Martin E., Daugaard, Mads

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Bypassing Drug Resistance Mechanisms of Prostate Cancer with Small Molecules that Target Androgen Receptor-Chromatin Interactions von Dalal, Kush, Che, Meixia, Que, Nanette S, Sharma, Aishwariya, Yang, Rendong, Lallous, Nada, Borgmann, Hendrik, Ozistanbullu, Deniz, Tse, Ronnie, Ban, Fuqiang, Li, Huifang, Tam, Kevin J, Roshan-Moniri, Mani, LeBlanc, Eric, Gleave, Martin E, Gewirth, Daniel T, Dehm, Scott M, Cherkasov, Artem, Rennie, Paul S

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Developing novel Lin28 inhibitors by computer aided drug design von Matias-Barrios, Victor M., Radaeva, Mariia, Rosellinny, Graciella, Jia, Qiongqiong, Xie, Ning, Villanueva, Monica, Ibrahim, Hanadi, Smith, Jason, Gleave, Martin, Lallous, Nada, Straus, Suzana K., Cherkasov, Artem, Dong, Xuesen

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Structure-Based Study to Overcome Cross-Reactivity of Novel Androgen Receptor Inhibitors von Radaeva, Mariia, Li, Huifang, LeBlanc, Eric, Dalal, Kush, Ban, Fuqiang, Ciesielski, Fabrice, Chow, Bonny, Morin, Helene, Awrey, Shannon, Singh, Kriti, Rennie, Paul S., Lallous, Nada, Cherkasov, Artem

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The PHD finger of human UHRF1 reveals a new subgroup of unmethylated histone H3 tail readers von Lallous, Nada, Legrand, Pierre, McEwen, Alastair G, Ramón-Maiques, Santiago, Samama, Jean-Pierre, Birck, Catherine

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Drug-Discovery Pipeline for Novel Inhibitors of the Androgen Receptor von Dalal, Kush, Munuganti, Ravi, Morin, Hélène, Lallous, Nada, Rennie, Paul S., Cherkasov, Artem

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Androgen receptor plasticity and its implications for prostate cancer therapy von Snow, Oliver, Lallous, Nada, Singh, Kriti, Lack, Nathan, Rennie, Paul, Cherkasov, Artem

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Deep Learning Modeling of Androgen Receptor Responses to Prostate Cancer Therapies von Snow, Oliver, Lallous, Nada, Ester, Martin, Cherkasov, Artem

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PurificationDB: database of purification conditions for proteins von Garland, Olivia, Radaeva, Mariia, Pandey, Mohit, Cherkasov, Artem, Lallous, Nada

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Functional analysis of androgen receptor mutations that confer anti-androgen resistance identified in circulating cell-free DNA from prostate cancer patients von Lallous, Nada, Volik, Stanislav V, Awrey, Shannon, Leblanc, Eric, Tse, Ronnie, Murillo, Josef, Singh, Kriti, Azad, Arun A, Wyatt, Alexander W, LeBihan, Stephane, Chi, Kim N, Gleave, Martin E, Rennie, Paul S, Collins, Colin C, Cherkasov, Artem

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Novel Inhibitors of androgen receptor's DNA binding domain identified using an ultra-large virtual screening von Radaeva, Mariia, Morin, Helene, Pandey, Mohit, Ban, Fuqiang, Guo, Maria, LeBlanc, Eric, Lallous, Nada, Cherkasov, Artem

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Characterization of androgen receptor properties in mediating transcriptional biomolecular condensates in prostate cancer von Pinette, Nicholas C., Massah, Shabnam, Huang, Tian Hao, Kochkina, Sofia, Bembridge, Alex, Foo, Jane, Guo, Maria, Ibrahim, Hanadi, Cherkasov, Artem, Gsponer, Joerg, Lallous, Nada

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