Orally Active MMP-1 Sparing α-Tetrahydropyranyl and α-Piperidinyl Sulfone Matrix Metalloproteinase (MMP) Inhibitors with Efficacy in Cancer, Arthritis, and Cardiovascular Disease von Becker, Daniel P, Barta, Thomas E, Bedell, Louis J, Boehm, Terri L, Bond, Brian R, Carroll, Jeffery, Carron, Chris P, DeCrescenzo, Gary A, Easton, Alan M, Freskos, John N, Funckes-Shippy, Chris L, Heron, Marcia, Hockerman, Susan, Howard, Carol Pearcy, Kiefer, James R, Li, Madeleine H, Mathis, Karl J, McDonald, Joseph J, Mehta, Pramod P, Munie, Grace E, Sunyer, Teresa, Swearingen, Craig A, Villamil, Clara I, Welsch, Dean, Williams, Jennifer M, Yu, Ying, Yao, Jun

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Synthesis and Structure−Activity Relationships of β- and α-Piperidine Sulfone Hydroxamic Acid Matrix Metalloproteinase Inhibitors with Oral Antitumor Efficacy von Becker, Daniel P, Villamil, Clara I, Barta, Thomas E, Bedell, Louis J, Boehm, Terri L, DeCrescenzo, Gary A, Freskos, John N, Getman, Daniel P, Hockerman, Susan, Heintz, Robert, Howard, Susan Carol, Li, Madeleine H, McDonald, Joseph J, Carron, Chris P, Funckes-Shippy, Chris L, Mehta, Pramod P, Munie, Grace E, Swearingen, Craig A

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MMP-13 selective alpha-sulfone hydroxamates: Identification of selective P1′ amides von Fobian, Yvette M., Freskos, John N., Barta, Thomas E., Bedell, Louis J., Heintz, Robert, Kassab, Darren J., Kiefer, James R., Mischke, Brent V., Molyneaux, John M., Mullins, Patrick, Munie, Grace E., Becker, Daniel P.

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MMP-13 selective α-sulfone hydroxamates: A survey of P1′ heterocyclic amide isosteres von Barta, Thomas E., Becker, Daniel P., Bedell, Louis J., Easton, Alan M., Hockerman, Susan L., Kiefer, James, Munie, Grace E., Mathis, Karl J., Li, Madeleine H., Rico, Joseph G., Villamil, Clara I., Williams, Jennifer M.

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Synthesis and activity of selective MMP inhibitors with an aryl backbone von E. Barta, Thomas, P. Becker, Daniel, J. Bedell, Louis, A. De Crescenzo, Gary, J. McDonald, Joseph, E. Munie, Grace, Rao, Shashi, Shieh, Huey-Sheng, Stegeman, Roderick, M. Stevens, Anna, I. Villamil, Clara

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Selective, orally active MMP inhibitors with an aryl backbone von Barta, Thomas E., Becker, Daniel P., Bedell, Louis J., De Crescenzo, Gary A., McDonald, Joseph J., Mehta, Pramod, Munie, Grace E., Villamil, Clara I.

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Effects of SC-56525, a Potent, Orally Active Renin Inhibitor, in Salt-Depleted and Renal Hypertensive Dogs von McMahon, Ellen G, Yang, Po-Chang, Babler, Maribeth A, Bittner, Stephen E, Suleymanov, Osman D, Cain-Janicki, Kimberly J, Bedell, Louis J, Hanson, Gunnar J, Cook, Chyung S

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Design of MHC class II (DR4) ligands using conformationally restricted imino acids at p3 and p5 von Hanson, Gunnar J., Vuletich, Jennifer L., Bedell, Louis J., Bono, Christine P., Howard, Susan C., Welply, Joseph K., Woulfe, Susan L., Zacheis, Michelle L.

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HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS von LOUIS J. BEDELL

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AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR von CAROL P HOWARD, DEBORAH A. MISCHKE, THERESA R FLETCHER, GUNNAR J. HANSON, THOMAS E. BARTA, LOUIS J BEDELL, JOSEPH G RICO, NATHAN W STEHLE, MADELEINE H LI, JOHN N. FRESKOS, DANIEL P. GETMAN, DANIEL P. BECKER, PATRICK B MULLINS, SUSAN L. HOCKERMAN, JOSEPH J. MCDONALD, CLARA I. VILLAMIL, JEFFREY N CARROLL, GARY A. DECRESCENZO, STEPHEN A. KOLODZIEJ, TERRI L. BOEHM

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ChemInform Abstract: Selective, Orally Active MMP Inhibitors with an Aryl Backbone von Barta, Thomas E., Becker, Daniel P., Bedell, Louis J., De Crescenzo, Gary A., McDonald, Joseph J., Mehta, Pramod, Munie, Grace E., Villamil, Clara I.

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PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS von CHEN, YIYUAN, BEDELL, LOUIS, J, BECKER, DANIEL, P, BOEHM, TERRI, L, BROWN, DAVID, L, BARTA, THOMAS, E, CARROLL, JEFFERY, N

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Aromatic sulfone hydroxamates and their use as protease inhibitors von BEDELL Louis J, BOEHM Terri L, CARROLL Jeffrey, BARTA Thomas E, DECRESCENZO Gary A, BECKER Daniel P, FOBIAN Yvette, Marlene

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PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS von CHEN, YIYUAN, BEDELL, LOUIS, J, BECKER, DANIEL, P, BOEHM, TERRI, L, BROWN, DAVID, L, BARTA, THOMAS, E, CARROLL, JEFFERY, N

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Sulfonyl aryl or heteroaryl hydroxamic acid compounds von SHASHIDHAR RAO N, VILLAMIL CLARA I, DECRESCENZO GARY A, MISCHKE BRENT V, BEDELL LOUIS J, BARTA THOMAS E, FRESKOS JOHN N, BECKER DANIEL P, GETMAN DANIEL P, MCDONALD JOSEPH J

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Sulfonyl aryl or heteroaryl hydroxamic acid compounds von Bedell, Louis J, McDonald, Joseph J, Barta, Thomas E, Becker, Daniel P, Shashidhar, Rao N, Freskos, John N, Mischke, Brent V, Getman, Daniel P, DeCrescenzo, Gary A, Villamil, Clara I

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Aromatic sulfone hydroxamates and their use as protease inhibitors von FRESKOS JOHN N.,FOBIAN YVETTE M.,BARTA THOMAS E.,BECKER DANIEL P.,BEDELL LOUIS J.,BOEHM TERRI L.,HOCKERMAN SUSAN L.,KASSAB DARREN J.,KOLODZIEJ STEVE A.,MCDONALD JOSEPH,NORTON MONICA B.,RICO JOSEPH G, JUAN JANE

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COMPOSTOS A BASE DE ACIDO HETEROARILO HIDROXAMICO OU ACIDO SULFONILOARILO BIVALENTE HIDROXAMICO von JOHN N. FRESKOS, SHASHIDHAR N. RAO, DANIEL P. BECKER, JOSEPH J. MCDONALD, BRENT V. MISCHKE, THOMAS E. BARTA, LOUIS J. BEDELL

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Divalente sulfonyl-aryl eller heteroarylhydroxamsyreforbindelser von BEDELL, LOUIS, J, MISCHKE, BRENT, V, BECKER, DANIEL, P, RAO, SHASHIDHAR, N, FRESKOS, JOHN, N, BARTA, THOMAS, E, MCDONALD, JOSEPH, J

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DIVALENTE SULFONYL-ARYL-ODER HETEROARYL HYDROXAMSÄUREVERBINDUNGEN von BEDELL, LOUIS, J, MISCHKE, BRENT, V, BECKER, DANIEL, P, RAO, SHASHIDHAR, N, FRESKOS, JOHN, N, BARTA, THOMAS, E, MCDONALD, JOSEPH, J

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