Enantiotropically-related polymorphs of {4-(4-chloro-3-fluorophenyl)-2-[4-(methyloxy)phenyl]-1,3-thiazol-5-yl} acetic acid: Crystal structures and multinuclear solid-state NMR von Vogt, Frederick G., Katrincic, Lee M., Long, Stacey T., Mueller, Ronald L., Carlton, Robert A., Sun, Yan T., Johnson, Matthew N., Copley, Royston C.B., Light, Mark E.

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Design of Potent, Selective, and Orally Bioavailable Inhibitors of Cysteine Protease Cathepsin K von Tavares, Francis X, Boncek, Virginia, Deaton, David N, Hassell, Anne M, Long, Stacey T, Miller, Aaron B, Payne, Alan A, Miller, Larry R, Shewchuk, Lisa M, Wells-Knecht, Kevin, Willard, Derril H, Wright, Lois L, Zhou, Hui-Qiang

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Acyclic, orally bioavailable ketone-based cathepsin K inhibitors von Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Samano, Vicente, Tavares, Francis X., Wells-Knecht, Kevin J., Wright, Lois L., Zhou, Hui-Qiang Q.

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Design of small molecule ketoamide-based inhibitors of cathepsin K von Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Larry R., Payne, J.Alan, Wells-Knecht, Kevin J., Wright, Lois L.

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A structural screening approach to ketoamide-based inhibitors of cathepsin K von Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Wells-Knecht, Kevin J., Wright, Lois L.

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Semicarbazone-based inhibitors of cathepsin K, are they prodrugs for aldehyde inhibitors? von Adkison, Kim K., Barrett, David G., Deaton, David N., Gampe, Robert T., Hassell, Anne M., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.

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Orally bioavailable small molecule ketoamide-based inhibitors of cathepsin K von Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., Miller, Larry R., Tavares, Francis X., Wells-Knecht, Kevin J., Wright, Lois L., Zhou, Hui-Qiang Q.

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Novel, potent P2–P3 pyrrolidine derivatives of ketoamide-based cathepsin K inhibitors von Barrett, David G., Catalano, John G., Deaton, David N., Hassell, Anne M., Long, Stacey T., Miller, Aaron B., Miller, Larry R., Ray, John A., Samano, Vicente, Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.

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P2-P3 conformationally constrained ketoamide-based inhibitors of cathepsin K von BARRETT, David G, BONCEK, Virginia M, PAYNE, J. Alan, RAY, John A, SAMANO, Vicente, SHEWCHUK, Lisa M, TAVARES, Francis X, WELLS-KNECHT, Kevin J, WILLARD, Derril H, WRIGHT, Lois L, ZHOU, Hui-Qiang Q, CATALANO, John G, DEATON, David N, HASSELL, Anne M, JURGENSEN, Cynthia H, LONG, Stacey T, MCFADYEN, Robert B, MILLER, Aaron B, MILLER, Larry R

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Potent and selective P2-P3 ketoamide inhibitors of cathepsin K with good pharmacokinetic properties via favorable P1', P1, and/or P3 substitutions von BARRETT, David G, CATALANO, John G, WRIGHT, Lois L, DEATON, David N, HASSELL, Anne M, LONG, Stacey T, MILLER, Aaron B, MILLER, Larry R, SHEWCHUK, Lisa M, WELLS-KNECHT, Kevin J, WILLARD, Derril H

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Crystal Structure Prediction for Eniluracil von Sacchetti, Mark, Varlashkin, Peter G., Long, Stacey T., Lancaster, Robert W.

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Excipient compatibility as assessed by isothermal microcalorimetry von Phipps, Mark A., Winnike, Richard A., Long, Stacey T., Viscomi, Frank

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PHARMACEUTICS, PREFORMULATION AND DRUG DELIVERY Enantiotropically-Related Polymorphs of {4-(4-Chloro-3-Fluorophenyl)-2-[4-(Methyloxy)Phenyl]-1, 3-Thiazol-S-yl} Acetic Acid : Crysta... von VOGT, Frederick G, KATRINCIC, Lee M, LONG, Stacey T, MUELLER, Ronald L, CARLTON, Robert A, SUN, Yan T, JOHNSON, Matthew N, COPLEY, Royston C. B, LIGHT, Mark E

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P 2–P 3 conformationally constrained ketoamide-based inhibitors of cathepsin K von Barrett, David G., Boncek, Virginia M., Catalano, John G., Deaton, David N., Hassell, Anne M., Jurgensen, Cynthia H., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Ray, John A., Samano, Vicente, Shewchuk, Lisa M., Tavares, Francis X., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L., Zhou, Hui-Qiang Q.

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Potent and selective P 2–P 3 ketoamide inhibitors of cathepsin K with good pharmacokinetic properties via favorable P 1′, P 1, and/or P 3 substitutions von Barrett, David G., Catalano, John G., Deaton, David N., Hassell, Anne M., Long, Stacey T., Miller, Aaron B., Miller, Larry R., Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.

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Novel, potent P super(2)-P super(3) pyrrolidine derivatives of ketoamide-based cathepsin K inhibitors von Barrett, David G, Catalano, John G, Deaton, David N, Hassell, Anne M, Long, Stacey T, Miller, Aaron B, Miller, Larry R, Ray, John A, Samano, Vicente, Shewchuk, Lisa M, Wells-Knecht, Kevin J, Willard, Derril H, Wright, Lois L

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NOVEL CRYSTALLINE FORMS OF AN ANTIVIRAL BENZIMIDAZOLE COMPOUND von LANCASTER ROBERT W, GLOVER BOBBY N, SCHMITT ERIC A, RIZZOLIO MICHELE C, HUANG LIAN-FENG, LONG STACEY T, SICKLES BARRY R

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Orally Bioavailable Small Molecule Ketoamide-Based Inhibitors of Cathepsin K von Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., Miller, Larry R., Tavares, Francis X., Wells-Knecht, Kevin J., Wright, Lois L., Zhou, Hui-Qiang Q.

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Design of Small Molecule Ketoamide-Based Inhibitors of Cathepsin K von Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Larry R., Payne, J. Alan, Wells-Knecht, Kevin J., Wright, Lois L.

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BENTUK KRISTALIN BARU DARI SENYAWA BENZIMIDAZOL ANTIVIRAL von ROBERT W. LANCASTER, LIAN FENG HUANG, BORRY H. CARTER, MICHELE C. RIZZOLIO, ERIC A. SCHMITT, BOBBY N. GLOVER, BARRY R. SICKLESS, STACEY T. LONG

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