Apo2L/TRAIL and the Death Receptor 5 Agonist Antibody AMG 655 Cooperate to Promote Receptor Clustering and Antitumor Activity von Graves, Jonathan D., Kordich, Jennifer J., Huang, Tzu-Hsuan, Piasecki, Julia, Bush, Tammy L., Sullivan, Timothy, Foltz, Ian N., Chang, Wesley, Douangpanya, Heather, Dang, Thu, O’Neill, Jason W., Mallari, Rommel, Zhao, Xiaoning, Branstetter, Daniel G., Rossi, John M., Long, Alexander M., Huang, Xin, Holland, Pamela M.

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Structural Basis for the Potent and Selective Inhibition of Casein Kinase 1 Epsilon von Long, Alexander M, Zhao, Huilin, Huang, Xin

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Structure-Based Design of Novel Inhibitors of the MDM2–p53 Interaction von Rew, Yosup, Sun, Daqing, Gonzalez-Lopez De Turiso, Felix, Bartberger, Michael D, Beck, Hilary P, Canon, Jude, Chen, Ada, Chow, David, Deignan, Jeffrey, Fox, Brian M, Gustin, Darin, Huang, Xin, Jiang, Min, Jiao, Xianyun, Jin, Lixia, Kayser, Frank, Kopecky, David J, Li, Yihong, Lo, Mei-Chu, Long, Alexander M, Michelsen, Klaus, Oliner, Jonathan D, Osgood, Tao, Ragains, Mark, Saiki, Anne Y, Schneider, Steve, Toteva, Maria, Yakowec, Peter, Yan, Xuelei, Ye, Qiuping, Yu, Dongyin, Zhao, Xiaoning, Zhou, Jing, Medina, Julio C, Olson, Steven H

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Discovery of 1H‑Pyrazol-3(2H)‑ones as Potent and Selective Inhibitors of Protein Kinase R‑like Endoplasmic Reticulum Kinase (PERK) von Smith, Adrian L, Andrews, Kristin L, Beckmann, Holger, Bellon, Steven F, Beltran, Pedro J, Booker, Shon, Chen, Hao, Chung, Young-Ah, D’Angelo, Noel D, Dao, Jennifer, Dellamaggiore, Kenneth R, Jaeckel, Peter, Kendall, Richard, Labitzke, Katja, Long, Alexander M, Materna-Reichelt, Silvia, Mitchell, Petia, Norman, Mark H, Powers, David, Rose, Mark, Shaffer, Paul L, Wu, Michelle M, Lipford, J. Russell

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Selective and Potent Morpholinone Inhibitors of the MDM2–p53 Protein–Protein Interaction von Gonzalez, Ana Z, Eksterowicz, John, Bartberger, Michael D, Beck, Hilary P, Canon, Jude, Chen, Ada, Chow, David, Duquette, Jason, Fox, Brian M, Fu, Jiasheng, Huang, Xin, Houze, Jonathan B, Jin, Lixia, Li, Yihong, Li, Zhihong, Ling, Yun, Lo, Mei-Chu, Long, Alexander M, McGee, Lawrence R, McIntosh, Joel, McMinn, Dustin L, Oliner, Jonathan D, Osgood, Tao, Rew, Yosup, Saiki, Anne Y, Shaffer, Paul, Wortman, Sarah, Yakowec, Peter, Yan, Xuelei, Ye, Qiuping, Yu, Dongyin, Zhao, Xiaoning, Zhou, Jing, Olson, Steven H, Medina, Julio C, Sun, Daqing

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Ordering of the N‑Terminus of Human MDM2 by Small Molecule Inhibitors von Michelsen, Klaus, Jordan, John B, Lewis, Jeffrey, Long, Alexander M, Yang, Evelyn, Rew, Yosup, Zhou, Jing, Yakowec, Peter, Schnier, Paul D, Huang, Xin, Poppe, Leszek

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Rational Design and Binding Mode Duality of MDM2–p53 Inhibitors von Gonzalez-Lopez de Turiso, Felix, Sun, Daqing, Rew, Yosup, Bartberger, Michael D, Beck, Hilary P, Canon, Jude, Chen, Ada, Chow, David, Correll, Tiffany L, Huang, Xin, Julian, Lisa D, Kayser, Frank, Lo, Mei-Chu, Long, Alexander M, McMinn, Dustin, Oliner, Jonathan D, Osgood, Tao, Powers, Jay P, Saiki, Anne Y, Schneider, Steve, Shaffer, Paul, Xiao, Shou-Hua, Yakowec, Peter, Yan, Xuelei, Ye, Qiuping, Yu, Dongyin, Zhao, Xiaoning, Zhou, Jing, Medina, Julio C, Olson, Steven H

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c-Met Inhibitors with Novel Binding Mode Show Activity against Several Hereditary Papillary Renal Cell Carcinoma-related Mutations von Bellon, Steven F., Kaplan-Lefko, Paula, Yang, Yajing, Zhang, Yihong, Moriguchi, Jodi, Rex, Karen, Johnson, Carol W., Rose, Paul E., Long, Alexander M., O'Connor, Anne B., Gu, Yan, Coxon, Angela, Kim, Tae-Seong, Tasker, Andrew, Burgess, Teresa L., Dussault, Isabelle

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Discovery and Optimization of Triazolopyridazines as Potent and Selective Inhibitors of the c-Met Kinase von Albrecht, Brian K, Harmange, Jean-Christophe, Bauer, David, Berry, Loren, Bode, Christiane, Boezio, Alessandro A, Chen, April, Choquette, Deborah, Dussault, Isabelle, Fridrich, Cary, Hirai, Satoko, Hoffman, Doug, Larrow, Jay F, Kaplan-Lefko, Paula, Lin, Jasmine, Lohman, Julia, Long, Alexander M, Moriguchi, Jodi, O’Connor, Anne, Potashman, Michele H, Reese, Monica, Rex, Karen, Siegmund, Aaron, Shah, Kavita, Shimanovich, Roman, Springer, Stephanie K, Teffera, Yohannes, Yang, Yajing, Zhang, Yihong, Bellon, Steven F

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Crystal structure of a bacteriophage T7 DNA replication complex at 2.2  resolution von Ellenberger, Tom, Doublié, Sylvie, Tabor, Stanley, Long, Alexander M, Richardson, Charles C

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Screening for lysine-specific demethylase-1 inhibitors using a label-free high-throughput mass spectrometry assay von Plant, Matthew, Dineen, Tom, Cheng, Alan, Long, Alexander M., Chen, Hao, Morgenstern, Kurt A.

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Remote Density Measurements of Molten Salts via Neutron Radiography von Long, Alexander M., Parker, S. Scott, Carver, D. Travis, Jackson, J. Matt, Monreal, Marisa J., Newmark, Darcy A., Vogel, Sven C.

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Novel 2,3-Dihydro-1,4-Benzoxazines as Potent and Orally Bioavailable Inhibitors of Tumor-Driven Angiogenesis von La, Daniel S, Belzile, Julie, Bready, James V, Coxon, Angela, DeMelfi, Thomas, Doerr, Nicholas, Estrada, Juan, Flynn, Julie C, Flynn, Shaun R, Graceffa, Russell F, Harriman, Shawn P, Larrow, Jay F, Long, Alexander M, Martin, Matthew W, Morrison, Michael J, Patel, Vinod F, Roveto, Philip M, Wang, Ling, Weiss, Matthew M, Whittington, Douglas A, Teffera, Yohannes, Zhao, Zhiyang, Polverino, Anthony J, Harmange, Jean-Christophe

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Demonstration of neutron time‐of‐flight diffraction with an event‐mode imaging detector von Jäger, Tim T., Losko, Adrian S., Wolfertz, Alexander, Schmidt, Søren, Bertelsen, Mads, Khaplanov, Anton, Agnew, Sean R., Funama, Fumiaki, Morgano, Manuel, Roth, Markus, Gochanour, Jason R., Long, Alexander M., Lutterotti, Luca, Vogel, Sven C.

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Evolution of a Highly Selective and Potent 2-(Pyridin-2-yl)-1,3,5-triazine Tie-2 Kinase Inhibitor von Hodous, Brian L, Geuns-Meyer, Stephanie D, Hughes, Paul E, Albrecht, Brian K, Bellon, Steve, Bready, James, Caenepeel, Sean, Cee, Victor J, Chaffee, Stuart C, Coxon, Angela, Emery, Maurice, Fretland, Jenne, Gallant, Paul, Gu, Yan, Hoffman, Doug, Johnson, Rebecca E, Kendall, Richard, Kim, Joseph L, Long, Alexander M, Morrison, Michael, Olivieri, Philip R, Patel, Vinod F, Polverino, Anthony, Rose, Paul, Tempest, Paul, Wang, Ling, Whittington, Douglas A, Zhao, Huilin

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Small‐angle scattering and dark‐field imaging for validation of a new neutron far‐field interferometer von Wolf, Caitlyn M., Bajcsy, Peter, Chen, Wei-Ren, Dalgliesh, Robert M., Daugherty, M. Cyrus, de Campo, Liliana, Funama, Fumiaki, He, Lilin, Huber, Michael G, Jacobson, David L., Kienzle, Paul, Kim, Youngju, King, Hubert, Klimov, Nikolai N., LaManna, Jacob M., Li, Fankang, Long, Alexander M., Murphy, Ryan, Nagy, Gergely, Robinson, Sarah M., Sathe, Pushkar, Smith, Gregory N., Sokolova, Anna, Vogel, Sven C., Watkins, Erik B., Zhang, Yuxuan, Hussey, Daniel S., Weigandt, Katie M.

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Flexible 3D printed silicones for gamma and neutron radiation shielding von Talley, Samantha J., Robison, Tom, Long, Alexander M., Lee, So Young, Brounstein, Zachary, Lee, Kwan-Soo, Geller, Drew, Lum, Ed, Labouriau, Andrea

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Modulation of Ligand-Gated Glycine Receptors Via Functional Monoclonal Antibodies von Simard, Jeffrey R., Michelsen, Klaus, Wang, Yan, Yang, Chunhua, Youngblood, Beth, Grubinska, Barbara, Taborn, Kristin, Gillie, Daniel J., Cook, Kevin, Chung, Kyu, Long, Alexander M., Hall, Brian E., Shaffer, Paul L., Foti, Robert S., Gingras, Jacinthe

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The Complex, Unique, and Powerful Imaging Instrument for Dynamics (CUPI2D) at the Spallation Neutron Source (invited) von Brügger, Adrian, Bilheux, Hassina Z., Lin, Jiao Y. Y., Nelson, George J., Kiss, Andrew M., Morris, Jonathan, Connolly, Matthew J., Long, Alexander M., Tremsin, Anton S., Strzelec, Andrea, Anderson, Mark H., Agasie, Robert, Finney, Charles E. A., Wissink, Martin L., Hubler, Mija H., Pellenq, Roland J.-M., White, Claire E., Heuser, Brent J., Craft, Aaron E., Harp, Jason M., Tan, Chuting, Morris, Kathryn, Junghans, Ann, Sevanto, Sanna, Warren, Jeffrey M., Esteban Florez, Fernando L., Biris, Alexandru S., Cekanova, Maria, Kardjilov, Nikolay, Schillinger, Burkhard, Frost, Matthew J., Vogel, Sven C.

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Effects of Hydrogen Redistribution at High Temperatures in Yttrium Hydride Moderator Material von Trellue, Holly R., Long, Alexander M., Luther, Erik P., Carver, D. Travis, Mehta, Vedant K.

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