Discovery of 2‑Aminopyrimidines as Potent Agonists for the Bitter Taste Receptor TAS2R14 von Waterloo, Lukas, Hübner, Harald, Fierro, Fabrizio, Pfeiffer, Tara, Brox, Regine, Löber, Stefan, Weikert, Dorothee, Niv, Masha Y., Gmeiner, Peter

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Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back von Di Pizio, Antonella, Waterloo, Lukas A. W., Brox, Regine, Löber, Stefan, Weikert, Dorothee, Behrens, Maik, Gmeiner, Peter, Niv, Masha Y.

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Structure-based development of caged dopamine D2/D3 receptor antagonists von Gienger, Marie, Hübner, Harald, Löber, Stefan, König, Burkhard, Gmeiner, Peter

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The Bitter Taste Receptor TAS2R14 as a Drug Target von Waterloo, Lukas A W, Löber, Stefan, Gmeiner, Peter

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Presynaptic vesicular accumulation is required for antipsychotic efficacy in psychotic-like rats von Uzuneser, Taygun C, Weiss, Eva-Maria, Dahlmanns, Jana, Kalinichenko, Liubov S, Amato, Davide, Kornhuber, Johannes, Alzheimer, Christian, Hellmann, Jan, Kaindl, Jonas, Hübner, Harald, Löber, Stefan, Gmeiner, Peter, Grömer, Teja W, Müller, Christian P

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Discovery of dopamine D4 receptor antagonists with planar chirality von Sanna, Fabrizio, Ortner, Birgit, Hübner, Harald, Löber, Stefan, Tschammer, Nuska, Gmeiner, Peter

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Bioisosteric Replacement Leading to Biologically Active [2.2]Paracyclophanes with Altered Binding Profiles for Aminergic G-Protein-Coupled Receptors von Skultety, Marika, Hübner, Harald, Löber, Stefan, Gmeiner, Peter

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Synthesis and binding profile of haloperidol-based bivalent ligands targeting dopamine D sub(2)-like receptors von Salama, Ismail, Lober, Stefan, Huebner, Harald, Gmeiner, Peter

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Click chemistry on solid support: synthesis of a new REM resin and application for the preparation of tertiary amines von Löber, Stefan, Gmeiner, Peter

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Bivalent molecular probes for dopamine D2-like receptors von Huber, Daniela, Löber, Stefan, Hübner, Harald, Gmeiner, Peter

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A Chimeric Ligand Approach Leading to Potent Antiprion Active Acridine Derivatives:  Design, Synthesis, and Biological Investigations von Dollinger, Silke, Löber, Stefan, Klingenstein, Ralf, Korth, Carsten, Gmeiner, Peter

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Tricyclic antidepressants, quinacrine and a novel, synthetic chimera thereof clear prions by destabilizing detergent‐resistant membrane compartments von Klingenstein, Ralf, Löber, Stefan, Kujala, Pekka, Godsave, Susan, Leliveld, S. Rutger, Gmeiner, Peter, Peters, Peter J., Korth, Carsten

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Synthesis, Radiofluorination, and In Vitro Evaluation of Pyrazolo[1,5-a]pyridine-Based Dopamine D4 Receptor Ligands: Discovery of an Inverse Agonist Radioligand for PET von Prante, Olaf, Tietze, Rainer, Hocke, Carsten, Löber, Stefan, Hübner, Harald, Kuwert, Torsten, Gmeiner, Peter

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Rationally Based Efficacy Tuning of Selective Dopamine D4 Receptor Ligands Leading to the Complete Antagonist 2-[4-(4-Chlorophenyl)piperazin-1- ylmethyl]pyrazolo[1,5-a]pyridine (FA... von Löber, Stefan, Hübner, Harald, Utz, Wolfgang, Gmeiner, Peter

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Recent advances in the search for D3 - and D4 -selective drugs: probes, models and candidates von Löber, Stefan, Hübner, Harald, Tschammer, Nuska, Gmeiner, Peter

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GPCR crystal structures: Medicinal chemistry in the pocket von Shonberg, Jeremy, Kling, Ralf C., Gmeiner, Peter, Löber, Stefan

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Structure-based discovery of opioid analgesics with reduced side effects von Manglik, Aashish, Lin, Henry, Aryal, Dipendra K., McCorvy, John D., Dengler, Daniela, Corder, Gregory, Levit, Anat, Kling, Ralf C., Bernat, Viachaslau, Hübner, Harald, Huang, Xi-Ping, Sassano, Maria F., Giguère, Patrick M., Löber, Stefan, Da Duan, Scherrer, Grégory, Kobilka, Brian K., Gmeiner, Peter, Roth, Bryan L., Shoichet, Brian K.

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Novel azulene derivatives for the treatment of erectile dysfunction von Löber, Stefan, Hübner, Harald, Buschauer, Armin, Sanna, Fabrizio, Argiolas, Antonio, Melis, Maria Rosaria, Gmeiner, Peter

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Quinpramine ameliorates rat experimental autoimmune neuritis and redistributes MHC class II molecules von Meyer zu Hörste, Gerd, Mausberg, Anne K, Müller, Johanna I, Lehmann, Helmar C, Löber, Stefan, Gmeiner, Peter, Hartung, Hans-Peter, Stüve, Olaf, Korth, Carsten, Kieseier, Bernd C

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Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype von Hocke, Carsten, Prante, Olaf, Löber, Stefan, Hübner, Harald, Gmeiner, Peter, Kuwert, Torsten

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