Quantitative Phosphoproteomics Analysis of ERBB3/ERBB4 Signaling von Wandinger, Sebastian K, Lahortiga, Idoya, Jacobs, Kris, Klammer, Martin, Jordan, Nicole, Elschenbroich, Sarah, Parade, Marc, Jacoby, Edgar, Linders, Joannes T M, Brehmer, Dirk, Cools, Jan, Daub, Henrik

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Structural Investigation of B‑Raf Paradox Breaker and Inducer Inhibitors von Arora, Rohit, Di Michele, Michela, Stes, Elisabeth, Vandermarliere, Elien, Martens, Lennart, Gevaert, Kris, Van Heerde, Erika, Linders, Joannes T. M, Brehmer, Dirk, Jacoby, Edgar, Bonnet, Pascal

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MELK-T1, a small-molecule inhibitor of protein kinase MELK, decreases DNA-damage tolerance in proliferating cancer cells von Beke, Lijs, Kig, Cenk, Linders, Joannes T M, Boens, Shannah, Boeckx, An, van Heerde, Erika, Parade, Marc, De Bondt, An, Van den Wyngaert, Ilse, Bashir, Tarig, Ogata, Souichi, Meerpoel, Lieven, Van Eynde, Aleyde, Johnson, Christopher N, Beullens, Monique, Brehmer, Dirk, Bollen, Mathieu

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KCNE1 induces fenestration in the Kv7.1/KCNE1 channel complex that allows for highly specific pharmacological targeting von Wrobel, Eva, Rothenberg, Ina, Krisp, Christoph, Hundt, Franziska, Fraenzel, Benjamin, Eckey, Karina, Linders, Joannes T. M., Gallacher, David J., Towart, Rob, Pott, Lutz, Pusch, Michael, Yang, Tao, Roden, Dan M., Kurata, Harley T., Schulze-Bahr, Eric, Strutz-Seebohm, Nathalie, Wolters, Dirk, Seebohm, Guiscard

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Correction to Structural Investigation of B‑Raf Paradox Breaker and Inducer Inhibitors von Arora, Rohit, Di Michele, Michela, Stes, Elisabeth, Vandermarliere, Elien, Martens, Lennart, Gevaert, Kris, Van Heerde, Erika, Linders, Joannes T. M, Brehmer, Dirk, Jacoby, Edgar, Bonnet, Pascal

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Limited Proteolysis Combined with Stable Isotope Labeling Reveals Conformational Changes in Protein (Pseudo)kinases upon Binding Small Molecules von Di Michele, Michela, Stes, Elisabeth, Vandermarliere, Elien, Arora, Rohit, Astorga-Wells, Juan, Vandenbussche, Jonathan, van Heerde, Erika, Zubarev, Roman, Bonnet, Pascal, Linders, Joannes T. M, Jacoby, Edgar, Brehmer, Dirk, Martens, Lennart, Gevaert, Kris

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Fragment-Based Discovery of Type I Inhibitors of Maternal Embryonic Leucine Zipper Kinase von Johnson, Christopher N, Berdini, Valerio, Beke, Lijs, Bonnet, Pascal, Brehmer, Dirk, Coyle, Joseph E, Day, Phillip J, Frederickson, Martyn, Freyne, Eddy J. E, Gilissen, Ron A. H. J, Hamlett, Christopher C. F, Howard, Steven, Meerpoel, Lieven, McMenamin, Rachel, Patel, Sahil, Rees, David C, Sharff, Andrew, Sommen, François, Wu, Tongfei, Linders, Joannes T. M

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Structure-Based Design of Type II Inhibitors Applied to Maternal Embryonic Leucine Zipper Kinase von Johnson, Christopher N, Adelinet, Christophe, Berdini, Valerio, Beke, Lijs, Bonnet, Pascal, Brehmer, Dirk, Calo, Frederick, Coyle, Joseph E, Day, Phillip J, Frederickson, Martyn, Freyne, Eddy J. E, Gilissen, Ron A. H. J, Hamlett, Christopher C. F, Howard, Steven, Meerpoel, Lieven, Mevellec, Laurence, McMenamin, Rachel, Pasquier, Elisabeth, Patel, Sahil, Rees, David C, Linders, Joannes T. M

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Pharmacological dissection of Kv7.1 channels in systemic and pulmonary arteries von Chadha, Preet S, Zunke, Friederike, Davis, Alison J, Jepps, Thomas A, Linders, Joannes TM, Schwake, Michael, Towart, Rob, Greenwood, Iain A

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Design, synthesis and characterisation of a novel type II B-RAF paradox breaker inhibitor von Arora, Rohit, Linders, Joannes T.M., Aci-Sèche, Samia, Verheyen, Thomas, Van Heerde, Erika, Brehmer, Dirk, Chaikuad, Apirat, Knapp, Stefan, Bonnet, Pascal

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Correction: MELK-T1, a small-molecule inhibitor of protein kinase MELK, decreases DNA-damage tolerance in proliferating cancer cells von Beke, Lijs, Kig, Cenk, Linders, Joannes T M, Boens, Shannah, Boeckx, An, van Heerde, Erika, Parade, Marc, De Bondt, An, Van den Wyngaert, Ilse, Bashir, Tarig, Ogata, Souichi, Meerpoel, Lieven, Van Eynde, Aleyde, Johnson, Christopher N, Beullens, Monique, Brehmer, Dirk, Bollen, Mathieu

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High-content assays for evaluating cellular and hepatic diacylglycerol acyltransferase activity von Qi, Jenson, Lang, Wensheng, Giardino, Edward, Caldwell, Gary W., Smith, Charles, Minor, Lisa K., Darrow, Andrew L., Willemsens, Gustaaf, DeWaepenaert, Katharina, Roevens, Peter, Linders, Joannes T.M., Liang, Yin, Connelly, Margery A.

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Probes for Narcotic Receptor-Mediated Phenomena. 33. Construction of a Strained trans-5,6-Ring System by Displacement of a Nitro-Activated Aromatic Fluorine. Synthesis of the Penul... von Hashimoto, Akihiro, Przybyl, Anna K, Linders, Joannes T. M, Kodato, Shinichi, Tian, Xinrong, Deschamps, Jeffrey R, George, Clifford, Flippen-Anderson, Judith L, Jacobson, Arthur E, Rice, Kenner C

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Synthesis of rac-(1R,4aR,9aR)-2-methyl-1,3,4,9a-tetrahydro-2H-1,4a-propanobenzofuro[2,3-c]pyridin-6-ol. An unusual double rearrangement leading to the ortho- and para-f oxide-bridg... von Kodato, Shinichi, Linders, Joannes T M, Gu, Xiao-Hui, Yamada, Koichiro, Flippen-Anderson, Judith L, Deschamps, Jeffrey R, Jacobson, Arthur E, Rice, Kenner C

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Synthesis and evaluation of conformationally restricted N-[2-(3,4-dichlorophenyl)ethyl]-N-methyl-2-(1-pyrrolidinyl)ethylamines at .sigma. receptors. 2. Piperazines, bicyclic amines... von de Costa, Brian R, He, Xiaoshu, Linders, Joannes T. M, Dominguez, Celia, Gu, Zi Qiang, Williams, Wanda, Bowen, Wayne

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Synthesis and Biological Evaluation of Methylene-Bridged Analogs of the Potent Cannabinoid Receptor Antagonist Rimonabant von Ślusarczyk, Magdalena, De Borggraeve, Wim M., Hoornaert, Georges, Deroose, Frederik, Linders, Joannes T. M.

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An expeditious preparation of E-2-amino-5-hydroxyadamantane and its Z-isomer von Jaroskova, Libuse, Van der Veken, Louis, de Belser, Paul, Diels, Gaston, de Groot, Alex, Linders, Joannes T.M.

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Synthesis, configuration, and activity of isomeric 2-phenyl-2-(N-piperidinyl)bicyclo[3.1.0]hexanes at phencyclidine and .sigma. binding sites von De Costa, Brian R, Mattson, Mariena V, George, Clifford, Linders, Joannes T. M

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Pharmacological dissection of K v 7.1 channels in systemic and pulmonary arteries von Chadha, Preet S, Zunke, Friederike, Davis, Alison J, Jepps, Thomas A, Linders, Joannes TM, Schwake, Michael, Towart, Rob, Greenwood, Iain A

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Synthesis and binding properties of MK-801 isothiocyanates; (+)-3-isothiocyanato-5-methyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine hydrochloride: a new, potent and selec... von Linders, Joannes T. M, Monn, James A, Mattson, Mariena V, George, Clifford, Jacobson, Arthur E, Rice, Kenner C

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