Structural complementarity facilitates E7820-mediated degradation of RBM39 by DCAF15 von Faust, Tyler B., Yoon, Hojong, Nowak, Radosław P., Donovan, Katherine A., Li, Zhengnian, Cai, Quan, Eleuteri, Nicholas A., Zhang, Tinghu, Gray, Nathanael S., Fischer, Eric S.

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Bruton tyrosine kinase degradation as a therapeutic strategy for cancer von Dobrovolsky, Dennis, Wang, Eric S., Morrow, Sara, Leahy, Catharine, Faust, Tyler, Nowak, Radosław P., Donovan, Katherine A., Yang, Guang, Li, Zhengnian, Fischer, Eric S., Treon, Steven P., Weinstock, David M., Gray, Nathanael S.

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Broad-spectrum activity against mosquito-borne flaviviruses achieved by a targeted protein degradation mechanism von Liu, Han-Yuan, Li, Zhengnian, Reindl, Theresia, He, Zhixiang, Qiu, Xueer, Golden, Ryan P., Donovan, Katherine A., Bailey, Adam, Fischer, Eric S., Zhang, Tinghu, Gray, Nathanael S., Yang, Priscilla L.

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Discovery of Potent Degraders of the Dengue Virus Envelope Protein von Li, Zhengnian, Liu, Han‐Yuan, He, Zhixiang, Chakravarty, Antara, Golden, Ryan P., Jiang, Zixuan, You, Inchul, Yue, Hong, Donovan, Katherine A., Du, Guangyan, Che, Jianwei, Tse, Jason, Che, Isaac, Lu, Wenchao, Fischer, Eric S., Zhang, Tinghu, Gray, Nathanael S., Yang, Priscilla L.

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Molecular Bidents with Two Electrophilic Warheads as a New Pharmacological Modality von Li, Zhengnian, Jiang, Jie, Ficarro, Scott B., Beyett, Tyler S., To, Ciric, Tavares, Isidoro, Zhu, Yingde, Li, Jiaqi, Eck, Michael J., Jänne, Pasi A., Marto, Jarrod A., Zhang, Tinghu, Che, Jianwei, Gray, Nathanael S.

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A Concise Stereocontrolled Total Synthesis of (±)-Stemoamide von Li, Zhengnian, Zhang, Lijuan, Qiu, Fayang G.

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Mapping the Degradable Kinome Provides a Resource for Expedited Degrader Development von Donovan, Katherine A., Ferguson, Fleur M., Bushman, Jonathan W., Eleuteri, Nicholas A., Bhunia, Debabrata, Ryu, SeongShick, Tan, Li, Shi, Kun, Yue, Hong, Liu, Xiaoxi, Dobrovolsky, Dennis, Jiang, Baishan, Wang, Jinhua, Hao, Mingfeng, You, Inchul, Teng, Mingxing, Liang, Yanke, Hatcher, John, Li, Zhengnian, Manz, Theresa D., Groendyke, Brian, Hu, Wanyi, Nam, Yunju, Sengupta, Sandip, Cho, Hanna, Shin, Injae, Agius, Michael P., Ghobrial, Irene M., Ma, Michelle W., Che, Jianwei, Buhrlage, Sara J., Sim, Taebo, Gray, Nathanael S., Fischer, Eric S.

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Rewiring cancer drivers to activate apoptosis von Gourisankar, Sai, Krokhotin, Andrey, Ji, Wenzhi, Liu, Xiaofan, Chang, Chiung-Ying, Kim, Samuel H., Li, Zhengnian, Wenderski, Wendy, Simanauskaite, Juste M., Yang, Haopeng, Vogel, Hannes, Zhang, Tinghu, Green, Michael R., Gray, Nathanael S., Crabtree, Gerald R.

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Exploring the target scope of KEAP1 E3 ligase-based PROTACs von Du, Guangyan, Jiang, Jie, Henning, Nathaniel J., Safaee, Nozhat, Koide, Eriko, Nowak, Radosław P., Donovan, Katherine A., Yoon, Hojong, You, Inchul, Yue, Hong, Eleuteri, Nicholas A., He, Zhixiang, Li, Zhengnian, Huang, Hubert T., Che, Jianwei, Nabet, Behnam, Zhang, Tinghu, Fischer, Eric S., Gray, Nathanael S.

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Development and Characterization of a Wee1 Kinase Degrader von Li, Zhengnian, Pinch, Benika J., Olson, Calla M., Donovan, Katherine A., Nowak, Radosław P., Mills, Caitlin E., Scott, David A., Doctor, Zainab M., Eleuteri, Nicholas A., Chung, Mirra, Sorger, Peter K., Fischer, Eric S., Gray, Nathanael S.

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Discovery of CRBN-Dependent WEE1 Molecular Glue Degraders from a Multicomponent Combinatorial Library von Razumkov, Hlib, Jiang, Zixuan, Baek, Kheewoong, You, Inchul, Geng, Qixiang, Donovan, Katherine A., Tang, Michelle T., Metivier, Rebecca J., Mageed, Nada, Seo, Pooreum, Li, Zhengnian, Byun, Woong Sub, Hinshaw, Stephen M., Sarott, Roman C., Fischer, Eric S., Gray, Nathanael S.

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ZNL0325, a Pyrazolopyrimidine-Based Covalent Probe, Demonstrates an Alternative Binding Mode for Kinases von Li, Zhengnian, Lu, Wenchao, Beyett, Tyler S., Ficarro, Scott B., Jiang, Jie, Tse, Jason, Kim, Audrey Yong-Ju, Marto, Jarrod A., Che, Jianwei, Jänne, Pasi A., Eck, Michael J., Zhang, Tinghu, Gray, Nathanael S.

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Author Correction: Rewiring cancer drivers to activate apoptosis von Gourisankar, Sai, Krokhotin, Andrey, Ji, Wenzhi, Liu, Xiaofan, Chang, Chiung-Ying, Kim, Samuel H., Li, Zhengnian, Wenderski, Wendy, Simanauskaite, Juste M., Yang, Haopeng, Vogel, Hannes, Zhang, Tinghu, Green, Michael R., Gray, Nathanael S., Crabtree, Gerald R.

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Quinazolinones as allosteric fourth-generation EGFR inhibitors for the treatment of NSCLC von Gero, Thomas W., Heppner, David E., Beyett, Tyler S., To, Ciric, Azevedo, Seth C., Jang, Jaebong, Bunnell, Thomas, Feru, Frederic, Li, Zhengnian, Shin, Bo Hee, Soroko, Kara M., Gokhale, Prafulla C., Gray, Nathanael S., Jänne, Pasi A., Eck, Michael J., Scott, David A.

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Synthesis and Structure–Activity relationships of cyclin-dependent kinase 11 inhibitors based on a diaminothiazole scaffold von Li, Zhengnian, Ishida, Ryosuke, Liu, Yan, Wang, Jinhua, Li, Yina, Gao, Yang, Jiang, Jie, Che, Jianwei, Sheltzer, Jason M., Robers, Matthew B., Zhang, Tinghu, Westover, Kenneth D., Nabet, Behnam, Gray, Nathanael S.

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Identification of small molecule inhibitors targeting the Zika virus envelope protein von Pitts, Jared, Hsia, Chih-Yun, Lian, Wenlong, Wang, Jinhua, Pfeil, Marc-Philipp, Kwiatkowski, Nicholas, Li, Zhengnian, Jang, Jaebong, Gray, Nathanael S., Yang, Priscilla L.

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Triple Degradation of BTK, IKZF1 and IKZF3 in B-Cell Malignancies von Morrow, Sara, Dobrovolsky, Dennis, Wang, Eric, Nowak, Radosław P., Donovan, Katherine, Faust, Tyler, Yang, Guang, Li, Zhengnian, Fischer, Eric, Treon, Steven P, Weinstock, David M, Gray, Nathanael S.

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Benzopyrimidodiazepinone inhibitors of TNK2 von Groendyke, Brian J., Powell, Chelsea E., Feru, Frederic, Gero, Thomas W., Li, Zhengnian, Szabo, Hilary, Pang, Kevin, Feutrill, John, Chen, Bailing, Li, Bin, Gray, Nathanael S., Scott, David A.

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Discovery of a series of benzopyrimidodiazepinone TNK2 inhibitors via scaffold morphing von Li, Zhengnian, Powell, Chelsea E., Groendyke, Brian J., Gero, Thomas W., Feru, Frederic, Feutrill, John, Chen, Bailing, Li, Bin, Szabo, Hilary, Gray, Nathanael S., Scott, David A.

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Influence of TMGa Flux on the Improvement of GaN Films on Thick Freestanding Diamond Films von Cui, Shan Lin, Li, Zheng Nian, Gang, Hong

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