Structure-Based Design of β‑Site APP Cleaving Enzyme 1 (BACE1) Inhibitors for the Treatment of Alzheimer’s Disease von Yuan, Jing, Venkatraman, Shankar, Zheng, Yajun, McKeever, Brian M, Dillard, Lawrence W, Singh, Suresh B

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Optimization of orally bioavailable alkyl amine renin inhibitors von Xu, Zhenrong, Cacatian, Salvacion, Yuan, Jing, Simpson, Robert D., Jia, Lanqi, Zhao, Wei, Tice, Colin M., Flaherty, Patrick T., Guo, Joan, Ishchenko, Alexey, Singh, Suresh B., Wu, Zhongren, McKeever, Brian M., Scott, Boyd B., Bukhtiyarov, Yuri, Berbaum, Jennifer, Mason, Jennifer, Panemangalore, Reshma, Cappiello, Maria Grazia, Bentley, Ross, Doe, Christopher P., Harrison, Richard K., McGeehan, Gerard M., Dillard, Lawrence W., Baldwin, John J., Claremon, David A.

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Effects of the bace1 inhibitor bi 1181181 and the anti-abeta antibody m266 on abeta in rat brain homogenate and CSF von Hobson, Scott, Lenter, Martin C, Sauer, Achim, Fuchs, Klaus, Lala, Deepak S, Dillard, Lawrence W, Dorner-Ciossek, Cornelia

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Cloning, Characterization and Site-Directed Mutagenesis of Canine Renin von Bukhtiyarov, Yuri, Zecher, Marianne, Panemangalore, Reshma, Wu, Zhongren, Bruno, Joseph G, Yuan, Jing, Xu, Zhenrong, Dillard, Lawrence W, McGeehan, Gerard M, Harrison, Richard K, Scott, Boyd B

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Pharmacological characterization of the new bace1 inhibitor bi 1181181 von Dorner-Ciossek, Cornelia, Hobson, Scott, Fuchs, Klaus, Sauer, Achim, Bauer, Margit, Morales-Ramos, Angel, Venkatraman, Shankar, Dillard, Lawrence W, Kruk, Barbara, Howard, Lamont, Bukhtiyarov, Yuri, Zhao, Yi, Lala, Deepak S

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Synthesis of 2-amino-5-benzoyl-4-(2-furyl)thiazoles as adenosine A(2A) receptor antagonists von Cole, Andrew G, Stauffer, Tara M, Rokosz, Laura L, Metzger, Axel, Dillard, Lawrence W, Zeng, Wenguang, Henderson, Ian

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Synthesis of 2-amino-5-benzoyl-4-(2-furyl)thiazoles as adenosine A2A receptor antagonists von COLE, Andrew G, STAUFFER, Tara M, ROKOSZ, Laura L, METZGER, Axel, DILLARD, Lawrence W, WENGUANG ZENG, HENDERSON, Ian

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Complex Synthetic Chemical Libraries Indexed with Molecular Tags von Michael H. J. Ohlmeyer, Swanson, Robert N., Dillard, Lawrence W., Reader, John C., Asouline, Gigi, Kobayashi, Ryuji, Wigler, Michael, Still, W. Clark

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Discovery of VTP-27999, an Alkyl Amine Renin Inhibitor with Potential for Clinical Utility von Jia, Lanqi, Simpson, Robert D, Yuan, Jing, Xu, Zhenrong, Zhao, Wei, Cacatian, Salvacion, Tice, Colin M, Guo, Joan, Ishchenko, Alexey, Singh, Suresh B, Wu, Zhongren, McKeever, Brian M, Bukhtiyarov, Yuri, Johnson, Judith A, Doe, Christopher P, Harrison, Richard K, McGeehan, Gerard M, Dillard, Lawrence W, Baldwin, John J, Claremon, David A

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Biphenyl/diphenyl ether renin inhibitors: Filling the S1 pocket of renin via the S3 pocket von Yuan, Jing, Simpson, Robert D., Zhao, Wei, Tice, Colin M., Xu, Zhenrong, Cacatian, Salvacion, Jia, Lanqi, Flaherty, Patrick T., Guo, Joan, Ishchenko, Alexey, Wu, Zhongren, McKeever, Brian M., Scott, Boyd B., Bukhtiyarov, Yuri, Berbaum, Jennifer, Panemangalore, Reshma, Bentley, Ross, Doe, Christopher P., Harrison, Richard K., McGeehan, Gerard M., Singh, Suresh B., Dillard, Lawrence W., Baldwin, John J., Claremon, David A.

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Stereospecific total syntheses of decahydroquinoline alkaloids (.+-.)-195A and (.+-.)-2-epi-195A von Polniaszek, Richard P, Dillard, Lawrence W

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Design and optimization of renin inhibitors: Orally bioavailable alkyl amines von Tice, Colin M., Xu, Zhenrong, Yuan, Jing, Simpson, Robert D., Cacatian, Salvacion T., Flaherty, Patrick T., Zhao, Wei, Guo, Joan, Ishchenko, Alexey, Singh, Suresh B., Wu, Zhongren, Scott, Boyd B., Bukhtiyarov, Yuri, Berbaum, Jennifer, Mason, Jennifer, Panemangalore, Reshma, Cappiello, Maria Grazia, Müller, Dominik, Harrison, Richard K., McGeehan, Gerard M., Dillard, Lawrence W., Baldwin, John J., Claremon, David A.

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P4‐168: Effects of the bace1 inhibitor bi 1181181 and the anti‐abeta antibody m266 on abeta in rat brain homogenate and CSF von Hobson, Scott, Lenter, Martin C., Sauer, Achim, Fuchs, Klaus, Lala, Deepak S., Dillard, Lawrence W., Dorner-Ciossek, Cornelia

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P1‐314: Pharmacological characterization of the new bace1 inhibitor bi 1181181 von Dorner-Ciossek, Cornelia, Hobson, Scott, Fuchs, Klaus, Sauer, Achim, Bauer, Margit, Morales-Ramos, Angel, Venkatraman, Shankar, Dillard, Lawrence W., Kruk, Barbara, Howard, Lamont, Bukhtiyarov, Yuri, Zhao, Yi, Lala, Deepak S.

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Diastereoselective addition of organometallic reagents to chiral iminium ions: Synthesis of ( S)-(+)-cryptostyline I von Polniaszek, Richard P., Dillard, Lawrence W.

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Synthesis of 2-amino-5-benzoyl-4-(2-furyl)thiazoles as adenosine A 2A receptor antagonists von Cole, Andrew G., Stauffer, Tara M., Rokosz, Laura L., Metzger, Axel, Dillard, Lawrence W., Zeng, Wenguang, Henderson, Ian

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A Paradigm for Drug Discovery Employing Encoded Combinatorial Libraries von Burbaum, Jonathan J., Michael H. J. Ohlmeyer, Reader, John C., Henderson, Ian, Dillard, Lawrence W., Li, Ge, Randle, Troy L., Sigal, Nolan H., Chelsky, Daniel, Baldwin, John J.

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INHIBITORS OF BETA-SECRETASE von CLAREMON, DAVID A, FUCHS, KLAUS, MCKEEVER, BRIAN, YUAN, JING, HEINE, NIKLAS, DILLARD, LAWRENCE W, XU, ZHENRONG, VENKATRAMAN, SHANKAR, WU, GUOSHENG, WU, ZHONGREN, LEFTHERIS, KATERINA, ZHENG, YAJUN, JIA, LANQI, MORALES-RAMOS, ANGEL, CACATIAN, SALVACION, SINGH, SURESH

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Complex combinatorial chemical libraries encoded with tags von READER JOHN C.,STILL W. CLARK,DILLARD LAWRENCE W.,OHLMEYER MICHAEL H. J.,WIGLER MICHAEL H

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Inhibitors of beta-secretase von YUAN JING, DILLARD LAWRENCE W, ZHENG YAJUN, JIA LANQI

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