Drug discovery management, small is still beautiful: Why a number of companies get it wrong von Knutsen, Lars J.S.

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Discovery and Characterization of 6-{4-[3-(R)-2-Methylpyrrolidin-1-yl)propoxy]phenyl}-2H-pyridazin-3-one (CEP-26401, Irdabisant): A Potent, Selective Histamine H3 Receptor Inverse... von Hudkins, Robert L, Raddatz, Rita, Tao, Ming, Mathiasen, Joanne R, Aimone, Lisa D, Becknell, Nadine C, Prouty, Catherine P, Knutsen, Lars J. S, Yazdanian, Mehran, Moachon, Gilbert, Ator, Mark A, Mallamo, John P, Marino, Michael J, Bacon, Edward R, Williams, Michael

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Emerging Opportunities for Antipsychotic Drug Discovery in the Postgenomic Era von Marino, Michael J, Knutsen, Lars J. S, Williams, Michael

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Diffuse gastric cancer: Emerging mechanisms of tumor initiation and progression von Monster, Jooske L., Kemp, Lars J.S., Gloerich, Martijn, van der Post, Rachel S.

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Crater wear mechanism of TiAlN coatings during high-speed metal turning von Moreno, Maiara, Andersson, Jon M., Boyd, Robert, Johansson-Jöesaar, Mats P., Johnson, Lars J.S., Odén, Magnus, Rogström, Lina

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High temperature phase decomposition in TixZryAlzN von Lind, Hans, Pilemalm, Robert, Rogström, Lina, Tasnadi, Ferenc, Ghafoor, Naureen, Forsén, Rikard, S. Johnson, Lars J., Johansson-Jöesaar, Mats P., Odén, Magnus, Abrikosov, Igor A.

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Synthesis and SAR of novel 2-arylthiazolidinones as selective analgesic N-type calcium channel blockers von Knutsen, Lars J.S., Hobbs, Christopher J., Earnshaw, Christopher G., Fiumana, Andrea, Gilbert, Jenny, Mellor, Sarah L., Radford, Fleur, Smith, Nichola J., Birch, Philip J., Russell Burley, J., Ward, Stuart D.C., James, Iain F.

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Reduction of multiple hits in atom probe tomography von Thuvander, Mattias, Kvist, Anders, Johnson, Lars J.S., Weidow, Jonathan, Andrén, Hans-Olof

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Resolving mass spectral overlaps in atom probe tomography by isotopic substitutions - case of TiSi 15 N von Engberg, David L J, Johnson, Lars J S, Jensen, Jens, Thuvander, Mattias, Hultman, Lars

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Cell division‐dependent dissemination following E‐cadherin loss underlies initiation of diffuse‐type gastric cancer von Monster, Jooske L, Kemp, Lars JS, Busslinger, Georg A, Vliem, Marjolein J, Derks, Lucca LM, Staes, Annelot AL, Bisseling, Tanya M, Clevers, Hans, Post, Rachel S, Gloerich, Martijn

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Nanolabyrinthine ZrAlN thin films by self-organization of interwoven single-crystal cubic and hexagonal phases von Ghafoor, Naureen, Johnson, Lars J. S., Klenov, Dmitri O., Demeulemeester, Jelly, Desjardins, Patrick, Petrov, Ivan, Hultman, Lars, Odén, Magnus

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Synthesis of Novel GABA Uptake Inhibitors. 3. Diaryloxime and Diarylvinyl Ether Derivatives of Nipecotic Acid and Guvacine as Anticonvulsant Agents von Knutsen, Lars J. S, Andersen, Knud Erik, Lau, Jesper, Lundt, Behrend F, Henry, Rodger F, Morton, Howard E, Nærum, Lars, Petersen, Hans, Stephensen, Henrik, Suzdak, Peter D, Swedberg, Michael D. B, Thomsen, Christian, Sørensen, Per O

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The Effect of Cathodic Arc Guiding Magnetic Field on the Growth of (Ti0.36Al0.64)N Coatings von Chaar, Ana B. B., Syed, Bilal, Hsu, Tun-Wei, Johansson-Jöesaar, Mats, Andersson, Jon M., Henrion, Gérard, Johnson, Lars J. S., Mücklich, Frank, Odén, Magnus

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Synthesis of Novel GABA Uptake Inhibitors. 4. Bioisosteric Transformation and Successive Optimization of Known GABA Uptake Inhibitors Leading to a Series of Potent Anticonvulsant D... von Andersen, Knud Erik, Sørensen, Jan L, Huusfeldt, Per O, Knutsen, Lars J. S, Lau, Jesper, Lundt, Behrend F, Petersen, Hans, Suzdak, Peter D, Swedberg, Michael D. B

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The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinec... von Andersen, Knud Erik, Braestrup, Claus, Groenwald, Frederik C, Joergensen, Anker S, Nielsen, Erik B, Sonnewald, Ursula, Soerensen, Per O, Suzdak, Peter D, Knutsen, Lars J. S

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Antagonists of the human adenosine A2A receptor. Part 1 Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives von GILLESPIE, Roger J, ADAMS, David R, JORDAN, Allan M, KNIGHT, Antony R, KNUTSEN, Lars J. S, LAWRENCE, Anthony, LERPINIERE, Joanne, MISRA, Anil, PORTER, Richard H. P, PRATT, Robert M, SHEPHERD, Robin, UPTON, Rebecca, BEBBINGTON, David, WARD, Simon E, WEISS, Scott M, WILLIAMSON, Douglas S, BENWELL, Karen, CLIFFE, Ian A, DAWSON, Claire E, DOURISH, Colin T, FLETCHER, Allan, GAUR, Suneel, GILES, Paul R

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Adhesive wear of TiAlN coatings during low speed turning of stainless steel 316L von Moreno, Maiara, Andersson, Jon M., M'Saoubi, Rachid, Kryzhanivskyy, Vyacheslav, Johansson-Jöesaar, Mats P., Johnson, Lars J.S., Odén, Magnus, Rogström, Lina

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Diffuse gastric cancer: Emerging mechanisms of tumor initiation and progression von Monster, Jooske L, Kemp, Lars J S, Gloerich, Martijn, van der Post, Rachel S

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Wear of Mo- and W-alloyed TiAlN coatings during high-speed turning of stainless steel von Moreno, Maiara, Andersson, Jon M., Johansson-Jöesaar, Mats P., Friedrich, Birgit E., Boyd, Robert, Schramm, Isabella C., Johnson, Lars J.S., Odén, Magnus, Rogström, Lina

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N-Substituted Adenosines as Novel Neuroprotective A1 Agonists with Diminished Hypotensive Effects von Knutsen, Lars J. S, Lau, Jesper, Petersen, Hans, Thomsen, Christian, Weis, Jan U, Shalmi, Michael, Judge, Martin E, Hansen, Anker Jon, Sheardown, Malcolm J

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