Combining Machine Learning and Molecular Dynamics to Predict P‑Glycoprotein Substrates von Esposito, Carmen, Wang, Shuzhe, Lange, Udo E. W, Oellien, Frank, Riniker, Sereina

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De Novo Design, Synthesis, and Biological Evaluation of 3,4-Disubstituted Pyrrolidine Sulfonamides as Potent and Selective Glycine Transporter 1 Competitive Inhibitors von Wang, Ying, Zhao, Hongyu, Brewer, Jason T, Li, Huanqiu, Lao, Yanbin, Amberg, Willi, Behl, Berthold, Akritopoulou-Zanze, Irini, Dietrich, Justin, Lange, Udo E. W, Pohlki, Frauke, Hoft, Carolin, Hornberger, Wilfried, Djuric, Stevan W, Sydor, Jens, Mezler, Mario, Relo, Ana Lucia, Vasudevan, Anil

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Discovery of Novel Aminotetralines and Aminochromanes as Selective and Competitive Glycine Transporter 1 (GlyT1) Inhibitors von Amberg, Willi, Lange, Udo E. W, Ochse, Michael, Pohlki, Frauke, Behl, Berthold, Relo, Ana Lucia, Hornberger, Wilfried, Hoft, Carolin, Mezler, Mario, Sydor, Jens, Wang, Ying, Zhao, Hongyu, Brewer, Jason T, Dietrich, Justin, Li, Huanqiu, Akritopoulou-Zanze, Irini, Lao, Yanbin, Hannick, Steven M, Ku, Yi-Yin, Vasudevan, Anil

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Enzymatic Late‐Stage Oxidation of Lead Compounds with Solubilizing Biomimetic Docking/Protecting groups von Vickers, Clare, Backfisch, Gisela, Oellien, Frank, Piel, Isabel, Lange, Udo E. W.

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Frontispiece: Enzymatic Late‐Stage Oxidation of Lead Compounds with Solubilizing Biomimetic Docking/Protecting groups von Vickers, Clare, Backfisch, Gisela, Oellien, Frank, Piel, Isabel, Lange, Udo E. W.

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Emerging technologies for metabolite generation and structural diversification von Cusack, Kevin P., Koolman, Hannes F., Lange, Udo E.W., Peltier, Hillary M., Piel, Isabel, Vasudevan, Anil

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Amine Additives Greatly Expand the Scope of Asymmetric Hydrosilylation of Imines von Verdaguer, Xavier, Lange, Udo E. W., Buchwald, Stephen L.

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Orally active thrombin inhibitors. Part 2: Optimization of the P2-moiety von Lange, Udo E.W., Baucke, Dorit, Hornberger, Wilfried, Mack, Helmut, Seitz, Werner, Höffken, H. Wolfgang

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Orally active thrombin inhibitors. Part 1: Optimization of the P1-moiety von Mack, Helmut, Baucke, Dorit, Hornberger, Wilfried, Lange, Udo E.W., Seitz, Werner, Höffken, H. Wolfgang

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Highly Enantioselective Imine Hydrosilylation Using (S,S)-Ethylenebis(η5-tetrahydroindenyl)titanium Difluoride von Verdaguer, Xavier, Lange, Udo E. W., Reding, Matthew T., Buchwald, Stephen L.

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Synthesis and SAR of highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drugs von KLING, Andreas, LANGE, Udo E. W, UNGER, Liliane, WICKE, Karsten, SCHELLHAAS, Kurt, STEINER, Gerd, MACK, Helmut, BAKKER, Margot H. M, DRESCHER, Karla U, HORNBERGER, Wilfried, HUTCHINS, Charles W, MÖLLER, Achim, MÜLLER, Reinhold, SCHMIDT, Martin

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Solid-phase synthesis of thrombin inhibitors von Lange, Udo E.W., Zechel, Christian

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d-Phe-Pro-Arg type thrombin inhibitors: unexpected selectivity by modification of the P1 moiety von Lange, Udo E.W, Baucke, Dorit, Hornberger, Wilfried, Mack, Helmut, Seitz, Werner, Höffken, H.Wolfgang

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Solid-Phase synthesis of endothelin receptor antagonists von Lange, Udo E.W, Braje, Wilfried M, Amberg, Willi, Kettschau, Georg

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Design and synthesis of 1,5- and 2,5-substituted tetrahydrobenzazepinones as novel potent and selective integrin αvβ3antagonists von KLING, Andreas, BACKFISCH, Gisela, DELZER, Jürgen, GENESTE, Herve, GRAEF, Claudia, HORNBERGER, Wilfried, LANGE, Udo E. W, LAUTERBACH, Arnulf, SEITZ, Werner, SUBKOWSKI, Thomas

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ChemInform Abstract: Emerging Technologies for Metabolite Generation and Structural Diversification von Cusack, Kevin P., Koolman, Hannes F., Lange, Udo E. W., Peltier, Hillary M., Piel, Isabel, Vasudevan, Anil

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Synthesis and SAR of N-substituted dibenzazepinone derivatives as novel potent and selective αVβ3 antagonists von KLING, Andreas, BACKFISCH, Gisela, SEITZ, Werner, SUBKOWSKI, Thomas, DELZER, Jürgen, GENESTE, Hervé, GRAEF, Claudia, HOLZENKAMP, Uta, HORNBERGER, Wilfried, LANGE, Udo E. W, LAUTERBACH, Arnulf, MACK, Helmut

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Synthesis of highly potent and selective hetaryl ureas as integrin αvβ3-Receptor antagonists von LANGE, Udo E. W, BACKFISCH, Gisela, DELZER, Jürgen, GENESTE, Hervé, GRAEF, Claudia, HORNBERGER, Wilfried, KLING, Andreas, LAUTERBACH, Arnulf, SUBKOWSKI, Thomas, ZECHEL, Christian

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Highly potent and selective αvβ3-receptor antagonists: Solid-phase synthesis and SAR of 1-substituted 4-amino-1H-pyrimidin-2-ones von ZECHEL, Christian, BACKFISCH, Gisela, SUBKOWSKI, Thomas, DELZER, Jürgen, GENESTE, Hervé, GRAEF, Claudia, HORNBERGER, Wilfried, KLING, Andreas, LANGE, Udo E. W, LAUTERBACH, Arnulf, SEITZ, Werner

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Synthesis and SAR of N-substituted dibenzazepinone derivatives as novel potent and selective alpha(V)beta(3) antagonists von Kling, Andreas, Backfisch, Gisela, Delzer, Jürgen, Geneste, Hervé, Graef, Claudia, Holzenkamp, Uta, Hornberger, Wilfried, Lange, Udo E W, Lauterbach, Arnulf, Mack, Helmut, Seitz, Werner, Subkowski, Thomas

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