Identification of a peptide inhibitor for the histone methyltransferase WHSC1 von Morrison, Michael J, Boriack-Sjodin, P Ann, Swinger, Kerren K, Wigle, Tim J, Sadalge, Dipti, Kuntz, Kevin W, Scott, Margaret Porter, Janzen, William P, Chesworth, Richard, Duncan, Kenneth W, Harvey, Darren M, Lampe, John W, Mitchell, Lorna H, Copeland, Robert A

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Conformational-Design-Driven Discovery of EZM0414: A Selective, Potent SETD2 Inhibitor for Clinical Studies von Alford, Joshua S., Lampe, John W., Brach, Dorothy, Chesworth, Richard, Cosmopoulos, Kat, Duncan, Kenneth W., Eckley, Sean T., Kutok, Jeffrey L., Raimondi, Alejandra, Riera, Thomas V., Shook, Brian, Tang, Cuyue, Totman, Jennifer, Farrow, Neil A.

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Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical Studies von Lampe, John W, Alford, Joshua S, Boriak-Sjodin, P. Ann, Brach, Dorothy, Cosmopoulos, Kat, Duncan, Kenneth W, Eckley, Sean T, Foley, Megan A, Harvey, Darren M, Motwani, Vinny, Munchhof, Michael J, Raimondi, Alejandra, Riera, Thomas V, Tang, Cuyue, Thomenius, Michael J, Totman, Jennifer, Farrow, Neil A

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Indazoles: Regioselective Protection and Subsequent Amine Coupling Reactions von Slade, David J, Pelz, Nicholas F, Bodnar, Wanda, Lampe, John W, Watson, Paul S

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Total Synthesis of (-)- and (+)-Balanol(1) von Lampe, John W., Hughes, Philip F., Biggers, Christopher K., Smith, Shelley H., Hu, Hong

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(Imidazolylphenyl)pyrrol-2-one inhibitors of cardiac cAMP phosphodiesterase von Lampe, John W, Chou, Yuo Ling, Hanna, Reda G, Di Meo, Susan V, Erhardt, Paul W, Hagedorn, Alfred A, Ingebretsen, William R, Cantor, Elinor

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Examination of the olefin–olefin ring closing metathesis to prepare Latrunculin B von She, Jin, Lampe, John W., Polianski, Alexandra B., Watson, Paul S.

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Total Synthesis of (−)- and (+)-Balanol1 von Lampe, John W, Hughes, Philip F, Biggers, Christopher K, Smith, Shelley H, Hu, Hong

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Synthesis and pharmacological studies of N-[4-[2-hydroxy-3-[[2-[4-(1H-imidazol-1-yl)phenoxy]ethyl]amino]propoxy]phenyl]methanesulfonamide, a novel antiarrhythmic agent with class I... von Morgan, Thomas K, Lis, Randall, Lumma, William C, Wohl, Ronald A, Nickisch, Klaus, Phillips, Gary B, Lind, Joan M, Lampe, John W, Di Meo, Susan V

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Heterocyclic analogs of benzamide antiarrhythmic agents von Hanna, Reda, Lampe, John W, Lumma, William C, Erhardt, Paul W, Wong, Samuel S, Sullivan, Mark E

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PYRIDIN-2-ONE COMPOUNDS USEFUL AS SMARCA2 ANTAGONISTS von Lampe, John W, Munchhof, Michael John, Duncan, Kenneth William, Moradei, Oscar, Harvey, Darren Martin, Campbell, John Emmerson

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Synthesis and Protein Kinase C Inhibitory Activities of Acyclic Balanol Analogs That Are Highly Selective for Protein Kinase C over Protein Kinase A von Defauw, Jean M., Murphy, Marcia M., Jagdmann, G. Erik, Hu, Hong, Lampe, John W., Hollinshead, Sean P., Mitchell, Thomas J., Crane, Heidi M., Heerding, Julia M., Mendoza, José S., Davis, Jefferson E., Darges, James W., Hubbard, Frederick R., Hall, Steven E.

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COMPOSÉS DE PYRIDIN-2-ONE UTILES EN TANT QU'ANTAGONISTES DE SMARCA2 von CAMPBELL, John, Emmerson, HARVEY, Darren, Martin, MORADEI, Oscar, MUNCHHOF, Michael, John, DUNCAN, Kenneth, William, LAMPE, John, W

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PYRIDIN-2-ONE COMPOUNDS USEFUL AS SMARCA2 ANTAGONISTS von HARVEY, Darren, Martin, CAMPBELL, John, Emmerson, MORADEI, Oscar, MUNCHHOF, Michael, John, DUNCAN, Kenneth, William, LAMPE, John, W

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Pyridin-2-one compounds useful as smarca2 antagonists von MUNCHHOF Michael John, MORADEI Oscar, DUNCAN Kenneth William, LAMPE John W, HARVEY DARREN MARTIN, CAMPBELL John Emmerson

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Pyridin-2-one compounds useful as SMARCA2 antagonists von MORADEI, Oscar, CAMPBELL, John Emmerson, MUNCHHOF, Michael John, LAMPE, John W, HARVEY, Darren Martin, DUNCAN, Kenneth William

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PYRIDIN-2-ONE COMPOUNDS USEFUL AS SMARCA2 ANTAGONISTS von HARVEY, DARREN MARTIN, LAMPE, JOHN W, CAMPBELL, JOHN EMMERSON, MORADEI, OSCAR, DUNCAN, KENNETH WILLIAM, MUNCHHOF, MICHAEL JOHN

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Potent and selective PKC inhibitory 5-membered ring analogs of balanol with replacement of the carboxamide moiety von Jagdmann, G.Erik, Defauw, Jean M., Lampe, John W., Darges, James W., Kalter, Kiyomi

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TRICYCLIC COMPOUNDS AS INHIBITORS OF MUTANT IDH ENZYMES von HUANG, Chunhui, ELLIS, J. Michael, ESPOSITE, Sara, UJJAINWALLA, Feroze, CHILDERS, Matthew, L, SCIAMMETTA, Nunzio, FISCHER, Christian, LAMPE, John, W, OTTE, Ryan, D, SLOMAN, David, L, PARKER, Dann, L., Jr, REUTERSHAN, Michael, WHITE, Catherine, BOGEN, Stephane, L, LLINAS, Francesc Xavier Fradera, HONG, Qingmei, MACHACEK, Michelle, R, WU, Zhicai, SHAO, Pengcheng, P, MCMASTERS, Daniel, R, KIM, Alexander, J

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PYRIDIN-2-ONE COMPOUNDS USEFUL AS SMARCA2 ANTAGONISTS von DUNCAN KENNETH WILLIAM, CAMPBELL JOHN EMMERSON, MUNCHHOF MICHAEL JOHN, MORADEI OSCAR, LAMPE JOHN W, HARVEY DARREN

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