Comprehensive characterization of the Published Kinase Inhibitor Set von Elkins, Jonathan M, Fedele, Vita, Szklarz, Marta, Abdul Azeez, Kamal R, Salah, Eidarus, Mikolajczyk, Jowita, Romanov, Sergei, Sepetov, Nikolai, Huang, Xi-Ping, Roth, Bryan L, Al Haj Zen, Ayman, Fourches, Denis, Muratov, Eugene, Tropsha, Alex, Morris, Joel, Teicher, Beverly A, Kunkel, Mark, Polley, Eric, Lackey, Karen E, Atkinson, Francis L, Overington, John P, Bamborough, Paul, Müller, Susanne, Price, Daniel J, Willson, Timothy M, Drewry, David H, Knapp, Stefan, Zuercher, William J

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Optimization and SAR for dual ErbB-1/ErbB-2 tyrosine kinase inhibition in the 6-furanylquinazoline series von Petrov, Kimberly G., Zhang, Yue-Mei, Carter, Malcolm, Cockerill, G. Stuart, Dickerson, Scott, Gauthier, Cassandra A., Guo, Yu, Mook, Robert A., Rusnak, David W., Walker, Ann L., Wood, Edgar R., Lackey, Karen E.

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A public-private partnership to unlock the untargeted kinome von Knapp, Stefan, Arruda, Paulo, Blagg, Julian, Burley, Stephen, Drewry, David H, Edwards, Aled, Fabbro, Doriano, Gillespie, Paul, Gray, Nathanael S, Kuster, Bernhard, Lackey, Karen E, Mazzafera, Paulo, Tomkinson, Nicholas C O, Willson, Timothy M, Workman, Paul, Zuercher, William J

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RET Activation Inhibits Doxorubicin-induced Apoptosis in SK-N-MC Cells von SKINNER, Michael A, LACKEY, Karen E, FREEMERMAN, Alex J

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The discovery of potent and selective 4-aminothienopyridines as B-Raf kinase inhibitors von Tang, Jun, Lackey, Karen E., Dickerson, Scott H.

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Discovery and in vitro evaluation of potent kinase inhibitors: Pyrido[1′,2′:1,5]pyrazolo[3,4- d]pyrimidines von Alberti, Michael J., Auten, Elizabeth P., Lackey, Karen E., McDonald, Octerloney B., Wood, Edgar R., Preugschat, Frank, Cutler, Geoffrey J., Kane-Carson, Laurie, Liu, Wei, Jung, David K.

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Oxindole-Based Inhibitors of Cyclin-Dependent Kinase 2 (CDK2):  Design, Synthesis, Enzymatic Activities, and X-ray Crystallographic Analysis von Bramson, H. Neal, Corona, John, Davis, Stephen T, Dickerson, Scott H, Edelstein, Mark, Frye, Stephen V, Gampe, Robert T, Harris, Phil A, Hassell, Anne, Holmes, William D, Hunter, Robert N, Lackey, Karen E, Lovejoy, Brett, Luzzio, Michael J, Montana, Val, Rocque, Warren J, Rusnak, David, Shewchuk, Lisa, Veal, James M, Walker, Duncan H, Kuyper, Lee F

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Knowledge-based design of 7-azaindoles as selective B-Raf inhibitors von Tang, Jun, Hamajima, Toshihiro, Nakano, Masato, Sato, Hideyuki, Dickerson, Scott H., Lackey, Karen E.

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Synthesis of 2-chloro-5,7-dihydro-6 H -pyrrolo[2,3- d ]pyrimidin-6-one von Cheung, Mui, Harris, Philip A, Lackey, Karen E

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Discovery and in vitro evaluation of potent kinase inhibitors : Pyrido[1',2':1,5]pyrazolo[3,4-d]pyrimidines: G-protein-coupled receptors in drug discovery von ALBERTI, Michael J, AUTEN, Elizabeth P, LACKEY, Karen E, MCDONALD, Octerloney B, WOOD, Edgar R, PREUGSCHAT, Frank, CUTLER, Geoffrey J, KANE-CARSON, Laurie, WEI LIU, JUNG, David K

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DERIVADOS DE AZOXOINDOL COMO INHIBIDORES DE TRK PROTEINA QUINASA PARA EL TRATAMIENTO DE CANCER Y DOLOR CRONICO von WOOD, EDGAR, R. III, LACKEY, KAREN, E

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Discovery and in vitro Evaluation of Potent Kinase Inhibitors: Pyrido[1′,2′:1,5]pyrazolo[3,4-d]pyrimidines von Alberti, Michael J., Auten, Elizabeth P., Lackey, Karen E., McDonald, Octerloney B., Wood, Edgar R., Preugschat, Frank, Cutler, Geoffrey J., Kane-Carson, Laurie, Liu, Wei, Jung, David K.

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DERIVADOS DE QUINAZOLINA Y PIRIDOPIRIMIDINA von COCKERILL, GEORGE STUART, LACKEY, KAREN E, GUNTRIP, STEPHEN B, SMITH, KATHRYN J, CARTER, MALCOLM CLIVE

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ΠΑΡΑΓΩΓΑ ΚΙΝΑΖΟΛΙΝΗΣ ΚΑΙ ΠΥΡΙΔΟΠΥΡΙΜΙΔΙΝΗΣ von CARTER MALCOME CLIVE, COCKERILL GEORGE STUART, LACKEY KAREN E, SMITH KATHRYN J, GUNTRIP STEPHEN B

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HETEROCYCLIC COMPOUNDS von LACKEY KAREN E, COCKERILL GEORGE S

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HETEROCYCLIC COMPOUNDS von LACKEY KAREN E, COCKERILL GEORGE S

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AZAOXOINDOL DERIVATE ALS TRK PROTEIN KINASE HEMMSTOFFE ZUR BEHANDLUNG VON KREBS UND CHRONISCHEM SCHMERZ von WOOD, EDGAR, R. III, LACKEY, KAREN, E

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AZAOXOINDOLE DERIVATIVES AS Trk PROTEIN KINASE INHIBITORS FOR THE TREATMENT OF CANCER AND CHRONIC PAIN von WOOD, EDGAR, R. III, LACKEY, KAREN, E

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Anilinoquinazaolines as protein tyrosine kianse inhibitors von LACKEY KAREN E, COCKERILL GEORGE S

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Chemical compounds von LACKEY KAREN E, WOOD EDGAR R.III

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